GB1538822A - N-(benzthiazol-2-yl)-oxamic acid derivatives and the preparation thereof - Google Patents
N-(benzthiazol-2-yl)-oxamic acid derivatives and the preparation thereofInfo
- Publication number
- GB1538822A GB1538822A GB50911/77A GB5091177A GB1538822A GB 1538822 A GB1538822 A GB 1538822A GB 50911/77 A GB50911/77 A GB 50911/77A GB 5091177 A GB5091177 A GB 5091177A GB 1538822 A GB1538822 A GB 1538822A
- Authority
- GB
- United Kingdom
- Prior art keywords
- benzthiazol
- preparation
- acid derivatives
- oxamic acid
- oxamic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
- C07D317/62—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring
- C07D317/66—Nitrogen atoms not forming part of a nitro radical
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pulmonology (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19762656468 DE2656468A1 (en) | 1976-12-14 | 1976-12-14 | N- (BENZTHIAZOL-2-YL) -OXAMID ACID DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1538822A true GB1538822A (en) | 1979-01-24 |
Family
ID=5995427
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB50911/77A Expired GB1538822A (en) | 1976-12-14 | 1977-12-07 | N-(benzthiazol-2-yl)-oxamic acid derivatives and the preparation thereof |
Country Status (17)
| Country | Link |
|---|---|
| JP (1) | JPS5377058A (en) |
| AR (1) | AR216496A1 (en) |
| AT (1) | AT360523B (en) |
| AU (1) | AU510730B2 (en) |
| BE (1) | BE861794A (en) |
| CS (1) | CS203179B2 (en) |
| DD (1) | DD133329A5 (en) |
| DE (1) | DE2656468A1 (en) |
| ES (1) | ES465034A1 (en) |
| FI (1) | FI57594C (en) |
| FR (1) | FR2374317A1 (en) |
| GB (1) | GB1538822A (en) |
| HU (1) | HU175340B (en) |
| NL (1) | NL7713580A (en) |
| SE (1) | SE7714074L (en) |
| SU (1) | SU680647A3 (en) |
| ZA (1) | ZA777236B (en) |
Cited By (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4321372A (en) | 1980-06-16 | 1982-03-23 | Pfizer Inc. | Antiulcer thiazol-2-ylcarbamoyl-carboxylic acids, esters and amides |
| FR2497805A1 (en) * | 1981-01-09 | 1982-07-16 | Usv Pharma Corp | NOVEL HETEROCYCLIC COMPOUNDS USEFUL AS ANTIALLERGIC AGENTS |
| US4407810A (en) | 1980-07-19 | 1983-10-04 | Basf Aktiengesellschaft | Thiazol-2-yl-oxamic acid derivatives, and therapeutic agents containing these compounds |
| EP0295656A1 (en) * | 1987-06-17 | 1988-12-21 | Eisai Co., Ltd. | Benzothiazole derivative, its use, and pharmaceutical compositions comprising it |
| WO2001097786A2 (en) * | 2000-06-21 | 2001-12-27 | F. Hoffmann-La Roche Ag | Benzothiazole derivatives |
| US7087761B2 (en) | 2003-01-07 | 2006-08-08 | Hoffmann-La Roche Inc. | Cyclization process for substituted benzothiazole derivatives |
| US7238808B2 (en) | 2005-03-23 | 2007-07-03 | Hoffmann-La Roche Inc. | Acetylenyl-pyrazolo-pyrimidine derivatives |
| US7368446B2 (en) | 2004-05-24 | 2008-05-06 | Hoffmann-La Roche Inc. | 4-hydroxy-4-methyl-piperidine-1-carboxylic acid (4-methoxy-7-morpholin-4-yl-benzothiazol-2-yl)-amide |
