FI111362B - Menetelmä terapeuttisesti käyttökelpoisten N-heteroaryyliamidijohdannaisten valmistamiseksi - Google Patents

Menetelmä terapeuttisesti käyttökelpoisten N-heteroaryyliamidijohdannaisten valmistamiseksi Download PDF

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FI111362B
FI111362B FI904537A FI904537A FI111362B FI 111362 B FI111362 B FI 111362B FI 904537 A FI904537 A FI 904537A FI 904537 A FI904537 A FI 904537A FI 111362 B FI111362 B FI 111362B
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Finland
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nmr
cdcl
title compound
chcl
acid amide
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FI904537A
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Finnish (fi)
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FI904537A0 (fi
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Ernest S Hamanaka
George Chang
Peter A Mccarthy
Thien Truong
Frederick J Walker
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Pfizer
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pyridine Compounds (AREA)
  • Furan Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Quinoline Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
  • Hydrogenated Pyridines (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
FI904537A 1989-09-15 1990-09-14 Menetelmä terapeuttisesti käyttökelpoisten N-heteroaryyliamidijohdannaisten valmistamiseksi FI111362B (fi)

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PCT/US1989/004033 WO1991004027A1 (en) 1989-09-15 1989-09-15 New n-aryl and n-heteroarylamide and urea derivatives as inhibitors of acyl coenzyme a: cholesterol acyl transferase (acat)
US8904033 1989-09-15

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AU6255390A (en) 1991-04-18
PL291471A1 (en) 1992-06-26
DE69018908T2 (de) 1995-08-24
FI904537A0 (fi) 1990-09-14
WO1991004027A1 (en) 1991-04-04
ES2071033T3 (es) 1995-06-16
DK0609960T3 (da) 1999-09-27
PL291470A1 (en) 1992-07-13
GR3029826T3 (en) 1999-06-30
CN1050183A (zh) 1991-03-27
HUT70027A (en) 1995-09-28
IL110324A0 (en) 1994-10-21
NO904022L (no) 1991-03-18
PT95310A (pt) 1991-05-22
DE69032981D1 (de) 1999-04-08
PL165370B1 (pl) 1994-12-30
NO904022D0 (no) 1990-09-14
ATE177082T1 (de) 1999-03-15
HU9302945D0 (en) 1993-12-28
IE66324B1 (en) 1995-12-27
EP0609960A1 (en) 1994-08-10
EP0418071B1 (en) 1995-04-26
ES2127878T3 (es) 1999-05-01
EP0609960B1 (en) 1999-03-03
CA2025301C (en) 2001-10-16
IL110321A0 (en) 1994-10-21
KR910006233A (ko) 1991-04-27
JPH03120243A (ja) 1991-05-22
PL291472A1 (en) 1992-07-13
ZA907346B (en) 1992-05-27
DD298092A5 (de) 1992-02-06
CA2025301A1 (en) 1991-03-16
IL95610A (en) 1994-12-29
MX22406A (es) 1994-01-31
EP0418071A3 (en) 1992-03-25
EP0418071A2 (en) 1991-03-20
DK0418071T3 (da) 1995-09-04
AU652345B2 (en) 1994-08-25
DE69018908D1 (de) 1995-06-01
IE903336A1 (en) 1991-04-10
KR930011303B1 (ko) 1993-11-29
NZ235323A (en) 1993-02-25
PL165357B1 (pl) 1994-12-30
IL95610A0 (en) 1991-06-30
DE69032981T2 (de) 1999-07-08
JPH0825974B2 (ja) 1996-03-13
EG19358A (en) 1994-12-30
ATE121730T1 (de) 1995-05-15
PT95310B (pt) 1997-06-30

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