ES469648A1 - Un procedimiento para preparar derivados de oleandomicina - Google Patents

Un procedimiento para preparar derivados de oleandomicina

Info

Publication number
ES469648A1
ES469648A1 ES469648A ES469648A ES469648A1 ES 469648 A1 ES469648 A1 ES 469648A1 ES 469648 A ES469648 A ES 469648A ES 469648 A ES469648 A ES 469648A ES 469648 A1 ES469648 A1 ES 469648A1
Authority
ES
Spain
Prior art keywords
compounds
semi
synthetic
oleandomycin derivatives
oleandomycin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES469648A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/883,608 external-priority patent/US4136253A/en
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of ES469648A1 publication Critical patent/ES469648A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)

Abstract

Un procedimiento para preparar un compuesto que se selecciona de: **(Fórmula)** y una sal de adición de ácido, farmacéuticamente aceptable del mismo en donde R es alquilo de uno a tres átomos de carbono; piridilo; 1,1,1-trifluoetilo; fenilo; fenilo monosubstituido en donde el sustituyente es fluor, cloro, bromo, yodo, hidroxi, motoxi, ciano, carboxamido, nitro, amino, carbometoxi, carbobenciloxi, carboxi, trifluometilo, alquilo de uno a cuatro átomos de carbono o acetamido; fenilo disubsustituido en donde el substituyente es cada uno cloro, nitro, amino, metoxi o metilo; triclorofenilo; hidroxidicloro; bencilo; naftilo; tienilo; clorotienilo; 2-acetamido-5-tiazolilo; 2-bencimidazolilo; dimetil-2-pirimidinilo; pirrilo; furilo; tienilo, pirrilo o furilo monosubstituidos, en donde cada substituyente es carbometoxi o alquilo de uno a dos átomos de carbono; o 1-metil-55-carbometoxi-3-pirrilo.
ES469648A 1977-05-11 1978-05-10 Un procedimiento para preparar derivados de oleandomicina Expired ES469648A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US79585077A 1977-05-11 1977-05-11
US05/883,608 US4136253A (en) 1977-05-11 1978-03-06 Semi-synthetic 4"-sulfonylamino-oleandomycin derivatives

Publications (1)

Publication Number Publication Date
ES469648A1 true ES469648A1 (es) 1979-09-16

Family

ID=27121658

Family Applications (1)

Application Number Title Priority Date Filing Date
ES469648A Expired ES469648A1 (es) 1977-05-11 1978-05-10 Un procedimiento para preparar derivados de oleandomicina

Country Status (31)

Country Link
JP (1) JPS53149990A (es)
AR (1) AR219529A1 (es)
AT (1) AT357263B (es)
AU (1) AU500587B1 (es)
CA (1) CA1098123A (es)
CH (1) CH631461A5 (es)
CS (1) CS199728B2 (es)
DD (1) DD135907A5 (es)
DE (1) DE2820411C2 (es)
DK (1) DK148845C (es)
EG (1) EG13371A (es)
ES (1) ES469648A1 (es)
FI (1) FI67709C (es)
FR (1) FR2390453A1 (es)
GB (1) GB1590162A (es)
GR (1) GR70056B (es)
HU (1) HU180279B (es)
IE (1) IE46839B1 (es)
IL (1) IL54688A (es)
IT (1) IT1094816B (es)
LU (1) LU79638A1 (es)
NL (1) NL174254C (es)
NO (1) NO145384C (es)
NZ (1) NZ187229A (es)
PH (1) PH15382A (es)
PL (1) PL111988B1 (es)
PT (1) PT68019B (es)
RO (1) RO75819A (es)
SE (1) SE446340B (es)
SU (1) SU860707A1 (es)
YU (1) YU40963B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4124755A (en) * 1978-01-03 1978-11-07 Pfizer Inc. 11-Alkanoyl-4"-deoxy-4"-isonitrilo-oleandomycin derivatives
US4133950A (en) * 1978-01-03 1979-01-09 Pfizer Inc. 4"-Deoxy-4"-carbamate and dithiocarbamate derivatives of oleandomycin and its esters

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3836519A (en) * 1973-05-04 1974-09-17 Abbott Lab Sulfonyl derivatives of erythromycin

Also Published As

Publication number Publication date
FI781478A (fi) 1978-11-12
DK205878A (da) 1978-11-12
DK148845B (da) 1985-10-21
IT1094816B (it) 1985-08-10
JPS53149990A (en) 1978-12-27
FR2390453A1 (fr) 1978-12-08
LU79638A1 (fr) 1979-12-06
NL174254C (nl) 1984-05-16
YU40963B (en) 1986-08-31
CS199728B2 (en) 1980-07-31
PH15382A (en) 1982-12-17
AR219529A1 (es) 1980-08-29
GB1590162A (en) 1981-05-28
NO145384C (no) 1982-03-10
ATA338978A (de) 1979-11-15
SE446340B (sv) 1986-09-01
RO75819A (ro) 1981-04-30
PL206687A1 (pl) 1979-04-23
IE780953L (en) 1978-11-11
EG13371A (en) 1981-06-30
YU108278A (en) 1983-01-21
NZ187229A (en) 1980-02-21
PT68019B (en) 1979-10-24
GR70056B (es) 1982-07-26
AU500587B1 (en) 1979-05-24
IL54688A0 (en) 1978-07-31
FR2390453B1 (es) 1980-07-04
CA1098123A (en) 1981-03-24
SE7804080L (sv) 1978-11-12
HU180279B (en) 1983-02-28
IT7823229A0 (it) 1978-05-10
SU860707A1 (ru) 1981-08-30
AT357263B (de) 1980-06-25
FI67709B (fi) 1985-01-31
IE46839B1 (en) 1983-10-05
DE2820411A1 (de) 1978-11-16
DE2820411C2 (de) 1983-05-11
NO145384B (no) 1981-11-30
NO781656L (no) 1978-11-14
JPS5633400B2 (es) 1981-08-03
DD135907A5 (de) 1979-06-06
IL54688A (en) 1982-01-31
DK148845C (da) 1986-04-14
FI67709C (fi) 1985-05-10
NL7805007A (nl) 1978-11-14
PL111988B1 (en) 1980-09-30
NL174254B (nl) 1983-12-16
PT68019A (en) 1978-06-01
CH631461A5 (en) 1982-08-13

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19990201