DK22192A - 17-(formamido-sulfonylmethylen)-steroider og fremgangsmaade til deres fremstilling. - Google Patents

17-(formamido-sulfonylmethylen)-steroider og fremgangsmaade til deres fremstilling. Download PDF

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Publication number
DK22192A
DK22192A DK022192A DK22192A DK22192A DK 22192 A DK22192 A DK 22192A DK 022192 A DK022192 A DK 022192A DK 22192 A DK22192 A DK 22192A DK 22192 A DK22192 A DK 22192A
Authority
DK
Denmark
Prior art keywords
sulphonylmethyl
formamido
steroids
procedures
preparation
Prior art date
Application number
DK022192A
Other languages
English (en)
Other versions
DK22192D0 (da
DK166831B1 (da
Inventor
Albert Mattheus Van Leusen
Adiaan Marinus Van Leusen
Original Assignee
Gist Brocades Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gist Brocades Nv filed Critical Gist Brocades Nv
Publication of DK22192D0 publication Critical patent/DK22192D0/da
Publication of DK22192A publication Critical patent/DK22192A/da
Application granted granted Critical
Publication of DK166831B1 publication Critical patent/DK166831B1/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0038—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 with an androstane skeleton, including 18- or 19-substituted derivatives, 18-nor derivatives and also derivatives where position 17-beta is substituted by a carbon atom not directly bonded to a further carbon atom and not being part of an amide group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002—Carbocyclic rings fused
    • C07J53/004—3 membered carbocyclic rings
    • C07J53/005—3 membered carbocyclic rings in position 12
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK022192A 1983-04-29 1992-02-21 17-(formamido-sulfonylmethylen)-steroider og fremgangsmaade til deres fremstilling DK166831B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP83200616 1983-04-29
EP83200616A EP0123734A1 (en) 1983-04-29 1983-04-29 17-(Isocyano-sulfonylmethylene)-steroids, 17-(formamido-sulfonylmethylene)-steroids and their preparation

Publications (3)

Publication Number Publication Date
DK22192D0 DK22192D0 (da) 1992-02-21
DK22192A true DK22192A (da) 1992-02-21
DK166831B1 DK166831B1 (da) 1993-07-19

Family

ID=8190949

Family Applications (2)

Application Number Title Priority Date Filing Date
DK212184A DK166545B1 (da) 1983-04-29 1984-04-27 17-(isocyano-sulfonylmethylen)-steroider og fremgangsmaade til deres fremstilling
DK022192A DK166831B1 (da) 1983-04-29 1992-02-21 17-(formamido-sulfonylmethylen)-steroider og fremgangsmaade til deres fremstilling

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK212184A DK166545B1 (da) 1983-04-29 1984-04-27 17-(isocyano-sulfonylmethylen)-steroider og fremgangsmaade til deres fremstilling

Country Status (17)

