ES480916A1 - Un procedimiento para la preparacion de antibioticos de ce- falosporina. - Google Patents
Un procedimiento para la preparacion de antibioticos de ce- falosporina.Info
- Publication number
- ES480916A1 ES480916A1 ES480916A ES480916A ES480916A1 ES 480916 A1 ES480916 A1 ES 480916A1 ES 480916 A ES480916 A ES 480916A ES 480916 A ES480916 A ES 480916A ES 480916 A1 ES480916 A1 ES 480916A1
- Authority
- ES
- Spain
- Prior art keywords
- antibiotics
- formula
- activity
- organisms
- strains
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/587—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Los antibióticos de cefalosporina se emplean ampliamente en el tratamiento de enfermedades originadas por bacterias patógenas en seres humanos y animales, y son especialmente útiles en el tratamiento de enfermedades originadas por bacterias que son resistentes a otros antibióticos tales como compuestos de penicilina, y en el tratamiento de pacientes sensibles a la penicilina. En muchos casos se desea emplear un antibiótico de cefalosporina que presenta actividad frente a los microorganismos tanto gram-positivos como gram-negativos, y una cantidad significativa de investigación ha sido dirigida al desarrollo de diversos tipos de antibióticos de cefalosporina de amplio espectro.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB23041/78A GB1604723A (en) | 1978-05-26 | 1978-05-26 | 7-(2-aminothiazol-4-yl)-2-oxyimino-acetamido)-cephem derivatives |
GB2304278A GB1604724A (en) | 1978-05-26 | 1978-05-26 | 7-(2-aminothiazol-4-yl)-2-oxymino-acedamido)-cephem derivatives |
GB7842166 | 1978-10-27 | ||
GB7842196 | 1978-10-27 |
Publications (1)
Publication Number | Publication Date |
---|---|
ES480916A1 true ES480916A1 (es) | 1980-02-01 |
Family
ID=27448575
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES480918A Expired ES480918A1 (es) | 1978-05-26 | 1979-05-25 | Un procedimiento para la preparacion de antibioticos de ce- falosporina. |
ES480916A Expired ES480916A1 (es) | 1978-05-26 | 1979-05-25 | Un procedimiento para la preparacion de antibioticos de ce- falosporina. |
ES480917A Expired ES480917A1 (es) | 1978-05-26 | 1979-05-25 | Un procedimiento para la preparacion de antibioticos de ce- falosporina. |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES480918A Expired ES480918A1 (es) | 1978-05-26 | 1979-05-25 | Un procedimiento para la preparacion de antibioticos de ce- falosporina. |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES480917A Expired ES480917A1 (es) | 1978-05-26 | 1979-05-25 | Un procedimiento para la preparacion de antibioticos de ce- falosporina. |
Country Status (21)
Country | Link |
---|---|
US (1) | US4621081A (es) |
AR (2) | AR231986A1 (es) |
AT (2) | AT369748B (es) |
AU (1) | AU524734B2 (es) |
CH (1) | CH648851A5 (es) |
DE (1) | DE2921332A1 (es) |
DK (1) | DK216879A (es) |
ES (3) | ES480918A1 (es) |
FI (1) | FI791679A (es) |
FR (1) | FR2426694A1 (es) |
HU (1) | HU182960B (es) |
IE (1) | IE49175B1 (es) |
IL (1) | IL57398A (es) |
IT (1) | IT1116185B (es) |
LU (1) | LU81320A1 (es) |
NL (1) | NL7904123A (es) |
NO (1) | NO791730L (es) |
NZ (1) | NZ190559A (es) |
PH (1) | PH15928A (es) |
PT (3) | PT69672A (es) |
