ES398949A1 - Procedimiento para la fabricacion de nuevos derivados de bezilftalazona, basicamente sustituidos y sus sales. - Google Patents

Procedimiento para la fabricacion de nuevos derivados de bezilftalazona, basicamente sustituidos y sus sales.

Info

Publication number
ES398949A1
ES398949A1 ES398949A ES398949A ES398949A1 ES 398949 A1 ES398949 A1 ES 398949A1 ES 398949 A ES398949 A ES 398949A ES 398949 A ES398949 A ES 398949A ES 398949 A1 ES398949 A1 ES 398949A1
Authority
ES
Spain
Prior art keywords
formula
combination
see
see formula
residue
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES398949A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ASTA-WERKE AG
Asta Medica GmbH
Original Assignee
ASTA-WERKE AG
Asta Werke AG Chemische Fabrik
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ASTA-WERKE AG, Asta Werke AG Chemische Fabrik filed Critical ASTA-WERKE AG
Publication of ES398949A1 publication Critical patent/ES398949A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
ES398949A 1971-01-22 1972-01-18 Procedimiento para la fabricacion de nuevos derivados de bezilftalazona, basicamente sustituidos y sus sales. Expired ES398949A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH101271A CH572914A5 (es) 1971-01-22 1971-01-22

Publications (1)

Publication Number Publication Date
ES398949A1 true ES398949A1 (es) 1975-06-01

Family

ID=4200381

Family Applications (1)

Application Number Title Priority Date Filing Date
ES398949A Expired ES398949A1 (es) 1971-01-22 1972-01-18 Procedimiento para la fabricacion de nuevos derivados de bezilftalazona, basicamente sustituidos y sus sales.

Country Status (21)

Country Link
AR (1) AR197293A1 (es)
AT (1) AT313288B (es)
AU (1) AU3767472A (es)
BE (1) BE778269A (es)
CA (1) CA1010041A (es)
CH (1) CH572914A5 (es)
DE (1) DE2164058C3 (es)
DK (1) DK136981B (es)
ES (1) ES398949A1 (es)
FI (1) FI53704C (es)
FR (1) FR2122517B1 (es)
GB (1) GB1377231A (es)
HK (1) HK62577A (es)
HU (1) HU163979B (es)
IL (1) IL38496A (es)
NL (1) NL177116C (es)
OA (1) OA04087A (es)
PL (1) PL88930B1 (es)
SE (1) SE404604B (es)
YU (1) YU35361B (es)
ZA (1) ZA718712B (es)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3575135D1 (de) * 1984-09-14 1990-02-08 Asta Pharma Ag Substituierte benzylphthalazinon-derivate.
AU609210B2 (en) * 1987-11-13 1991-04-26 Viatris Gmbh & Co. Kg Azelastine embonate, processes for its preparation and pharmaceutical formulations which contain azelastine embonate as active substance
ATE84968T1 (de) * 1987-11-13 1993-02-15 Asta Medica Ag Azelastin enthaltende arzneimittel zur anwendung in der nase und/oder am auge.
ATE106883T1 (de) * 1987-11-13 1994-06-15 Asta Medica Ag Azelastin-embonat, verfahren zu seiner herstellung und pharmazeutische zubereitungen, die als wirkstoff azelastin-embonat enthalten.
DE3836579A1 (de) * 1987-11-13 1989-05-24 Asta Pharma Ag Azelastin enthaltende arzneimittel zur anwendung in der nase und/oder am auge
DE3912292A1 (de) * 1988-04-20 1989-11-09 Asta Pharma Ag Azelastin enthaltende arzneimittel mit kontrollierter wirkstoffabgabe
US5110814A (en) * 1989-01-11 1992-05-05 Asta Pharma Ag Azelastine and its salts used to combat psoriasis
DE59006184D1 (de) * 1989-05-05 1994-07-28 Asta Medica Ag Salze des Azelastins mit verbesserter Löslichkeit.
DE4207234A1 (de) * 1992-03-07 1993-09-09 Asta Medica Ag Neue aminocarbonsaeure-derivate mit antiallergischer/antiasthmatischer wirkung und verfahren zu deren herstellung
DE4343409C2 (de) * 1993-12-18 1997-03-20 Asta Medica Ag Verbessertes Verfahren zur Herstellung von Hexahydroazepinonen und Hexahydroazepinolen
DE4345224C2 (de) * 1993-12-18 1999-07-01 Asta Medica Ag Verfahren zur Herstellung von Säureadditionssalzen des Azelastins und Flezelastins
GB2389530B (en) 2002-06-14 2007-01-10 Cipla Ltd Pharmaceutical compositions
US8758816B2 (en) 2004-11-24 2014-06-24 Meda Pharmaceuticals Inc. Compositions comprising azelastine and methods of use thereof
US20070020330A1 (en) 2004-11-24 2007-01-25 Medpointe Healthcare Inc. Compositions comprising azelastine and methods of use thereof
TR201820559T4 (tr) 2004-11-24 2019-01-21 Meda Pharmaceuticals Inc Azelastin içeren kompozisyonlar ve bunların kullanım metotları.
AR060535A1 (es) * 2006-04-20 2008-06-25 Glaxo Group Ltd Pirido-piridazinonas y ftalazinonas como antagonistas duales de los receptores h1 y h3 de histamina

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1046625B (de) * 1957-08-15 1958-12-18 Hydrierwerk Rodleben Veb Verfahren zur Herstellung basisch substituierter Phthalazone
GB1100911A (en) * 1963-08-20 1968-01-24 Benger Lab Ltd Phthalazine derivatives
FR1512879A (fr) * 1966-10-28 1968-02-09 Hydrierwerk Rodleben Veb Procédé pour la fabrication de phtalazones avec substituants basiques

Also Published As

Publication number Publication date
ZA718712B (en) 1972-09-27
HK62577A (en) 1977-12-30
FR2122517B1 (es) 1975-08-01
NL177116B (nl) 1985-03-01
DE2164058B2 (de) 1980-10-23
PL88930B1 (es) 1976-10-30
FI53704B (es) 1978-03-31
IL38496A0 (en) 1972-03-28
YU11272A (en) 1980-06-30
DK136981B (da) 1977-12-27
SE404604B (sv) 1978-10-16
BE778269A (fr) 1972-07-19
DK136981C (es) 1978-06-05
DE2164058A1 (de) 1972-07-27
AU3767472A (en) 1973-07-12
HU163979B (es) 1973-12-28
AR197293A1 (es) 1974-03-29
YU35361B (en) 1980-12-31
AT313288B (de) 1974-02-11
OA04087A (fr) 1979-10-30
SU440838A3 (es) 1974-08-25
CH572914A5 (es) 1976-02-27
FR2122517A1 (es) 1972-09-01
CA1010041A (en) 1977-05-10
DE2164058C3 (de) 1981-08-13
NL177116C (nl) 1985-08-01
IL38496A (en) 1975-05-22
FI53704C (fi) 1978-07-10
GB1377231A (en) 1974-12-11
NL7200400A (es) 1972-07-25

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