SE8000512L - Sett att framstella penicillansyra-1,1-dioxid och estrar derav jemte mellanprodukter for settets genomforande - Google Patents

Sett att framstella penicillansyra-1,1-dioxid och estrar derav jemte mellanprodukter for settets genomforande

Info

Publication number
SE8000512L
SE8000512L SE8000512A SE8000512A SE8000512L SE 8000512 L SE8000512 L SE 8000512L SE 8000512 A SE8000512 A SE 8000512A SE 8000512 A SE8000512 A SE 8000512A SE 8000512 L SE8000512 L SE 8000512L
Authority
SE
Sweden
Prior art keywords
penicillanic acid
dioxide
vivo
readily hydrolyzable
esters
Prior art date
Application number
SE8000512A
Other languages
English (en)
Other versions
SE449103B (sv
Inventor
B S Moore
R D Carroll
R A Volkmann
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of SE8000512L publication Critical patent/SE8000512L/sv
Publication of SE449103B publication Critical patent/SE449103B/sv

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
SE8000512A 1979-03-05 1980-01-22 Sett att framstella penicillansyra-1,1-dioxid samt estrar derav SE449103B (sv)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1780879A 1979-03-05 1979-03-05
US1781079A 1979-03-05 1979-03-05

Publications (2)

Publication Number Publication Date
SE8000512L true SE8000512L (sv) 1980-09-06
SE449103B SE449103B (sv) 1987-04-06

Family

ID=26690337

Family Applications (2)

Application Number Title Priority Date Filing Date
SE8000512A SE449103B (sv) 1979-03-05 1980-01-22 Sett att framstella penicillansyra-1,1-dioxid samt estrar derav
SE8603309A SE8603309D0 (sv) 1979-03-05 1986-08-04 Mellanprodukter for framstellning av penicillansyra-1,1-dioxid och estrar derav

Family Applications After (1)

Application Number Title Priority Date Filing Date
SE8603309A SE8603309D0 (sv) 1979-03-05 1986-08-04 Mellanprodukter for framstellning av penicillansyra-1,1-dioxid och estrar derav

Country Status (36)

Country Link
KR (1) KR850001339B1 (sv)
AR (1) AR225031A1 (sv)
AT (1) AT366693B (sv)
AU (1) AU522572B2 (sv)
BG (1) BG33292A3 (sv)
CH (1) CH644608A5 (sv)
CS (1) CS215130B2 (sv)
DD (1) DD149367A5 (sv)
DE (1) DE3008257C2 (sv)
DK (2) DK159852C (sv)
EG (1) EG14437A (sv)
ES (1) ES8103094A1 (sv)
FI (1) FI70024C (sv)
FR (1) FR2450836B1 (sv)
GB (1) GB2045755B (sv)
GR (1) GR67234B (sv)
HK (1) HK66587A (sv)
HU (1) HU186304B (sv)
IE (1) IE49535B1 (sv)
IL (1) IL59515A (sv)
IN (1) IN153685B (sv)
IT (1) IT1130300B (sv)
KE (1) KE3464A (sv)
LU (1) LU82215A1 (sv)
MX (1) MX6032E (sv)
MY (1) MY8500319A (sv)
NL (1) NL180317C (sv)
NO (2) NO800618L (sv)
PL (1) PL125197B1 (sv)
PT (1) PT70897A (sv)
RO (1) RO80112A (sv)
SE (2) SE449103B (sv)
SG (1) SG55884G (sv)
SU (1) SU1192626A3 (sv)
UA (1) UA6342A1 (sv)
YU (1) YU42328B (sv)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN159362B (sv) * 1981-03-23 1987-05-09 Pfizer
US4419284A (en) * 1981-03-23 1983-12-06 Pfizer Inc. Preparation of halomethyl esters (and related esters) of penicillanic acid 1,1-dioxide
PT76527B (en) * 1982-04-19 1985-12-09 Gist Brocades Nv A process for the preparation of penicillanic acid 1,1-dioxide and derivatives thereof
IT1190897B (it) * 1982-06-29 1988-02-24 Opos Biochimica Srl Procedimento per la preparazione dell'estere 1-etossicarbonilossietilico dell'acido 6-(d(-)-alfa aminoalfa fenilacetamido)-penicillanico
US4606865A (en) * 1982-09-20 1986-08-19 Astra Lakemedel Aktiebolag Methods for the preparation of α-bromodiethylcarbonate
EP0139047A1 (en) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Process for the preparation of 6,6-dibromopenicillanic acid 1,1-dioxide
EP0139048A1 (en) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Process for the dehalogenation of 6,6-dibromopenicillanic acid 1,1-dioxide
US4596677A (en) * 1984-04-06 1986-06-24 Bristol-Myers Company Anhydropenicillin intermediates

