FI57594C - Foerfarande foer framstaellning av antiallergiskt verksamma n-(bentstiazol-2-yl)-oxamidsyra-derivat - Google Patents
Foerfarande foer framstaellning av antiallergiskt verksamma n-(bentstiazol-2-yl)-oxamidsyra-derivat Download PDFInfo
- Publication number
- FI57594C FI57594C FI773738A FI773738A FI57594C FI 57594 C FI57594 C FI 57594C FI 773738 A FI773738 A FI 773738A FI 773738 A FI773738 A FI 773738A FI 57594 C FI57594 C FI 57594C
- Authority
- FI
- Finland
- Prior art keywords
- melting point
- mol
- methoxy
- ethyl ester
- benzthiazol
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
- C07D317/62—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring
- C07D317/66—Nitrogen atoms not forming part of a nitro radical
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pulmonology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Immunology (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19762656468 DE2656468A1 (de) | 1976-12-14 | 1976-12-14 | N-(benzthiazol-2-yl)-oxamidsaeure- derivate und verfahren zu ihrer herstellung |
| DE2656468 | 1976-12-14 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| FI773738A FI773738A (fi) | 1978-06-15 |
| FI57594B FI57594B (fi) | 1980-05-30 |
| FI57594C true FI57594C (fi) | 1980-09-10 |
Family
ID=5995427
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI773738A FI57594C (fi) | 1976-12-14 | 1977-12-12 | Foerfarande foer framstaellning av antiallergiskt verksamma n-(bentstiazol-2-yl)-oxamidsyra-derivat |
Country Status (17)
| Country | Link |
|---|---|
| JP (1) | JPS5377058A (xx) |
| AR (1) | AR216496A1 (xx) |
| AT (1) | AT360523B (xx) |
| AU (1) | AU510730B2 (xx) |
| BE (1) | BE861794A (xx) |
| CS (1) | CS203179B2 (xx) |
| DD (1) | DD133329A5 (xx) |
| DE (1) | DE2656468A1 (xx) |
| ES (1) | ES465034A1 (xx) |
| FI (1) | FI57594C (xx) |
| FR (1) | FR2374317A1 (xx) |
| GB (1) | GB1538822A (xx) |
| HU (1) | HU175340B (xx) |
| NL (1) | NL7713580A (xx) |
| SE (1) | SE7714074L (xx) |
| SU (1) | SU680647A3 (xx) |
| ZA (1) | ZA777236B (xx) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2676775A (en) * | 1949-10-24 | 1954-04-27 | Gustav O Schulz | Electric flatiron cord holder |
| DE3017976A1 (de) * | 1980-05-10 | 1981-11-19 | Dr. Karl Thomae Gmbh, 7950 Biberach | Substituierte 2-amino-5-halogen-benzothiazole, verfahen zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
| US4321372A (en) | 1980-06-16 | 1982-03-23 | Pfizer Inc. | Antiulcer thiazol-2-ylcarbamoyl-carboxylic acids, esters and amides |
| DE3027527A1 (de) | 1980-07-19 | 1982-02-18 | Basf Ag, 6700 Ludwigshafen | Neue oxamidsaeure-derivate, verfahren zu ihrer herstellung und diese enthaltende therapeutische mittel |
| GB2090826B (en) * | 1981-01-09 | 1985-06-12 | Usv Pharma Corp | New heterocyclic compounds useful as anti-allergie agents |
| DE3135250A1 (de) * | 1981-09-05 | 1983-03-17 | Basf Ag, 6700 Ludwigshafen | Tricyclische thiazolyloxamate, verfahren zu ihrer herstellung und diese enthaltende therapeutische mittel |
| US4826860A (en) * | 1987-03-16 | 1989-05-02 | Warner-Lambert Company | Substituted 2-aminobenzothiazoles and derivatives useful as cerebrovascular agents |
| FI91859C (fi) * | 1987-06-17 | 1994-08-25 | Eisai Co Ltd | Analogiamenetelmä antiallergisena aineena aktiivisen bentsotiatsolijohdannaisen valmistamiseksi |
| MXPA02012596A (es) * | 2000-06-21 | 2003-04-10 | Hoffmann La Roche | Derivados de benzotiazol. |
| US7087761B2 (en) | 2003-01-07 | 2006-08-08 | Hoffmann-La Roche Inc. | Cyclization process for substituted benzothiazole derivatives |
| JP4668265B2 (ja) | 2004-05-24 | 2011-04-13 | エフ．ホフマン−ラ ロシュ アーゲー | ４−ヒドロキシ−４−メチル−ピペリジン−１−カルボン酸（４−メトキシ−７−モルホリン−４−イル−ベンゾチアゾール−２−イル）−アミド |
| ATE400557T1 (de) | 2004-11-05 | 2008-07-15 | Hoffmann La Roche | Verfahren zur herstellung von isonikotinsäurederivaten |
| MX2007011483A (es) | 2005-03-23 | 2007-10-12 | Hoffmann La Roche | Derivados de acetilenil-pirazolo-pirimidina como antagonistas de glutamato metabotropico 2. |
| CA2623721C (en) | 2005-09-27 | 2014-05-13 | F. Hoffmann-La Roche Ag | Oxadiazolyl pyrazolo-pyrimidines as mglur2 antagonists |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4150140A (en) * | 1976-12-23 | 1979-04-17 | The Upjohn Company | Benzothiazolyl oxanic acids, esters and salts |
-
1976
- 1976-12-14 DE DE19762656468 patent/DE2656468A1/de not_active Withdrawn
