FI107536B - Makrolidien fluorisokerijohdannaiset - Google Patents

Makrolidien fluorisokerijohdannaiset Download PDF

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Publication number
FI107536B
FI107536B FI944016A FI944016A FI107536B FI 107536 B FI107536 B FI 107536B FI 944016 A FI944016 A FI 944016A FI 944016 A FI944016 A FI 944016A FI 107536 B FI107536 B FI 107536B
Authority
FI
Finland
Prior art keywords
formula
compound
prepared
process according
ococh
Prior art date
Application number
FI944016A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI944016A (fi
FI944016A0 (fi
Inventor
Kevin Koch
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI944016A publication Critical patent/FI944016A/fi
Publication of FI944016A0 publication Critical patent/FI944016A0/fi
Application granted granted Critical
Publication of FI107536B publication Critical patent/FI107536B/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Immunology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
FI944016A 1992-03-02 1994-09-01 Makrolidien fluorisokerijohdannaiset FI107536B (fi)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US84480292A 1992-03-02 1992-03-02
US84480292 1992-03-02
US94723992A 1992-09-18 1992-09-18
US94723992 1992-09-18
PCT/US1993/000428 WO1993018049A1 (en) 1992-03-02 1993-01-27 Fluorosugar derivatives of macrolides
US9300428 1993-01-27

Publications (3)

Publication Number Publication Date
FI944016A FI944016A (fi) 1994-09-01
FI944016A0 FI944016A0 (fi) 1994-09-01
FI107536B true FI107536B (fi) 2001-08-31

Family

ID=27126528

Family Applications (1)

Application Number Title Priority Date Filing Date
FI944016A FI107536B (fi) 1992-03-02 1994-09-01 Makrolidien fluorisokerijohdannaiset

Country Status (6)

Country Link
US (1) US5612316A (ja)
EP (1) EP0629208A1 (ja)
JP (1) JP2564765B2 (ja)
CA (1) CA2132457C (ja)
FI (1) FI107536B (ja)
WO (1) WO1993018049A1 (ja)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1998024904A2 (en) 1996-12-02 1998-06-11 Magainin Pharmaceuticals Inc. Il-9 receptor variants, useful in treating and diagnosing atopic allergies including asthma and related disorders
US6441114B1 (en) 1999-06-11 2002-08-27 3M Innovative Properties Company Adhesives for use on fluorine-containing or polycarbonate surfaces
US7452692B2 (en) * 2002-02-13 2008-11-18 Teva Gyógyszergyár Zártkörüen Müködö Részvénytársaság Method for extracting a macrolide from biomatter
PL374059A1 (en) * 2002-02-13 2005-09-19 Teva Gyogyszergyar Reszvenytarsasag Method for extracting a macrolide from biomatter
US7160867B2 (en) 2003-05-16 2007-01-09 Isotechnika, Inc. Rapamycin carbohydrate derivatives
DE10330960B4 (de) * 2003-07-08 2005-09-08 Stockhausen Gmbh Wirkstoffdotierte absorbierende Polymerteilchen , Zusammensetzung beinhaltend Polykondensatmatrix und absorbierendes Polymer zur Freisetzung einer Wundheilsubstanz
CA2571710A1 (en) 2004-06-24 2006-11-02 Nicholas Valiante Small molecule immunopotentiators and assays for their detection
WO2006069333A1 (en) * 2004-12-22 2006-06-29 Teva Gyógyszergyár Zàrtköruen Muködo Rèszvènytàrsasàg Method of purifying macrolides
JP2007527434A (ja) * 2005-01-05 2007-09-27 テバ ジョジセルジャール ザ−トケルエン ムケド レ−スベニュタ−ルシャシャ−グ 非晶質タクロリマス及びその調製
US20080000834A1 (en) * 2006-03-15 2008-01-03 Ladislav Cvak Process for purifying Tacrolimus

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4894366A (en) * 1984-12-03 1990-01-16 Fujisawa Pharmaceutical Company, Ltd. Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same
JPH05504944A (ja) * 1989-08-18 1993-07-29 藤沢薬品工業株式会社 巨大環式化合物
IE904050A1 (en) * 1989-11-13 1991-05-22 Merck & Co Inc Aminomacrolides and derivatives having immunosuppressive¹activity
EP0466365A3 (en) * 1990-07-03 1992-04-15 Merck & Co. Inc. Novel immunosuppressant fermentation products of a microorganism
US5023262A (en) * 1990-08-14 1991-06-11 American Home Products Corporation Hydrogenated rapamycin derivatives

Also Published As

Publication number Publication date
CA2132457C (en) 1998-06-16
JPH07500351A (ja) 1995-01-12
FI944016A (fi) 1994-09-01
US5612316A (en) 1997-03-18
EP0629208A1 (en) 1994-12-21
JP2564765B2 (ja) 1996-12-18
FI944016A0 (fi) 1994-09-01
CA2132457A1 (en) 1993-09-16
WO1993018049A1 (en) 1993-09-16

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