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN149747B (sv) * 1977-06-07 1982-04-03 Pfizer
CA1158639A (en) * 1978-12-11 1983-12-13 Eric M. Gordon 6-bromopenicillanic acid sulfone
DE3068390D1 (en) * 1979-01-10 1984-08-09 Beecham Group Plc Penicillin derivatives, process for their preparation and pharmaceutical compositions containing certain of these compounds
IE49880B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd Penicillin derivatives

Also Published As

Publication number Publication date
YU58580A (en) 1983-02-28
IT8020367A0 (it) 1980-03-05
IE800429L (en) 1980-09-05
GB2045755A (en) 1980-11-05
PL125197B1 (en) 1983-04-30
UA6342A1 (uk) 1994-12-29
ES489185A0 (es) 1981-02-16
NL180317C (nl) 1987-02-02
NL180317B (nl) 1986-09-01
MY8500319A (en) 1985-12-31
DK166353B (da) 1993-04-13
AU522572B2 (en) 1982-06-17
SE8603309L (sv) 1986-08-04
DK145690D0 (da) 1990-06-14
YU42328B (en) 1988-08-31
LU82215A1 (fr) 1980-09-24
KR850001339B1 (ko) 1985-09-19
DK159852B (da) 1990-12-17
AT366693B (de) 1982-04-26
PT70897A (en) 1980-04-01
DE3008257C2 (de) 1984-03-01
IL59515A0 (en) 1980-06-30
BG33292A3 (en) 1983-01-14
FI800661A (fi) 1980-09-06
FR2450836A1 (fr) 1980-10-03
IT1130300B (it) 1986-06-11
PL222448A1 (sv) 1981-01-02
FR2450836B1 (fr) 1986-03-21
HK66587A (en) 1987-09-25
NL8001285A (nl) 1980-09-09
SU1192626A3 (ru) 1985-11-15
RO80112A (ro) 1982-10-26
DK159852C (da) 1991-05-06
AR225031A1 (es) 1982-02-15
MX6032E (es) 1984-10-04
DK145690A (da) 1990-06-14
SE449103B (sv) 1987-04-06
FI70024C (fi) 1986-09-12
ES8103094A1 (es) 1981-02-16
ATA119080A (de) 1981-09-15
AU5610480A (en) 1980-09-11
CH644608A5 (de) 1984-08-15
FI70024B (fi) 1986-01-31
SG55884G (en) 1985-03-08
KE3464A (en) 1984-10-12
SE8603309D0 (sv) 1986-08-04
HU186304B (en) 1985-07-29
DD149367A5 (de) 1981-07-08
IL59515A (en) 1983-02-23
DK166353C (da) 1993-09-06
EG14437A (en) 1984-09-30
CS215130B2 (en) 1982-07-30
GR67234B (sv) 1981-06-25
GB2045755B (en) 1983-01-26
DK92680A (da) 1980-09-06
DE3008257A1 (de) 1980-09-11
IE49535B1 (en) 1985-10-16
IN153685B (sv) 1984-08-04
NO800618L (no) 1980-09-08
NO823127L (no) 1980-09-08

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