ES2857743T3 - 1,4-diazepinas fusionadas como degradadores de proteína BET - Google Patents

1,4-diazepinas fusionadas como degradadores de proteína BET Download PDF

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Publication number
ES2857743T3
ES2857743T3 ES17778012T ES17778012T ES2857743T3 ES 2857743 T3 ES2857743 T3 ES 2857743T3 ES 17778012 T ES17778012 T ES 17778012T ES 17778012 T ES17778012 T ES 17778012T ES 2857743 T3 ES2857743 T3 ES 2857743T3
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ES
Spain
Prior art keywords
chlorophenyl
ethynyl
triazolo
diazepin
thieno
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ES17778012T
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English (en)
Spanish (es)
Inventor
Shaomeng Wang
Yang Hu
Chong Qin
Fuming Xu
Jiantao Hu
Weiguo Xiang
Bing Zhou
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University of Michigan System
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University of Michigan System
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
ES17778012T 2016-09-13 2017-09-13 1,4-diazepinas fusionadas como degradadores de proteína BET Active ES2857743T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201662393923P 2016-09-13 2016-09-13
PCT/US2017/051286 WO2018052949A1 (en) 2016-09-13 2017-09-13 Fused 1,4-diazepines as bet protein degraders

Publications (1)

Publication Number Publication Date
ES2857743T3 true ES2857743T3 (es) 2021-09-29

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Family Applications (1)

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ES17778012T Active ES2857743T3 (es) 2016-09-13 2017-09-13 1,4-diazepinas fusionadas como degradadores de proteína BET

Country Status (8)

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US (2) US10975093B2 (enExample)
EP (2) EP3858837A1 (enExample)
JP (1) JP7035027B2 (enExample)
CN (1) CN110072866A (enExample)
AU (1) AU2017326175B2 (enExample)
CA (1) CA3036841A1 (enExample)
ES (1) ES2857743T3 (enExample)
WO (1) WO2018052949A1 (enExample)

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Also Published As

Publication number Publication date
JP7035027B2 (ja) 2022-03-14
AU2017326175B2 (en) 2022-01-27
AU2017326175A1 (en) 2019-04-04
US20190263827A1 (en) 2019-08-29
JP2019526616A (ja) 2019-09-19
US10975093B2 (en) 2021-04-13
EP3512853B1 (en) 2020-12-23
US20220356192A1 (en) 2022-11-10
CA3036841A1 (en) 2018-03-22
WO2018052949A1 (en) 2018-03-22
EP3512853A1 (en) 2019-07-24
EP3858837A1 (en) 2021-08-04
CN110072866A (zh) 2019-07-30

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