ES469922A1 - Un procedimiento para la preparacion de un derivado del 1,1-dioxido del acido penicilanico - Google Patents

Un procedimiento para la preparacion de un derivado del 1,1-dioxido del acido penicilanico

Info

Publication number
ES469922A1
ES469922A1 ES469922A ES469922A ES469922A1 ES 469922 A1 ES469922 A1 ES 469922A1 ES 469922 A ES469922 A ES 469922A ES 469922 A ES469922 A ES 469922A ES 469922 A1 ES469922 A1 ES 469922A1
Authority
ES
Spain
Prior art keywords
dioxide
penicillanic acid
translation
preparation
machine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES469922A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of ES469922A1 publication Critical patent/ES469922A1/es
Expired legal-status Critical Current

Links

Classifications

    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

La presente invención proporciona ciertos nuevos compuestos de penicilina que son útiles como agentes antibacterianos y que son también inhibidores potentes de las betalactamasas microbianas. Estos nuevos compuestos de penicilina son el 1,1-dióxido del ácido penicilánico, y ésteres del mismo que son fácilmente hidrolizables in vivo. La invención proporciona asimismo derivados del 1,1-dióxido de ácido penicilánico que tienen un grupo protector de carboxi que tienen un grupo protector de carboxi que son útiles como intermedios para la preparación del 1,1-dióxido del ácido penicilánico; y la invención además consiste de 1-óxidos del ácido penicilánico y ciertos ésteres de los mismos que son también útiles como intermedios para el 1,1-dióxido del ácido penicilánico.
ES469922A 1977-06-07 1978-05-17 Un procedimiento para la preparacion de un derivado del 1,1-dioxido del acido penicilanico Expired ES469922A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US80432077A 1977-06-07 1977-06-07
US87938178A 1978-02-21 1978-02-21
US89045178A 1978-03-29 1978-03-29

Publications (1)

Publication Number Publication Date
ES469922A1 true ES469922A1 (es) 1979-09-16

Family

ID=27420003

Family Applications (3)

Application Number Title Priority Date Filing Date
ES469922A Expired ES469922A1 (es) 1977-06-07 1978-05-17 Un procedimiento para la preparacion de un derivado del 1,1-dioxido del acido penicilanico
ES477768A Expired ES477768A1 (es) 1977-06-07 1979-02-15 Un procedimiento para la preparacion de 1 alfa-oxido de aci-do penicilinico.
ES490102A Granted ES490102A0 (es) 1977-06-07 1980-03-31 Un procedimiento para la preparacion de 1beta-oxido de acidopenicilanico

Family Applications After (2)

Application Number Title Priority Date Filing Date
ES477768A Expired ES477768A1 (es) 1977-06-07 1979-02-15 Un procedimiento para la preparacion de 1 alfa-oxido de aci-do penicilinico.
ES490102A Granted ES490102A0 (es) 1977-06-07 1980-03-31 Un procedimiento para la preparacion de 1beta-oxido de acidopenicilanico

Country Status (3)

Country Link
CA (2) CA1119164A (es)
ES (3) ES469922A1 (es)
MX (1) MX5526E (es)

Also Published As

Publication number Publication date
ES477768A1 (es) 1980-06-16
CA1119164A (en) 1982-03-02
ES8107223A1 (es) 1981-08-16
CA1129773A (en) 1982-08-17
ES490102A0 (es) 1981-08-16
MX5526E (es) 1983-09-23

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