ES8608537A1 - Procedimiento de preparacion de 17-(isociano-sulfonilmetileno)-esteroides, 17-(formamido-sulfonilmetileno)-esteroides - Google Patents

Procedimiento de preparacion de 17-(isociano-sulfonilmetileno)-esteroides, 17-(formamido-sulfonilmetileno)-esteroides

Info

Publication number
ES8608537A1
ES8608537A1 ES532029A ES532029A ES8608537A1 ES 8608537 A1 ES8608537 A1 ES 8608537A1 ES 532029 A ES532029 A ES 532029A ES 532029 A ES532029 A ES 532029A ES 8608537 A1 ES8608537 A1 ES 8608537A1
Authority
ES
Spain
Prior art keywords
steroids
sulfonylmethylene
preparation
isocyano
formamido
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES532029A
Other languages
English (en)
Spanish (es)
Other versions
ES532029A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Gist Brocades NV
Original Assignee
Gist Brocades NV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gist Brocades NV filed Critical Gist Brocades NV
Publication of ES8608537A1 publication Critical patent/ES8608537A1/es
Publication of ES532029A0 publication Critical patent/ES532029A0/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0038—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 with an androstane skeleton, including 18- or 19-substituted derivatives, 18-nor derivatives and also derivatives where position 17-beta is substituted by a carbon atom not directly bonded to a further carbon atom and not being part of an amide group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002—Carbocyclic rings fused
    • C07J53/004—3 membered carbocyclic rings
    • C07J53/005—3 membered carbocyclic rings in position 12
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ES532029A 1983-04-29 1984-04-28 Procedimiento de preparacion de 17-(isociano-sulfonilmetileno)-esteroides, 17-(formamido-sulfonilmetileno)-esteroides Expired ES8608537A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP83200616A EP0123734A1 (en) 1983-04-29 1983-04-29 17-(Isocyano-sulfonylmethylene)-steroids, 17-(formamido-sulfonylmethylene)-steroids and their preparation

Publications (2)

Publication Number Publication Date
ES8608537A1 true ES8608537A1 (es) 1986-07-16
ES532029A0 ES532029A0 (es) 1986-07-16

Family

ID=8190949

Family Applications (2)

Application Number Title Priority Date Filing Date
ES532029A Expired ES8608537A1 (es) 1983-04-29 1984-04-28 Procedimiento de preparacion de 17-(isociano-sulfonilmetileno)-esteroides, 17-(formamido-sulfonilmetileno)-esteroides
ES553609A Expired ES8800263A1 (es) 1983-04-29 1986-04-01 Procedimiento de preparacion de 17-(isociano-sulfonilmetileno)-esteroides

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES553609A Expired ES8800263A1 (es) 1983-04-29 1986-04-01 Procedimiento de preparacion de 17-(isociano-sulfonilmetileno)-esteroides

Country Status (17)