| US7459563B2 (en) | 2004-11-05 | 2008-12-02 | Hoffmann-La Roche Inc. | Process for the preparation of isonicotinic acid derivatives |
| US7504404B2 (en) | 2005-09-27 | 2009-03-17 | Hoffmann-La Roche Inc. | Compounds as metabotropic glutamate receptor antagonists |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2676775A (en) * | 1949-10-24 | 1954-04-27 | Gustav O Schulz | Electric flatiron cord holder |
| DE3017976A1 (en) * | 1980-05-10 | 1981-11-19 | Dr. Karl Thomae Gmbh, 7950 Biberach | SUBSTITUTED 2-AMINO-5-HALOGEN-BENZOTHIAZOLES, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THESE COMPOUNDS |
| DE3135250A1 (en) * | 1981-09-05 | 1983-03-17 | Basf Ag, 6700 Ludwigshafen | TRICYCLIC THIAZOLYLOXAMATES, METHOD FOR THE PRODUCTION THEREOF AND THERAPEUTIC AGENTS CONTAINING THEM |
| US4826860A (en) * | 1987-03-16 | 1989-05-02 | Warner-Lambert Company | Substituted 2-aminobenzothiazoles and derivatives useful as cerebrovascular agents |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4150140A (en) * | 1976-12-23 | 1979-04-17 | The Upjohn Company | Benzothiazolyl oxanic acids, esters and salts |
-
1976
- 1976-12-14 DE DE19762656468 patent/DE2656468A1/en not_active Withdrawn
-
1977
- 1977-12-03 HU HU77BO1695A patent/HU175340B/en unknown
- 1977-12-05 ZA ZA00777236A patent/ZA777236B/en unknown
- 1977-12-07 GB GB50911/77A patent/GB1538822A/en not_active Expired
- 1977-12-07 CS CS778173A patent/CS203179B2/en unknown
- 1977-12-07 SU SU772550552A patent/SU680647A3/en active
- 1977-12-07 AR AR270289A patent/AR216496A1/en active
- 1977-12-08 DD DD7700202483A patent/DD133329A5/en unknown
- 1977-12-08 NL NL7713580A patent/NL7713580A/en not_active Application Discontinuation
- 1977-12-08 AU AU31377/77A patent/AU510730B2/en not_active Expired
- 1977-12-12 SE SE7714074A patent/SE7714074L/en not_active Application Discontinuation
- 1977-12-12 FI FI773738A patent/FI57594C/en not_active IP Right Cessation
- 1977-12-13 AT AT890777A patent/AT360523B/en not_active IP Right Cessation
- 1977-12-13 BE BE183407A patent/BE861794A/en unknown
- 1977-12-13 FR FR7737467A patent/FR2374317A1/en active Granted
- 1977-12-14 JP JP15041777A patent/JPS5377058A/en active Pending
- 1977-12-14 ES ES465034A patent/ES465034A1/en not_active Expired
Cited By (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4321372A (en) | 1980-06-16 | 1982-03-23 | Pfizer Inc. | Antiulcer thiazol-2-ylcarbamoyl-carboxylic acids, esters and amides |
| US4407810A (en) | 1980-07-19 | 1983-10-04 | Basf Aktiengesellschaft | Thiazol-2-yl-oxamic acid derivatives, and therapeutic agents containing these compounds |
| FR2497805A1 (en) * | 1981-01-09 | 1982-07-16 | Usv Pharma Corp | NOVEL HETEROCYCLIC COMPOUNDS USEFUL AS ANTIALLERGIC AGENTS |
| EP0295656A1 (en) * | 1987-06-17 | 1988-12-21 | Eisai Co., Ltd. | Benzothiazole derivative, its use, and pharmaceutical compositions comprising it |