SE (1) | SE7904577L (es) |
Families Citing this family (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE878514A (fr) * | 1978-09-04 | 1980-02-29 | Fujisawa Pharmaceutical Co | Procede de preparation de composes d'acide 3-cephem-4-carboxylique a disubstitution en positions 3 et 7, nouveaux produits ainsi obtenus et leur utilisation pour leur activite antibacterienne |
US4237128A (en) * | 1979-04-12 | 1980-12-02 | E. R. Squibb & Sons, Inc. | 7-[2-(2-Amino-4-thiazolyl)-2-[(1-carboxy-1,1-dialkyl)alkoxyimino]acetamido]cephem sulfoxides |
FR2476647A2 (fr) * | 1980-02-26 | 1981-08-28 | Roussel Uclaf | Procede de preparation de derives de l'acide 2-(2-amino protege 4-thiazolyl) 2-alkoxyimino acetique isomere syn |
GR75487B (es) * | 1981-06-22 | 1984-07-23 | Fujisawa Pharmaceutical Co | |
FR2516515A1 (fr) * | 1981-11-16 | 1983-05-20 | Sanofi Sa | Nouveaux derives de pyridinium thiomethyl cephalosporines, procede pour leur preparation et compositions pharmaceutiques les contenant |
DE3485860T2 (de) * | 1983-12-29 | 1993-01-14 | Mochida Pharm Co Ltd | Cephalosporinverbindungen, verfahren zu ihrer herstellung und pharmazeutishe praeparate. |
JPS60142987A (ja) * | 1983-12-29 | 1985-07-29 | Mochida Pharmaceut Co Ltd | セフアロスポリン誘導体 |
KR920004820B1 (ko) * | 1984-02-23 | 1992-06-18 | 메이지제과 주식회사 | 새로운 세팔로스포린 유도체의 제조방법 |
FI851934L (fi) * | 1984-05-30 | 1985-12-01 | Ici Plc | Kefalosporinderivat. |
US4840945A (en) * | 1985-04-01 | 1989-06-20 | Mochida Pharmaceutical Co., Ltd. | Cephalosporin derivatives |
JPH064645B2 (ja) * | 1985-11-27 | 1994-01-19 | 明治製菓株式会社 | 新規セフアロスポリン誘導体およびそれを含む抗菌剤 |
US4880797A (en) * | 1986-03-20 | 1989-11-14 | Banyu Pharmaceutical Co., Ltd. | Cephalosporin derivatives and antibacterial agents |
US4880798A (en) * | 1986-11-25 | 1989-11-14 | Mochida Pharmaceutical Co., Ltd. | Cephalosporin derivatives |
JPS63132893A (ja) * | 1986-11-25 | 1988-06-04 | Mochida Pharmaceut Co Ltd | 新規セフアロスポリン誘導体、その製法およびそれらを有効成分とする抗菌剤 |
JPS63154622A (ja) * | 1986-12-18 | 1988-06-27 | Meiji Seika Kaisha Ltd | セフアロスポリン誘導体を有効成分とする哺乳動物用抗菌剤 |
JPH01254686A (ja) * | 1988-04-05 | 1989-10-11 | Katayama Seiyakushiyo:Kk | セフエム化合物およびその製造法 |
US5202315A (en) * | 1989-05-11 | 1993-04-13 | Lucky, Ltd. | Cephalosporin compounds |
ATE123034T1 (de) * | 1990-03-24 | 1995-06-15 | Lucky Ltd | Cephalosporinzwischenverbindungen, verfahren zu ihrer herstellung sowie zur herstellung ihrer endprodukte. |
WO1992008721A1 (en) * | 1990-11-09 | 1992-05-29 | Lucky, Ltd. | Novel cephalosporin compounds and processes for preparation thereof |
KR0154901B1 (ko) * | 1992-12-26 | 1998-11-16 | 성재갑 | 신규 세팔로스포린계 항생제(v) |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4144393A (en) * | 1973-12-21 | 1979-03-13 | Glaxo Laboratories Limited | 3-Acetoxymethyl cephalosporins having at position-7 a carboxy substituted α-etherified hydroxyiminoarylacetamido group |
DE2714880A1 (de) * | 1977-04-02 | 1978-10-26 | Hoechst Ag | Cephemderivate und verfahren zu ihrer herstellung |
IE49211B1 (en) * | 1978-11-17 | 1985-08-21 | Glaxo Group Ltd | Cephalosporin antibiotics |
IL59680A (en) * | 1979-03-22 | 1983-07-31 | Glaxo Group Ltd | 7-(((z)-2-(2-aminothiazol-4-yl)-2-(2-carboxy(lower alkyl or cycloalkyl)oxyimino)acetimido)-3-((1-carbamoylmethylpyridinium)thiomethyl)-ceph-3-em-4-carboxylates,their preparation and pharmaceutical compositions comprising them |
