ES456370A1 - Procedimiento para preparar aril-3-oxazolidinonas-2. - Google Patents
Procedimiento para preparar aril-3-oxazolidinonas-2.Info
- Publication number
- ES456370A1 ES456370A1 ES456370A ES456370A ES456370A1 ES 456370 A1 ES456370 A1 ES 456370A1 ES 456370 A ES456370 A ES 456370A ES 456370 A ES456370 A ES 456370A ES 456370 A1 ES456370 A1 ES 456370A1
- Authority
- ES
- Spain
- Prior art keywords
- methyl
- hydrogen
- fluoro
- nitro
- carbon atoms
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 230000001225 therapeutic effect Effects 0.000 title 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 4
- 239000001257 hydrogen Substances 0.000 abstract 4
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 4
- 125000004432 carbon atom Chemical group C* 0.000 abstract 3
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 125000000113 cyclohexyl group Chemical group [H]C1([H])C([H])([H])C([H])([H])C([H])(*)C([H])([H])C1([H])[H] 0.000 abstract 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 2
- 125000001494 2-propynyl group Chemical group [H]C#CC([H])([H])* 0.000 abstract 1
- -1 acetylmethyl cyanomethyl Chemical group 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000004210 cyclohexylmethyl group Chemical group [H]C([H])(*)C1([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C1([H])[H] 0.000 abstract 1
- XNMQEEKYCVKGBD-UHFFFAOYSA-N dimethylacetylene Natural products CC#CC XNMQEEKYCVKGBD-UHFFFAOYSA-N 0.000 abstract 1
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
- C07D263/24—Oxygen atoms attached in position 2 with hydrocarbon radicals, substituted by oxygen atoms, attached to other ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Psychiatry (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pain & Pain Management (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR7605751A FR2342729A1 (fr) | 1976-03-01 | 1976-03-01 | Nouveaux derives de la carbamoyloxymethyl-5 oxazolidinone-2, leur procede de preparation et leur application en therapeutique |
| FR7619578A FR2356422A1 (fr) | 1976-03-01 | 1976-06-28 | Nouveaux hydroxymethyl-5 oxazolidinone-2, leur procede de preparation et leur application en therapeutique |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES456370A1 true ES456370A1 (es) | 1978-01-16 |
Family
ID=26219328
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES456370A Expired ES456370A1 (es) | 1976-03-01 | 1977-02-26 | Procedimiento para preparar aril-3-oxazolidinonas-2. |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US4150029A (enExample) |
| JP (1) | JPS6040428B2 (enExample) |
| AU (1) | AU509376B2 (enExample) |
| BE (1) | BE851893A (enExample) |
| CA (1) | CA1106380A (enExample) |
| CH (2) | CH618975A5 (enExample) |
| DE (1) | DE2708236A1 (enExample) |
| ES (1) | ES456370A1 (enExample) |
| FR (1) | FR2356422A1 (enExample) |
| GB (1) | GB1546741A (enExample) |
| GR (1) | GR60803B (enExample) |
| IT (1) | IT1071584B (enExample) |
| LU (1) | LU76848A1 (enExample) |
| MX (1) | MX4652E (enExample) |
| NL (1) | NL7702148A (enExample) |
| SE (1) | SE435928B (enExample) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| LU80081A1 (fr) * | 1977-08-26 | 1979-05-15 | Delalande Sa | Nouvelles hydroxymethyl-5 oxazolidinones-2,leur procede de preparation et leur application therapeutique |
| US4348393A (en) * | 1978-06-09 | 1982-09-07 | Delalande S.A. | N-Aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones |
| FR2456097A1 (fr) * | 1979-05-07 | 1980-12-05 | Delalande Sa | Nouveaux derives de la 5 h-furanone-2 et de la 3 h-dihydrofuranone-2, leur procede de preparation et leur application en therapeutique |
| US4226612A (en) * | 1979-07-02 | 1980-10-07 | Shell Oil Company | Certain herbicidal (2-oxo-3-oxazolidinyl)phenylureas |
| CA1171865A (en) * | 1980-06-04 | 1984-07-31 | Alain Lacour | N-aryl azolone derivatives, the process for preparing the same and their application in therapeutics |
| US4340606A (en) * | 1980-10-23 | 1982-07-20 | E. I. Du Pont De Nemours And Company | 3-(p-Alkylsulfonylphenyl)oxazolidinone derivatives as antibacterial agents |
| FR2528046B1 (fr) * | 1982-06-08 | 1985-06-21 | Delalande Sa | Derives de l'oxazolidinone-2 n-arylee optiquement actifs, inhibiteurs specifiques et reversibles de la monoamine oxydase de type b et leur procede de preparation |