| US6521754B2 (en) | 2000-06-21 | 2003-02-18 | Hoffman-La Roche Inc. | Benzothiazole derivatives with activity as adenosine receptor ligands |
| WO2001097786A3 (en) * | 2000-06-21 | 2002-12-12 | Hoffmann La Roche | Benzothiazole derivatives |
| US6835732B2 (en) | 2000-06-21 | 2004-12-28 | Hoffman-La Roche Inc. | Benzothiazole derivatives with activity as adenosine receptor ligands |
| US6963000B2 (en) | 2000-06-21 | 2005-11-08 | Hoffman-La Roche Inc. | Benzothiazole derivatives with activity as adenosine receptor ligands |
| WO2001097786A2 (en) * | 2000-06-21 | 2001-12-27 | F. Hoffmann-La Roche Ag | Benzothiazole derivatives |
| US7317007B2 (en) | 2000-06-21 | 2008-01-08 | Hoffmann-La Roche Inc. | Benzothiazole derivatives with activity as adenosine receptor ligands |
| US7087761B2 (en) | 2003-01-07 | 2006-08-08 | Hoffmann-La Roche Inc. | Cyclization process for substituted benzothiazole derivatives |
| US7368446B2 (en) | 2004-05-24 | 2008-05-06 | Hoffmann-La Roche Inc. | 4-hydroxy-4-methyl-piperidine-1-carboxylic acid (4-methoxy-7-morpholin-4-yl-benzothiazol-2-yl)-amide |
| US7459563B2 (en) | 2004-11-05 | 2008-12-02 | Hoffmann-La Roche Inc. | Process for the preparation of isonicotinic acid derivatives |
| US7238808B2 (en) | 2005-03-23 | 2007-07-03 | Hoffmann-La Roche Inc. | Acetylenyl-pyrazolo-pyrimidine derivatives |
| US7446113B2 (en) | 2005-03-23 | 2008-11-04 | Hoffman-La Roche Inc. | Acetylenyl-pyrazolo-pyrimidine derivatives |
| US7718661B2 (en) | 2005-03-23 | 2010-05-18 | Hoffmann-La Roche Inc. | Acetylenyl-pyrazolo-pyrimidine derivatives |
| US8063048B2 (en) | 2005-03-23 | 2011-11-22 | Hoffmann-La Roche Inc. | Acetylenyl-pyrazolo-pyrimidine derivatives |
| US7504404B2 (en) | 2005-09-27 | 2009-03-17 | Hoffmann-La Roche Inc. | Compounds as metabotropic glutamate receptor antagonists |
| US8093263B2 (en) | 2005-09-27 | 2012-01-10 | Hoffmann-La Roche Inc. | Substituted pyrazolo [1,5-a] pyrimidines as metabotropic glutamate antagonists |
| US8349844B2 (en) | 2005-09-27 | 2013-01-08 | Hoffmann-La Roche Inc. | Substituted pyrazolo [1,5-A] pyrimidines as metabotropic glutamate antagonists |
Also Published As
| Publication number | Publication date |
|---|---|
| ZA777236B (en) | 1978-11-29 |
| AR216496A1 (en) | 1979-12-28 |
| FR2374317B1 (en) | 1980-11-07 |
| AT360523B (en) | 1981-01-12 |
| CS203179B2 (en) | 1981-02-27 |
| FI773738A (en) | 1978-06-15 |
| FI57594C (en) | 1980-09-10 |
| ES465034A1 (en) | 1978-09-01 |
| DE2656468A1 (en) | 1978-06-15 |
| DD133329A5 (en) | 1978-12-27 |
| BE861794A (en) | 1978-06-13 |
| FI57594B (en) | 1980-05-30 |
| JPS5377058A (en) | 1978-07-08 |
| AU510730B2 (en) | 1980-07-10 |
| AU3137777A (en) | 1979-06-14 |
| ATA890777A (en) | 1980-06-15 |
| FR2374317A1 (en) | 1978-07-13 |
| HU175340B (en) | 1980-07-28 |
| NL7713580A (en) | 1978-06-16 |
| SE7714074L (en) | 1978-06-15 |
| SU680647A3 (en) | 1979-08-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed |