FI57104C - Foerfarande foer framstaellning av befruktningshindrande nya s-triatsolo(5,1-a)isokinolinderivat - Google Patents

Foerfarande foer framstaellning av befruktningshindrande nya s-triatsolo(5,1-a)isokinolinderivat Download PDF

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Publication number
FI57104C
FI57104C FI1591/74A FI159174A FI57104C FI 57104 C FI57104 C FI 57104C FI 1591/74 A FI1591/74 A FI 1591/74A FI 159174 A FI159174 A FI 159174A FI 57104 C FI57104 C FI 57104C
Authority
FI
Finland
Prior art keywords
formula
compound
group
phenyl
dihydro
Prior art date
Application number
FI1591/74A
Other languages
English (en)
Finnish (fi)
Other versions
FI159174A (es
FI57104B (fi
Inventor
Sale Amedeo Omodei
Pietro Consonni
Leonard J Lerner
Original Assignee
Lepetit Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB2516373A external-priority patent/GB1477302A/en
Priority claimed from GB3978973A external-priority patent/GB1477303A/en
Application filed by Lepetit Spa filed Critical Lepetit Spa
Publication of FI159174A publication Critical patent/FI159174A/fi
Publication of FI57104B publication Critical patent/FI57104B/fi
Application granted granted Critical
Publication of FI57104C publication Critical patent/FI57104C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44—Iso-indoles; Hydrogenated iso-indoles
    • C07D209/46—Iso-indoles; Hydrogenated iso-indoles with an oxygen atom in position 1
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C07D217/24—Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI1591/74A 1973-05-25 1974-05-24 Foerfarande foer framstaellning av befruktningshindrande nya s-triatsolo(5,1-a)isokinolinderivat FI57104C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB2516373A GB1477302A (en) 1973-05-25 1973-05-25 Triazolo-isoindole and triazolo-isoquinoline derivatives and their manufacture and uses
GB2516373 1973-05-25
GB3978973 1973-08-22
GB3978973A GB1477303A (en) 1973-08-22 1973-08-22 Pharmaceutical compositions

Publications (3)

Publication Number Publication Date
FI159174A FI159174A (es) 1974-11-26
FI57104B FI57104B (fi) 1980-02-29
FI57104C true FI57104C (fi) 1980-06-10

Family

ID=26257537

Family Applications (1)

Application Number Title Priority Date Filing Date
FI1591/74A FI57104C (fi) 1973-05-25 1974-05-24 Foerfarande foer framstaellning av befruktningshindrande nya s-triatsolo(5,1-a)isokinolinderivat

Country Status (24)

Country Link
US (2) US3895113A (es)
JP (1) JPS5315078B2 (es)
AR (2) AR208510A1 (es)
AT (1) AT334371B (es)
CA (2) CA1044237A (es)
CH (2) CH603166A5 (es)
DD (1) DD111077A5 (es)
DE (3) DE2424671C3 (es)
DK (1) DK151807C (es)
ES (2) ES426664A1 (es)
FI (1) FI57104C (es)
FR (3) FR2241292B1 (es)
HK (1) HK8978A (es)
HU (1) HU168537B (es)
IE (1) IE41612B1 (es)
IL (1) IL44978A (es)
IN (3) IN142266B (es)
LU (1) LU70151A1 (es)
NL (2) NL159580B (es)
NO (1) NO142079C (es)
RO (2) RO66801A (es)
SE (2) SE419543B (es)
SU (1) SU591149A3 (es)
YU (1) YU41042B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4129567A (en) * 1976-08-06 1978-12-12 Pfizer Inc. Quaternary salts as hypoglycemic agents
DE2707272C2 (de) * 1977-02-19 1982-12-02 Gruppo Lepetit S.p.A., 20158 Milano 2-(p-Chlorphenyl)-s-triazolo [5,1-a] isochinolin
GR70248B (es) * 1978-10-30 1982-09-01 Lepetit Spa
NL7907633A (nl) * 1978-10-30 1980-05-02 Lepetit Spa Werkwijze voor het bereiden van 2-fenyl-s-triazolo/5,1- -alpha/isochinolinen en aldus bereide verbindingen bevattende farmaceutische preparaten.
US4758427A (en) * 1985-08-08 1988-07-19 Ciba-Geigy Corporation Enhanced absorption of psychoactive 2-aryl-pyrazolo quinolines as a solid molecular dispersion in polyvinylpyrrolidone
ES2094772T3 (es) * 1990-06-01 1997-02-01 Kyowa Hakko Kogyo Kk Derivados de imidazonaftiridinas.
SE9300127L (sv) * 1993-01-19 1994-07-20 Eyvind Langvad Tricyliska kondenserade 1,2,4-triazoloderivat användbara såsom antiinflammatoriska medel
TWI461426B (zh) * 2009-05-27 2014-11-21 Merck Sharp & Dohme （二氫）咪唑並異〔５，１－ａ〕喹啉類