Country Link
US (1) US4647410A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
EP (2) EP0123734A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
JP (2) JPS59206399A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
KR (1) KR860001469B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AU (1) AU568643B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (1) CA1257249A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DE (1) DE3461381D1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DK (2) DK166545B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ES (2) ES8608537A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FI (1) FI82061C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GR (1) GR81997B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
HU (2) HU193207B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IE (1) IE57328B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IL (1) IL71658A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NO (1) NO167093C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NZ (1) NZ207985A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
PT (1) PT78503B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0123735A1 (en) * 1983-04-29 1984-11-07 Gist-Brocades N.V. New process for the preparation of 20-keto-delta-16-steroids and new intermediate compounds formed in this process
EP0336521B1 (en) * 1988-04-08 1992-04-01 Roussel-Uclaf 9-alpha-hydroxy-17-methylene steroids, process for their preparation and their use in the preparation of corticosteroids
HU226413B1 (en) * 1991-06-25 2008-11-28 Aventis Pharma Sa Novel 16-(nitro-substituted methyl)pregna-1,4-dien-3,20-dion derivatives and process for producing them
FR2681069B1 (fr) * 1991-09-06 1995-04-28 Roussel Uclaf Nouveau procede de preparation de l'hydrocortisone et nouveaux intermediaires.
FR2683530B1 (fr) * 1991-11-08 1994-01-21 Roussel Uclaf Nouveau procede de preparation de derives 20-oxo 17 alpha, 21-dihydroxyles du pregnane et nouveaux intermediaires.
EA009176B1 (ru) * 1995-12-11 2007-12-28 Дж.Д.Серл Энд Ко. Способ получения 7-альфа-карбоксил-9,11-эпоксистероидов и промежуточных продуктов, используемых для их получения, и общий способ эпоксидирования по олефиновым двойным связям
BR9714510A (pt) 1996-12-11 2000-11-28 Searle & Co Processo e preparo de esteróides de 9,11-époxi e intermediários úteis dos mesmos
US6887991B1 (en) 1996-12-11 2005-05-03 G. D. Searle & Company Processes for preparation of 9, 11-epoxy steroids and intermediates useful therein
EP1079859B1 (en) 1998-05-22 2010-07-14 The Board Of Trustees Of The Leland Stanford Junior University Bifunctional molecules and therapies based thereon
EP2341423A1 (en) 1999-11-02 2011-07-06 Canon Kabushiki Kaisha Print control method and apparatus
US7235655B2 (en) 2002-03-22 2007-06-26 Pharmacia & Upjohn Company Processes to prepare eplerenone
EP3827747A1 (en) 2005-04-28 2021-06-02 Otsuka Pharmaceutical Co., Ltd. Pharma-informatics system
EP1945240B1 (en) 2005-09-16 2016-12-28 Raptor Pharmaceutical Inc Compositions comprising receptor-associated protein (rap) variants specific for cr-containing proteins and uses thereof
PT2398500T (pt) 2009-02-20 2019-06-14 2 Bbb Medicines B V Sistema de entrega de medicamentos à base de glutationas
KR20180114970A (ko) 2009-05-06 2018-10-19 라보라토리 스킨 케어, 인크. 활성제-칼슘 포스페이트 입자 복합체를 포함하는 피부 전달 조성물 및 이들을 이용하는 방법
CN105481924B (zh) * 2015-11-24 2017-08-15 浙江省诸暨合力化学对外贸易有限公司 一种黄体酮的制备方法
US20240368212A1 (en) * 2021-08-26 2024-11-07 Brandeis University Selective isonitrile inhibitors of cytochrome p450 subtypes

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7807631A (nl) * 1978-07-17 1980-01-21 Gist Brocades Nv Isocyanoderivaten en hun bereiding.
FR2462445A1 (fr) * 1979-07-31 1981-02-13 Roussel Uclaf Nouveaux derives 17-/(hydroxymethyl) (formamido) methylene/steroides, leur procede de preparation et leur application a l'introduction de la chaine laterale hydroxyacetyle
FR2486947A1 (fr) * 1980-07-15 1982-01-22 Roussel Uclaf Nouveaux derives steroides 20-isonitriles 17(20) insatures, leur procede de preparation et leur application a la preparation des steroides 17a-hydroxy 20-ceto

Also Published As

Publication number Publication date
EP0123734A1 (en) 1984-11-07
HU193207B (en) 1987-08-28
KR860001469B1 (ko) 1986-09-26
HU194277B (en) 1988-01-28
ES553609A0 (es) 1987-11-01
DK212184A (da) 1984-10-30
GR81997B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1984-12-12
DK22192D0 (da) 1992-02-21
EP0124934A1 (en) 1984-11-14
AU2713384A (en) 1984-11-01
PT78503A (en) 1984-05-01
DK166831B1 (da) 1993-07-19
PT78503B (en) 1986-05-20
JPH0717673B2 (ja) 1995-03-01
DK166545B1 (da) 1993-06-07
US4647410A (en) 1987-03-03
IL71658A (en) 1988-03-31
ES532029A0 (es) 1986-07-16
JPS59206399A (ja) 1984-11-22
JPH0559097A (ja) 1993-03-09
ES8800263A1 (es) 1987-11-01
NO841700L (no) 1984-10-30
AU568643B2 (en) 1988-01-07
IE57328B1 (en) 1992-07-29
DE3461381D1 (en) 1987-01-08
FI841679A7 (fi) 1984-10-30
NZ207985A (en) 1986-11-12
KR840008461A (ko) 1984-12-15
FI82061B (fi) 1990-09-28
JPH053478B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1993-01-14
FI82061C (fi) 1991-01-10
NO167093B (no) 1991-06-24
DK22192A (da) 1992-02-21
IL71658A0 (en) 1984-07-31
IE841038L (en) 1984-10-29
FI841679A0 (fi) 1984-04-27
DK212184D0 (da) 1984-04-27
EP0124934B1 (en) 1986-11-20
HUT34220A (en) 1985-02-28
NO167093C (no) 1991-10-02
CA1257249A (en) 1989-07-11

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 20020506