Country Link
US (1) US4647410A (da)
EP (2) EP0123734A1 (da)
JP (2) JPS59206399A (da)
KR (1) KR860001469B1 (da)
AU (1) AU568643B2 (da)
CA (1) CA1257249A (da)
DE (1) DE3461381D1 (da)
DK (2) DK166545B1 (da)
ES (2) ES8608537A1 (da)
FI (1) FI82061C (da)
GR (1) GR81997B (da)
HU (2) HU194277B (da)
IE (1) IE57328B1 (da)
IL (1) IL71658A (da)
NO (1) NO167093C (da)
NZ (1) NZ207985A (da)
PT (1) PT78503B (da)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0123735A1 (en) * 1983-04-29 1984-11-07 Gist-Brocades N.V. New process for the preparation of 20-keto-delta-16-steroids and new intermediate compounds formed in this process
AU618350B2 (en) * 1988-04-08 1991-12-19 Aventis Pharma S.A. 9-alpha-hydroxy-17-methylene steroids, process for their preparation and their use in the preparation of corticosteroids
HU226413B1 (en) * 1991-06-25 2008-11-28 Aventis Pharma Sa Novel 16-(nitro-substituted methyl)pregna-1,4-dien-3,20-dion derivatives and process for producing them
FR2681069B1 (fr) * 1991-09-06 1995-04-28 Roussel Uclaf Nouveau procede de preparation de l'hydrocortisone et nouveaux intermediaires.
FR2683530B1 (fr) * 1991-11-08 1994-01-21 Roussel Uclaf Nouveau procede de preparation de derives 20-oxo 17 alpha, 21-dihydroxyles du pregnane et nouveaux intermediaires.
CN100384866C (zh) 1995-12-11 2008-04-30 G·D·瑟尔公司 制备7α-羧基9,11-环氧甾族化合物的方法和其中使用的中间体以及烯双键环氧化作用的一般方法
PT944644E (pt) 1996-12-11 2003-02-28 Searle & Co Processos para a preparacao de esteroides 9,11-epoxi e intermediarios uteis para esse efeito
US6887991B1 (en) 1996-12-11 2005-05-03 G. D. Searle & Company Processes for preparation of 9, 11-epoxy steroids and intermediates useful therein
ATE473759T1 (de) 1998-05-22 2010-07-15 Univ Leland Stanford Junior Bifunktionelle moleküle sowie darauf basierende therapien.
EP1098266A3 (en) 1999-11-02 2003-01-22 Canon Kabushiki Kaisha Print control method and apparatus
US7235655B2 (en) 2002-03-22 2007-06-26 Pharmacia & Upjohn Company Processes to prepare eplerenone
EP2392258B1 (en) 2005-04-28 2014-10-08 Proteus Digital Health, Inc. Pharma-informatics system
US9062126B2 (en) 2005-09-16 2015-06-23 Raptor Pharmaceuticals Inc. Compositions comprising receptor-associated protein (RAP) variants specific for CR-containing proteins and uses thereof
PL3395372T3 (pl) 2009-02-20 2022-07-25 EnhanX Biopharm Inc. Układ do dostarczania leków na bazie glutationu
CN102458374A (zh) 2009-05-06 2012-05-16 实验室护肤股份有限公司 包含活性剂-磷酸钙颗粒复合物的皮肤递送组合物及其使用方法
CN105481924B (zh) * 2015-11-24 2017-08-15 浙江省诸暨合力化学对外贸易有限公司 一种黄体酮的制备方法
EP4392036A4 (en) * 2021-08-26 2026-03-11 Univ Brandeis SELECTIVE CYTOCHROME P450 SUBTYPE INHIBITORS BASED ON ISONITRILE

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7807631A (nl) * 1978-07-17 1980-01-21 Gist Brocades Nv Isocyanoderivaten en hun bereiding.
FR2462445A1 (fr) * 1979-07-31 1981-02-13 Roussel Uclaf Nouveaux derives 17-/(hydroxymethyl) (formamido) methylene/steroides, leur procede de preparation et leur application a l'introduction de la chaine laterale hydroxyacetyle
FR2486947A1 (fr) * 1980-07-15 1982-01-22 Roussel Uclaf Nouveaux derives steroides 20-isonitriles 17(20) insatures, leur procede de preparation et leur application a la preparation des steroides 17a-hydroxy 20-ceto

Also Published As

Publication number Publication date
IL71658A0 (en) 1984-07-31
HU193207B (en) 1987-08-28
FI841679A7 (fi) 1984-10-30
HU194277B (en) 1988-01-28
DK212184D0 (da) 1984-04-27
PT78503A (en) 1984-05-01
ES8608537A1 (es) 1986-07-16
JPH0717673B2 (ja) 1995-03-01
IE57328B1 (en) 1992-07-29
DK22192D0 (da) 1992-02-21
NZ207985A (en) 1986-11-12
DK166545B1 (da) 1993-06-07
CA1257249A (en) 1989-07-11
AU2713384A (en) 1984-11-01
AU568643B2 (en) 1988-01-07
JPH0559097A (ja) 1993-03-09
DK212184A (da) 1984-10-30
ES8800263A1 (es) 1987-11-01
HUT34220A (en) 1985-02-28
IL71658A (en) 1988-03-31
FI82061B (fi) 1990-09-28
JPH053478B2 (da) 1993-01-14
PT78503B (en) 1986-05-20
JPS59206399A (ja) 1984-11-22
ES553609A0 (es) 1987-11-01
KR840008461A (ko) 1984-12-15
IE841038L (en) 1984-10-29
EP0124934B1 (en) 1986-11-20
EP0124934A1 (en) 1984-11-14
NO167093B (no) 1991-06-24
NO167093C (no) 1991-10-02
FI841679A0 (fi) 1984-04-27
KR860001469B1 (ko) 1986-09-26
GR81997B (da) 1984-12-12
US4647410A (en) 1987-03-03
DE3461381D1 (en) 1987-01-08
ES532029A0 (es) 1986-07-16
DK166831B1 (da) 1993-07-19
EP0123734A1 (en) 1984-11-07
FI82061C (fi) 1991-01-10
NO841700L (no) 1984-10-30

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Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
PBP Patent lapsed