ES453726A1 - Procedimiento para producir cefalosporinas y similares. - Google Patents

Procedimiento para producir cefalosporinas y similares.

Info

Publication number
ES453726A1
ES453726A1 ES453726A ES453726A ES453726A1 ES 453726 A1 ES453726 A1 ES 453726A1 ES 453726 A ES453726 A ES 453726A ES 453726 A ES453726 A ES 453726A ES 453726 A1 ES453726 A1 ES 453726A1
Authority
ES
Spain
Prior art keywords
group
unsubstituted
substituted
procedure
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES453726A
Other languages
English (en)
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sumitomo Chemical Co Ltd
Original Assignee
Sumitomo Chemical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sumitomo Chemical Co Ltd filed Critical Sumitomo Chemical Co Ltd
Publication of ES453726A1 publication Critical patent/ES453726A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/577-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with a further substituent in position 7, e.g. cephamycines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
ES453726A 1975-11-28 1976-11-27 Procedimiento para producir cefalosporinas y similares. Expired ES453726A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP50142647A JPS5268193A (en) 1975-11-28 1975-11-28 Synthesis of novel cephalosporin derivatives

Publications (1)

Publication Number Publication Date
ES453726A1 true ES453726A1 (es) 1978-01-16

Family

ID=15320206

Family Applications (4)

Application Number Title Priority Date Filing Date
ES453726A Expired ES453726A1 (es) 1975-11-28 1976-11-27 Procedimiento para producir cefalosporinas y similares.
ES463737A Expired ES463737A1 (es) 1975-11-28 1977-10-31 Metodo para producir cefalosporinas y similares
ES463735A Expired ES463735A1 (es) 1975-11-28 1977-10-31 Metodo de obtencion de cefalosporinas y similares.
ES463736A Expired ES463736A1 (es) 1975-11-28 1977-10-31 Procedimiento de obtencion de cefalosporinas y analogos.

Family Applications After (3)

Application Number Title Priority Date Filing Date
ES463737A Expired ES463737A1 (es) 1975-11-28 1977-10-31 Metodo para producir cefalosporinas y similares
ES463735A Expired ES463735A1 (es) 1975-11-28 1977-10-31 Metodo de obtencion de cefalosporinas y similares.
ES463736A Expired ES463736A1 (es) 1975-11-28 1977-10-31 Procedimiento de obtencion de cefalosporinas y analogos.

Country Status (19)

Country Link
US (2) US4125611A (OSRAM)
JP (1) JPS5268193A (OSRAM)
AT (4) AT352273B (OSRAM)
BE (1) BE848887A (OSRAM)
CA (1) CA1086716A (OSRAM)
CH (1) CH625527A5 (OSRAM)
CS (4) CS212257B2 (OSRAM)
DD (1) DD128562A5 (OSRAM)
DE (1) DE2653820A1 (OSRAM)
DK (1) DK535476A (OSRAM)
ES (4) ES453726A1 (OSRAM)
FR (1) FR2332758A1 (OSRAM)
GB (1) GB1532866A (OSRAM)
HU (1) HU173394B (OSRAM)
NL (1) NL7613206A (OSRAM)
NO (1) NO764054L (OSRAM)
NZ (1) NZ182740A (OSRAM)
SE (1) SE7613304L (OSRAM)
ZA (1) ZA767088B (OSRAM)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5268193A (en) * 1975-11-28 1977-06-06 Sumitomo Chem Co Ltd Synthesis of novel cephalosporin derivatives
AT375376B (de) * 1980-03-04 1984-07-25 Eisai Co Ltd Verfahren zur herstellung von neuen 7alphamethoxycephalosporinderivaten
US4503052A (en) * 1983-05-16 1985-03-05 Eli Lilly And Company 7-(2-(Substituted cinnolinoyl)amino)acetamido)-1-oxa-beta-lactams
US7183278B1 (en) 1998-11-04 2007-02-27 Meiji Seika Kaisha, Ltd. Picolinamide derivative and harmful organism control agent comprising said picolinamide derivative as active component
EP1159279B1 (en) 1999-03-09 2002-10-16 PHARMACIA & UPJOHN COMPANY 4-oxo-4,7-dihydro-thieno[2,3-b]pyridine-5-carboxamides as antiviral agents
DE60229364D1 (de) * 2001-03-01 2008-11-27 Shionogi & Co Stickstoffhaltige heteroarylverbindungen mit hiv-integrase inhibierender wirkung
WO2003020729A1 (en) 2001-08-30 2003-03-13 Pharmacia & Upjohn Company 4-THIOXO-4,7-DIHYDRO-THIENO[2,3-b]PYRIDINE-5-CARBOXAMIDES AS ANT IVIRAL AGENTS
WO2003020728A1 (en) * 2001-08-30 2003-03-13 Pharmacia & Upjohn Company 4-THIOXO-4,7-DIHYDRO-THIENO[2,3-b]PYRIDINE-5-CARBOTHIOAMIDES AS ANTIVIRAL AGENTS
AR038294A1 (es) * 2002-01-14 2005-01-12 Upjohn Co Oxotieno(3,2-b)piridincarboxamidas como agentes antivirales
AR038118A1 (es) * 2002-01-14 2004-12-29 Upjohn Co Compuestos derivados de la bencinamida del acido 7-oxo-4,7-dihidrotien[2,3-b[piridin-6-carboxilico 3-sustituido que son utiles como antivirales
AR038117A1 (es) * 2002-01-14 2004-12-29 Upjohn Co Agentes antivirales derivados de la 4- oxo-4,7 -dihidrofuro [2,3-b]piridin-5-carboxamida
ATE370948T1 (de) * 2002-01-17 2007-09-15 Merck & Co Inc Hydroxynaphthyridinoncarbonsäureamide, die sich als inhibitoren der hiv-integrase eignen

