ES8103094A1 - Un procedimiento para la preparacion de 1,1-dioxido de acidopenicilanico y esteres del mismo - Google Patents

Un procedimiento para la preparacion de 1,1-dioxido de acidopenicilanico y esteres del mismo

Info

Publication number
ES8103094A1
ES8103094A1 ES489185A ES489185A ES8103094A1 ES 8103094 A1 ES8103094 A1 ES 8103094A1 ES 489185 A ES489185 A ES 489185A ES 489185 A ES489185 A ES 489185A ES 8103094 A1 ES8103094 A1 ES 8103094A1
Authority
ES
Spain
Prior art keywords
penicillanic acid
esters
dioxide
vivo
readily hydrolyzable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES489185A
Other languages
English (en)
Spanish (es)
Other versions
ES489185A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of ES489185A0 publication Critical patent/ES489185A0/es
Publication of ES8103094A1 publication Critical patent/ES8103094A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
ES489185A 1979-03-05 1980-03-04 Un procedimiento para la preparacion de 1,1-dioxido de acidopenicilanico y esteres del mismo Expired ES8103094A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1780879A 1979-03-05 1979-03-05
US1781079A 1979-03-05 1979-03-05

Publications (2)

Publication Number Publication Date
ES489185A0 ES489185A0 (es) 1981-02-16
ES8103094A1 true ES8103094A1 (es) 1981-02-16

Family

ID=26690337

Family Applications (1)

Application Number Title Priority Date Filing Date
ES489185A Expired ES8103094A1 (es) 1979-03-05 1980-03-04 Un procedimiento para la preparacion de 1,1-dioxido de acidopenicilanico y esteres del mismo

Country Status (36)

Country Link
KR (1) KR850001339B1 (fi)
AR (1) AR225031A1 (fi)
AT (1) AT366693B (fi)
AU (1) AU522572B2 (fi)
BG (1) BG33292A3 (fi)
CH (1) CH644608A5 (fi)
CS (1) CS215130B2 (fi)
DD (1) DD149367A5 (fi)
DE (1) DE3008257C2 (fi)
DK (2) DK159852C (fi)
EG (1) EG14437A (fi)
ES (1) ES8103094A1 (fi)
FI (1) FI70024C (fi)
FR (1) FR2450836B1 (fi)
GB (1) GB2045755B (fi)
GR (1) GR67234B (fi)
HK (1) HK66587A (fi)
HU (1) HU186304B (fi)
IE (1) IE49535B1 (fi)
IL (1) IL59515A (fi)
IN (1) IN153685B (fi)
IT (1) IT1130300B (fi)
KE (1) KE3464A (fi)
LU (1) LU82215A1 (fi)
MX (1) MX6032E (fi)
MY (1) MY8500319A (fi)
NL (1) NL180317C (fi)
NO (2) NO800618L (fi)
PL (1) PL125197B1 (fi)
PT (1) PT70897A (fi)
RO (1) RO80112A (fi)
SE (2) SE449103B (fi)
SG (1) SG55884G (fi)
SU (1) SU1192626A3 (fi)
UA (1) UA6342A1 (fi)
YU (1) YU42328B (fi)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN159362B (fi) * 1981-03-23 1987-05-09 Pfizer
US4419284A (en) * 1981-03-23 1983-12-06 Pfizer Inc. Preparation of halomethyl esters (and related esters) of penicillanic acid 1,1-dioxide
PT76527B (en) * 1982-04-19 1985-12-09 Gist Brocades Nv A process for the preparation of penicillanic acid 1,1-dioxide and derivatives thereof
IT1190897B (it) * 1982-06-29 1988-02-24 Opos Biochimica Srl Procedimento per la preparazione dell'estere 1-etossicarbonilossietilico dell'acido 6-(d(-)-alfa aminoalfa fenilacetamido)-penicillanico
US4606865A (en) * 1982-09-20 1986-08-19 Astra Lakemedel Aktiebolag Methods for the preparation of α-bromodiethylcarbonate
EP0139047A1 (en) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Process for the preparation of 6,6-dibromopenicillanic acid 1,1-dioxide
EP0139048A1 (en) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Process for the dehalogenation of 6,6-dibromopenicillanic acid 1,1-dioxide
US4596677A (en) * 1984-04-06 1986-06-24 Bristol-Myers Company Anhydropenicillin intermediates

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN149747B (fi) * 1977-06-07 1982-04-03 Pfizer
CA1158639A (en) * 1978-12-11 1983-12-13 Eric M. Gordon 6-bromopenicillanic acid sulfone
DE3068390D1 (en) * 1979-01-10 1984-08-09 Beecham Group Plc Penicillin derivatives, process for their preparation and pharmaceutical compositions containing certain of these compounds
IE49880B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd Penicillin derivatives

Also Published As

Publication number Publication date
YU58580A (en) 1983-02-28
IT8020367A0 (it) 1980-03-05
IE800429L (en) 1980-09-05
SE8000512L (sv) 1980-09-06
GB2045755A (en) 1980-11-05
PL125197B1 (en) 1983-04-30
UA6342A1 (uk) 1994-12-29
ES489185A0 (es) 1981-02-16
NL180317C (nl) 1987-02-02
NL180317B (nl) 1986-09-01
MY8500319A (en) 1985-12-31
DK166353B (da) 1993-04-13
AU522572B2 (en) 1982-06-17
SE8603309L (sv) 1986-08-04
DK145690D0 (da) 1990-06-14
YU42328B (en) 1988-08-31
LU82215A1 (fr) 1980-09-24
KR850001339B1 (ko) 1985-09-19
DK159852B (da) 1990-12-17
AT366693B (de) 1982-04-26
PT70897A (en) 1980-04-01
DE3008257C2 (de) 1984-03-01
IL59515A0 (en) 1980-06-30
BG33292A3 (en) 1983-01-14
FI800661A (fi) 1980-09-06
FR2450836A1 (fr) 1980-10-03
IT1130300B (it) 1986-06-11
PL222448A1 (fi) 1981-01-02
FR2450836B1 (fr) 1986-03-21
HK66587A (en) 1987-09-25
NL8001285A (nl) 1980-09-09
SU1192626A3 (ru) 1985-11-15
RO80112A (ro) 1982-10-26
DK159852C (da) 1991-05-06
AR225031A1 (es) 1982-02-15
MX6032E (es) 1984-10-04
DK145690A (da) 1990-06-14
SE449103B (sv) 1987-04-06
FI70024C (fi) 1986-09-12
ATA119080A (de) 1981-09-15
AU5610480A (en) 1980-09-11
CH644608A5 (de) 1984-08-15
FI70024B (fi) 1986-01-31
SG55884G (en) 1985-03-08
KE3464A (en) 1984-10-12
SE8603309D0 (sv) 1986-08-04
HU186304B (en) 1985-07-29
DD149367A5 (de) 1981-07-08
IL59515A (en) 1983-02-23
DK166353C (da) 1993-09-06
EG14437A (en) 1984-09-30
CS215130B2 (en) 1982-07-30
GR67234B (fi) 1981-06-25
GB2045755B (en) 1983-01-26
DK92680A (da) 1980-09-06
DE3008257A1 (de) 1980-09-11
IE49535B1 (en) 1985-10-16
IN153685B (fi) 1984-08-04
NO800618L (no) 1980-09-08
NO823127L (no) 1980-09-08

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 20010217