US4237128A (en) * | 1979-04-12 | 1980-12-02 | E. R. Squibb & Sons, Inc. | 7-[2-(2-Amino-4-thiazolyl)-2-[(1-carboxy-1,1-dialkyl)alkoxyimino]acetamido]cephem sulfoxides |
-
1979
- 1979-05-24 AR AR276667A patent/AR231986A1/es active
- 1979-05-24 AR AR276666A patent/AR229882A1/es active
- 1979-05-25 PH PH22563A patent/PH15928A/en unknown
- 1979-05-25 ES ES480918A patent/ES480918A1/es not_active Expired
- 1979-05-25 ES ES480916A patent/ES480916A1/es not_active Expired
- 1979-05-25 DE DE19792921332 patent/DE2921332A1/de not_active Withdrawn
- 1979-05-25 NO NO791730A patent/NO791730L/no unknown
- 1979-05-25 IT IT49176/79A patent/IT1116185B/it active
- 1979-05-25 NZ NZ190559A patent/NZ190559A/xx unknown
- 1979-05-25 AU AU47420/79A patent/AU524734B2/en not_active Ceased
- 1979-05-25 HU HU79GA1288A patent/HU182960B/hu unknown
- 1979-05-25 PT PT69672A patent/PT69672A/pt unknown
- 1979-05-25 NL NL7904123A patent/NL7904123A/xx not_active Application Discontinuation
- 1979-05-25 FI FI791679A patent/FI791679A/fi not_active Application Discontinuation
- 1979-05-25 PT PT69673A patent/PT69673A/pt unknown
- 1979-05-25 PT PT69671A patent/PT69671A/pt unknown
- 1979-05-25 ES ES480917A patent/ES480917A1/es not_active Expired
- 1979-05-25 SE SE7904577A patent/SE7904577L/xx not_active Application Discontinuation
- 1979-05-25 LU LU81320A patent/LU81320A1/xx unknown
- 1979-05-25 IL IL57398A patent/IL57398A/xx unknown
- 1979-05-25 DK DK216879A patent/DK216879A/da not_active Application Discontinuation
- 1979-05-25 CH CH4917/79A patent/CH648851A5/de not_active IP Right Cessation
- 1979-05-28 FR FR7913524A patent/FR2426694A1/fr active Granted
- 1979-08-08 IE IE1027/79A patent/IE49175B1/en unknown
-
1980
- 1980-12-03 AT AT0590580A patent/AT369748B/de not_active IP Right Cessation
- 1980-12-03 AT AT0590680A patent/AT369749B/de not_active IP Right Cessation
-
1982
- 1982-09-27 US US06/423,555 patent/US4621081A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
AT369748B (de) | 1983-01-25 |
ES480917A1 (es) | 1980-02-01 |
AR229882A1 (es) | 1983-12-30 |
AR231986A1 (es) | 1985-04-30 |
NO791730L (no) | 1979-11-27 |
NZ190559A (en) | 1982-05-25 |
FR2426694B1 (es) | 1984-10-26 |
IT1116185B (it) | 1986-02-10 |
AT369749B (de) | 1983-01-25 |
IT7949176A0 (it) | 1979-05-25 |
SE7904577L (sv) | 1980-02-11 |
IE49175B1 (en) | 1985-08-21 |
PH15928A (en) | 1983-04-27 |
AU4742079A (en) | 1979-11-29 |
FI791679A (fi) | 1979-11-27 |
PT69672A (en) | 1979-06-01 |
HU182960B (en) | 1984-03-28 |
IE791027L (en) | 1979-11-26 |
IL57398A0 (en) | 1979-09-30 |
LU81320A1 (fr) | 1979-09-11 |
DK216879A (da) | 1979-11-27 |
IL57398A (en) | 1982-12-31 |
ATA590580A (de) | 1982-06-15 |
PT69671A (en) | 1979-06-01 |
CH648851A5 (de) | 1985-04-15 |
ES480918A1 (es) | 1980-02-01 |
AU524734B2 (en) | 1982-09-30 |
PT69673A (en) | 1979-06-01 |
NL7904123A (nl) | 1979-11-28 |
DE2921332A1 (de) | 1979-11-29 |
US4621081A (en) | 1986-11-04 |
FR2426694A1 (fr) | 1979-12-21 |
ATA590680A (de) | 1982-06-15 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD1A | Patent lapsed |
Effective date: 19971001 |