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1109860A (en) * 1972-12-08 1981-09-29 Shinji Terao Process for producing lactol-type cephalosporins
US4068074A (en) * 1974-04-05 1978-01-10 Yamanouchi Pharmaceutical Co., Ltd. Cephalosporin derivatives having at the 3-position of the cephem ring a heterocyclic thiomethyl group with a carboxy or sulfo group and at the 7-position of the cephem ring an α-heterocylic acylaminophenyl-acetamide group
CH606001A5 (OSRAM) * 1974-05-13 1978-10-13 Ciba Geigy Ag
US3989687A (en) * 1974-09-27 1976-11-02 Richardson-Merrell Inc. 4-Oxo-1-pyridinyl penicillin derivatives
JPS5268193A (en) * 1975-11-28 1977-06-06 Sumitomo Chem Co Ltd Synthesis of novel cephalosporin derivatives

Also Published As

Publication number Publication date
AT353970B (de) 1979-12-10
CH625527A5 (OSRAM) 1981-09-30
DD128562A5 (de) 1977-11-23
AT356817B (de) 1980-05-27
ATA581678A (de) 1979-05-15
AT352282B (de) 1979-09-10
ATA879876A (de) 1979-02-15
NZ182740A (en) 1979-01-11
JPS5268193A (en) 1977-06-06
NL7613206A (nl) 1977-06-01
DE2653820A1 (de) 1977-06-02
ES463736A1 (es) 1978-12-16
CS212257B2 (en) 1982-03-26
DK535476A (da) 1977-05-29
ATA679A (de) 1979-10-15
AU2001876A (en) 1978-06-01
CS212259B2 (cs) 1982-03-26
HU173394B (hu) 1979-04-28
AT352273B (de) 1979-09-10
ES463735A1 (es) 1978-12-16
FR2332758B1 (OSRAM) 1981-11-27
FR2332758A1 (fr) 1977-06-24
GB1532866A (en) 1978-11-22
US4226863A (en) 1980-10-07
CS212260B2 (cs) 1982-03-26
NO764054L (OSRAM) 1977-06-01
ES463737A1 (es) 1979-01-01
SE7613304L (sv) 1977-05-29
BE848887A (fr) 1977-03-16
US4125611A (en) 1978-11-14
ATA581778A (de) 1979-02-15
CA1086716A (en) 1980-09-30
CS212258B2 (cs) 1982-03-26
ZA767088B (en) 1977-10-26

Similar Documents

Publication Publication Date Title
AT320632B (de) Verfahren zur Herstellung von Furanderivaten
ES453726A1 (es) Procedimiento para producir cefalosporinas y similares.
ES456651A1 (es) Metodo de preparacion de cefalosporinas.
ES458307A1 (es) Un procedimiento de preparacion de nuevas 4-amino-piperidi- nas sustituidas en el nitrogeno del ciclo piperidico por unacadena aril-alcoilica o sus sales.
ES371709A1 (es) Un metodo para producir una penicilina sintetica.
ES443791A1 (es) Procedimiento para la preparacion de derivados del acido 3- cefem-4-carboxilico.
ES404745A1 (es) Un procedimiento para preparar cefalosporinas.
ES404315A1 (es) Un procedimiento de preparacion de un derivado de nitrosou-rea.
ES421417A1 (es) Procedimiento para la obtencion de composiciones desensibi-lizadoras para aplicacion de materiales registradores.
ES334350A1 (es) Un procedimiento de diazotipia.
SE385211B (sv) Sett att framstella organiska foreningar innehallande merkta atomer
ES401264A1 (es) Un procedimiento para la preparacion de una penicilina.
GB1244016A (en) Method for preparing penicillins
ES272079A1 (es) Procedimiento para la producción de compuestos heterocíclicos
ES299783A1 (es) Un procedimiento para la preparación de 1-naftilacetamidas alfasustituídas
ES403864A1 (es) Un procedimiento para la preparacion de antibioticos de ce-falosporina.
ES468581A1 (es) Metodo de produccion de compuestos terapeuticos cefalospori-nicos
SE7713979L (sv) Sett att framstella en blandning av 2-ketogulonat och 2-ketoglukonat
ES402382A1 (es) Un procedimiento para la preparacion de benzopiranos susti-tuidos.
ES367957A1 (es) Un procedimiento para la preparacion de derivados de benzo-diacepina.
FR2013456A1 (en) Mixed anhydrides of carboxylic and phos - phorous or phosphoric acids useful as
KR830002783A (ko) 3-비닐-세팔로스포린 유도체 제조방법
ES388250A1 (es) Un procedimiento para preparar compuestos de acido pirazo- lo-piridincarboxilico.
ES419266A1 (es) Un procedimiento para preparar derivados de quinazolina.
ES385778A1 (es) Un metodo para producir derivados de benzazocina.

Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19981001