| US5254577A (en) * | 1988-07-29 | 1993-10-19 | The Du Pont Merck Pharmaceutical Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
| US4948801A (en) * | 1988-07-29 | 1990-08-14 | E. I. Du Pont De Nemours And Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
| US5196543A (en) * | 1989-10-17 | 1993-03-23 | Delalande S.A. | 3-aryloxazolidinone derivatives, process for their preparation and their use in therapy |
| US5235063A (en) * | 1989-10-17 | 1993-08-10 | Delalande S.A. | Process of preparing by condensation certain |
| US5182296A (en) * | 1989-10-26 | 1993-01-26 | Tanabe Seiyaky Co., Ltd. | Naphthyloxazolidone derivatives |
| TW286317B (enExample) * | 1993-12-13 | 1996-09-21 | Hoffmann La Roche | |
| AU716493B2 (en) | 1995-09-01 | 2000-02-24 | Pharmacia & Upjohn Company | Phenyloxazolidinones having a C-C bond to 4-8 membered heterocyclic rings |
| DE69738457T2 (de) * | 1996-04-11 | 2008-12-24 | Pharmacia & Upjohn Co. Llc, Kalamazoo | Verfahren zur Herstellung von Oxazolidinonen |
| KR100619639B1 (ko) * | 1997-11-07 | 2006-09-06 | 파마시아 앤드 업존 캄파니 엘엘씨 | 옥사졸리디논의 제조 방법 |
| ID30299A (id) * | 1998-06-05 | 2001-11-22 | Astrazeneca Ab | Turunan oksazolidinon, proses pembuatannya dan komposisi farmasi yang mengandungnya |
| GB9928568D0 (en) | 1999-12-03 | 2000-02-02 | Zeneca Ltd | Chemical compounds |
| GB0009803D0 (en) * | 2000-04-25 | 2000-06-07 | Astrazeneca Ab | Chemical compounds |
| EP1328509B1 (en) * | 2000-10-17 | 2006-03-22 | Pharmacia & Upjohn Company LLC | Methods of producing oxazolidinone compounds |
| DE102008007802A1 (de) * | 2008-02-06 | 2009-08-13 | Sms Demag Ag | Verfahren und Einrichtung zur Regelung von Stellgrößen in hütten-technischen Anlagen |
| EP3914587A4 (en) * | 2019-01-18 | 2022-11-23 | Merck Sharp & Dohme LLC | OXAZOLIDINONE COMPOUNDS AND USES THEREOF AS ANTIBACTERIAL AGENTS |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH8A (fr) * | 1888-11-30 | Kuhn & Tieche | Nouveau mécanisme de remontoir et de mise à l'heure par le pendant pour montres de tous calibres | |
| GB1180089A (en) * | 1967-10-20 | 1970-02-04 | Delalande Sa | Acetylenic Derivatives of 2-Oxazolidinones and processes of preparation |
| GB1224995A (en) * | 1968-09-20 | 1971-03-10 | Delalande Sa | New 5-propargyloxymethyl-2-substituted oxazolidinones and their process of preparation |
| GB1250538A (enExample) * | 1969-03-18 | 1971-10-20 |
-
1976
- 1976-06-28 FR FR7619578A patent/FR2356422A1/fr active Granted
-
1977
- 1977-02-22 CH CH219177A patent/CH618975A5/fr not_active IP Right Cessation
- 1977-02-23 GR GR52833A patent/GR60803B/el unknown
- 1977-02-23 US US05/771,814 patent/US4150029A/en not_active Expired - Lifetime
- 1977-02-23 SE SE7702013A patent/SE435928B/xx not_active IP Right Cessation
- 1977-02-23 GB GB7593/77A patent/GB1546741A/en not_active Expired
- 1977-02-25 AU AU22689/77A patent/AU509376B2/en not_active Expired
- 1977-02-25 LU LU76848A patent/LU76848A1/xx unknown
- 1977-02-25 DE DE19772708236 patent/DE2708236A1/de not_active Ceased
- 1977-02-26 ES ES456370A patent/ES456370A1/es not_active Expired
- 1977-02-28 JP JP52021391A patent/JPS6040428B2/ja not_active Expired
- 1977-02-28 NL NL7702148A patent/NL7702148A/xx not_active Application Discontinuation
- 1977-02-28 MX MX775484U patent/MX4652E/es unknown
- 1977-02-28 BE BE175316A patent/BE851893A/xx unknown
- 1977-02-28 CA CA272,798A patent/CA1106380A/fr not_active Expired
- 1977-02-28 IT IT67439/77A patent/IT1071584B/it active
-
1980
- 1980-01-14 CH CH28380A patent/CH627460A5/fr not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| CH627460A5 (fr) | 1982-01-15 |
| CA1106380A (fr) | 1981-08-04 |
| IT1071584B (it) | 1985-04-10 |
| FR2356422B1 (enExample) | 1978-12-15 |
| FR2356422A1 (fr) | 1978-01-27 |
| CH618975A5 (enExample) | 1980-08-29 |
| DE2708236A1 (de) | 1977-09-08 |
| AU509376B2 (en) | 1980-05-08 |
| US4150029A (en) | 1979-04-17 |
| BE851893A (fr) | 1977-08-29 |
| SE7702013L (sv) | 1977-09-02 |
| GB1546741A (en) | 1979-05-31 |
| GR60803B (en) | 1978-08-30 |
| MX4652E (es) | 1982-07-16 |
| JPS6040428B2 (ja) | 1985-09-11 |
| SE435928B (sv) | 1984-10-29 |
| JPS52113959A (en) | 1977-09-24 |
| LU76848A1 (fr) | 1977-09-12 |
| AU2268977A (en) | 1978-08-31 |
| NL7702148A (nl) | 1977-09-05 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 19861126 |