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA884328A (en) * 1971-10-26 K. Reimlinger Hans S-triazolo(5,1-a)isoquinolines and derivatives thereof
CA883836A (en) * 1971-10-19 H. De Ruiter Ernest Selective hydrogenation of tri- and tetrazoloisquinolines
US2976146A (en) * 1958-11-28 1961-03-21 Eastman Kodak Co Novel cyan-forming couplers
GB1244501A (en) * 1968-03-09 1971-09-02 Aspro Nicholas Ltd Heterocyclic amines
US3758480A (en) * 1968-07-10 1973-09-11 Mallinckrodt Chemical Works S-triazolo(5,1-a)isoquinolines and derivatives thereof
AR204975A1 (es) * 1971-03-18 1976-03-31 Lepetit Spa Procedimiento para preparar 2-aminodihidro-isoquinolinas
US3775417A (en) * 1971-08-05 1973-11-27 Mallinckrodt Chemical Works Selective hydrogenation of tri-and tetrazoloisoquinolines

Also Published As

Publication number Publication date
CA1044237A (en) 1978-12-12
SU591149A3 (ru) 1978-01-30
SE434642B (sv) 1984-08-06
NO741894L (no) 1974-11-26
USRE30456E (en) 1980-12-23
AT334371B (de) 1976-01-10
AR212692A1 (es) 1978-09-15
FI159174A (es) 1974-11-26
FR2230369A1 (es) 1974-12-20
JPS5035195A (es) 1975-04-03
DK151807C (da) 1988-07-18
HK8978A (en) 1978-02-24
DD111077A5 (es) 1975-01-20
AR208510A1 (es) 1977-02-15
AU6881974A (en) 1975-11-13
CH603641A5 (es) 1978-08-31
DE2463023C2 (de) 1984-10-11
FR2272669B1 (es) 1978-07-21
ATA426174A (de) 1976-05-15
SE419543B (sv) 1981-08-10
CH603166A5 (es) 1978-08-15
FR2272669A1 (en) 1975-12-26
DK283274A (es) 1975-01-20
DK151807B (da) 1988-01-04
IE41612L (en) 1974-11-25
IL44978A0 (en) 1974-09-10
IL44978A (en) 1980-01-31
DE2424671A1 (de) 1974-12-12
FI57104B (fi) 1980-02-29
SE7710485L (sv) 1977-09-19
NO142079B (no) 1980-03-17
DE2424572A1 (de) 1974-12-12
DE2424671B2 (de) 1981-07-30
DE2424572C2 (de) 1983-07-21
RO66059A (ro) 1981-05-30
NL7406995A (es) 1974-11-27
YU41042B (en) 1986-10-31
FR2241292A1 (es) 1975-03-21
IE41612B1 (en) 1980-02-13
US3895113A (en) 1975-07-15
ES426664A1 (es) 1977-01-01
NL7801129A (nl) 1978-05-31
HU168537B (es) 1976-05-28
CA1024892A (en) 1978-01-24
DE2424671C3 (de) 1982-05-13
ES447548A1 (es) 1977-11-01
IN145039B (es) 1978-08-12
NO142079C (no) 1980-06-25
FR2230369B1 (es) 1978-06-30
JPS5315078B2 (es) 1978-05-22
LU70151A1 (es) 1974-10-09
YU141374A (en) 1983-01-21
IN145038B (es) 1978-08-12
FR2241292B1 (es) 1978-07-21
IN142266B (es) 1977-06-18
AU6881774A (en) 1975-11-13
RO66801A (fr) 1979-08-15
NL159580B (nl) 1979-03-15

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