-
1977
- 1977-12-03 HU HU77BO1695A patent/HU175340B/hu unknown
- 1977-12-05 ZA ZA00777236A patent/ZA777236B/xx unknown
- 1977-12-07 CS CS778173A patent/CS203179B2/cs unknown
- 1977-12-07 AR AR270289A patent/AR216496A1/es active
- 1977-12-07 SU SU772550552A patent/SU680647A3/ru active
- 1977-12-07 GB GB50911/77A patent/GB1538822A/en not_active Expired
- 1977-12-08 DD DD7700202483A patent/DD133329A5/xx unknown
- 1977-12-08 AU AU31377/77A patent/AU510730B2/en not_active Expired
- 1977-12-08 NL NL7713580A patent/NL7713580A/xx not_active Application Discontinuation
- 1977-12-12 SE SE7714074A patent/SE7714074L/xx not_active Application Discontinuation
- 1977-12-12 FI FI773738A patent/FI57594C/fi not_active IP Right Cessation
- 1977-12-13 FR FR7737467A patent/FR2374317A1/fr active Granted
- 1977-12-13 BE BE183407A patent/BE861794A/xx unknown
- 1977-12-13 AT AT890777A patent/AT360523B/de not_active IP Right Cessation
- 1977-12-14 JP JP15041777A patent/JPS5377058A/ja active Pending
- 1977-12-14 ES ES465034A patent/ES465034A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| FI773738A (fi) | 1978-06-15 |
| FR2374317A1 (fr) | 1978-07-13 |
| AR216496A1 (es) | 1979-12-28 |
| NL7713580A (nl) | 1978-06-16 |
| DE2656468A1 (de) | 1978-06-15 |
| FI57594B (fi) | 1980-05-30 |
| BE861794A (fr) | 1978-06-13 |
| CS203179B2 (en) | 1981-02-27 |
| AT360523B (de) | 1981-01-12 |
| SU680647A3 (ru) | 1979-08-15 |
| AU510730B2 (en) | 1980-07-10 |
| JPS5377058A (en) | 1978-07-08 |
| ZA777236B (en) | 1978-11-29 |
| ES465034A1 (es) | 1978-09-01 |
| SE7714074L (sv) | 1978-06-15 |
| GB1538822A (en) | 1979-01-24 |
| DD133329A5 (de) | 1978-12-27 |
| ATA890777A (de) | 1980-06-15 |
| AU3137777A (en) | 1979-06-14 |
| HU175340B (hu) | 1980-07-28 |
| FR2374317B1 (xx) | 1980-11-07 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| FI57594C (fi) | Foerfarande foer framstaellning av antiallergiskt verksamma n-(bentstiazol-2-yl)-oxamidsyra-derivat | |
| CA1102802A (en) | Benzothiazine derivatives | |
| FI91063B (fi) | Menetelmä kinoloniyhdisteiden valmistamiseksi | |
| CZ2000714A3 (cs) | 5-Alkyl-2-arylaminofenyloctové kyseliny a jejich deriváty, způsob jejich přípravy a farmaceutické prostředky, které je obsahují | |
| US5223513A (en) | Quinoline derivatives, their production and use | |
| US3455924A (en) | Dianisylimidazoles | |
| JPH09301958A (ja) | 新規ピリミジン化合物及び抗ロタウイルス剤 | |
| US4572910A (en) | Triazolo[1,5-c]pyrimidines substituted by nitrogen-containing heterocyclic rings | |
| NO794135L (no) | Substituerte 4(3h)-kinazolinoner, fremgangsmaate ved fremstilling og anvendelse av disse | |
| JPH0471914B2 (xx) | ||
| US3538086A (en) | 4-oxo-4h-pyrimido 2,1-b benzothiazoles | |
| OZEKI et al. | Studies on antiallergy agents. III. Synthesis of 2-anilino-1, 6-dihydro-6-oxo-5-pyrimidinecarboxylic acids and related compounds | |
| Zinnes et al. | 1, 2-Benzothiazines. 6. 3-Carbamoyl-4-hydroxy-2H-1, 2-benzothiazine 1, 1-dioxides as antiinflammatory agents | |
| US3726875A (en) | 1,3(2h,4h)-dioxoisoquinoline-4-carboxylate esters and process therefor | |
| EP0102175A1 (en) | 5-Oxo-5H-(1)benzopyrano(2,3-b)pyridine derivatives, their production and use | |
| NZ250458A (en) | 3-phenyl-benzofuran-2-yl- (and indol-2-yl-) acetamide, -propanamide and -urea derivatives; their preparation, intermediates and pharmaceutical compositions | |
| US4968708A (en) | Imidazo[2,1-B]benzothiazole compounds and antiulcer compositions containing the same | |
| US3944581A (en) | 5-Substituted-2,4-diphenylpyrimidines | |
| FI67706C (fi) | Foerfarande foer framstaellning av terapeutiskt anvaendbara n-5-tetrazolyl)-1-oxo-1h-tiazolo(3,2-a)pyrimidin-2-karboxyl atr | |
| US4254118A (en) | 1-Oxo-5H-pyrimido[2,1-c][1,4]benzthiazine-2-carboxylic acid esters | |
| EP0041630B1 (en) | New 3h-naphtho(1,2-d)imidazoles, the process for preparing them, the compounds for use as antiinflammatory agents and compositions containing them | |
| Bajaj et al. | Synthesis and psychotropic evaluation of some new N-substitutedbenzothia/oxazepinylphenothiazines | |
| US3303191A (en) | Novel 4-ketodihydro-2, 1-benzothiazine-2, 2-dioxides | |
| EP0397169B1 (en) | Novel benzothiazole derivatives | |
| JPH04273877A (ja) | 新規なイミダゾール誘導体 |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM | Patent lapsed |
Owner name: BOEHRINGER MANNHEIM GMBH |