ES2693761T3 - Composiciones de péptidos - Google Patents
Composiciones de péptidos Download PDFInfo
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- ES2693761T3 ES2693761T3 ES14719988.9T ES14719988T ES2693761T3 ES 2693761 T3 ES2693761 T3 ES 2693761T3 ES 14719988 T ES14719988 T ES 14719988T ES 2693761 T3 ES2693761 T3 ES 2693761T3
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
- C07K14/68—Melanocyte-stimulating hormone [MSH]
- C07K14/685—Alpha-melanotropin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Endocrinology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Diabetes (AREA)
- Gastroenterology & Hepatology (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Hematology (AREA)
- Reproductive Health (AREA)
- Obesity (AREA)
- Zoology (AREA)
- Toxicology (AREA)
- Immunology (AREA)
- Epidemiology (AREA)
- Emergency Medicine (AREA)
- Child & Adolescent Psychology (AREA)
- Gynecology & Obstetrics (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361790469P | 2013-03-15 | 2013-03-15 | |
| US201361790469P | 2013-03-15 | ||
| PCT/US2014/028590 WO2014144260A1 (en) | 2013-03-15 | 2014-03-14 | Peptide compositions |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2693761T3 true ES2693761T3 (es) | 2018-12-13 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES14719988.9T Active ES2693761T3 (es) | 2013-03-15 | 2014-03-14 | Composiciones de péptidos |
Country Status (10)
| Country | Link |
|---|---|
| US (4) | US10196425B2 (enExample) |
| EP (2) | EP2970388B1 (enExample) |
| JP (4) | JP6622690B2 (enExample) |
| CN (3) | CN118240012A (enExample) |
| AU (6) | AU2014227712B2 (enExample) |
| CA (1) | CA2906694A1 (enExample) |
| ES (1) | ES2693761T3 (enExample) |
| RU (2) | RU2725150C2 (enExample) |
| TR (1) | TR201815173T4 (enExample) |
| WO (1) | WO2014144260A1 (enExample) |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| SMT202100734T1 (it) | 2011-12-29 | 2022-03-21 | Rhythm Pharmaceuticals Inc | Metodo di trattamento di disturbi associati al recettore di melanocortina 4 in portatori eterozigoti |
| JP6538025B2 (ja) | 2013-03-15 | 2019-07-03 | リズム・ファーマシューティカルズ・インコーポレイテッド | 医薬組成物 |
| JP6622690B2 (ja) * | 2013-03-15 | 2019-12-18 | リズム・ファーマシューティカルズ・インコーポレイテッド | ペプチド組成物 |
| WO2016168388A2 (en) | 2015-04-14 | 2016-10-20 | Palatin Technologies, Inc. | Therapies for obesity, diabetes and related indications |
| MX2018003983A (es) * | 2015-09-30 | 2018-11-09 | Rhythm Pharmaceuticals Inc | Metodo de tratamiento de trastornos asociados a la via del receptor de melanocortina-4. |
| WO2018065345A1 (en) * | 2016-10-04 | 2018-04-12 | Dsm Ip Assets B.V. | Melanocortin-1-receptor agonists |
| US20200223889A1 (en) * | 2017-03-15 | 2020-07-16 | Novo Nordisk A/S | Bicyclic Compounds Capable of Binding to Melanocortin 4 Receptor |
| CA3096055A1 (en) | 2018-04-06 | 2019-10-10 | Rhythm Pharmaceuticals, Inc. | Compositions for treating kidney disease |
| WO2020053414A1 (en) * | 2018-09-14 | 2020-03-19 | Novo Nordisk A/S | Bicyclic compounds capable of acting as melanocortin 4 receptor agonists |
| JP2023542985A (ja) * | 2020-09-24 | 2023-10-12 | リズム ファーマシューティカルズ， インコーポレイテッド | メラノコルチン－４受容体経路関連障害の治療方法 |
| CN113209270B (zh) * | 2021-05-17 | 2022-02-22 | 宁波大学 | 丙谷二肽在制备防治急性肝衰竭药物中的应用 |
| CN113332416B (zh) * | 2021-05-17 | 2022-02-22 | 宁波大学 | 丙谷二肽在制备治疗非酒精性脂肪肝药物中的应用 |
| JP2024532294A (ja) * | 2021-08-24 | 2024-09-05 | ザ リージェンツ オブ ザ ユニバーシティ オブ ミシガン | Ｍｃ４ｒアゴニストペプチド |
| CN116789802A (zh) * | 2023-06-25 | 2023-09-22 | 湖北省农业科学院畜牧兽医研究所 | 一种山羊mc4r增强型突变体及其应用 |
| WO2025131101A1 (zh) * | 2023-12-22 | 2025-06-26 | 上海多米瑞生物技术有限公司 | 多肽化合物、其药物组合物及其用途 |
Family Cites Families (31)
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| EP0292291B1 (en) * | 1987-05-22 | 1994-08-10 | University Patents, Inc. | Linear and cyclic analogs of alpha-msh fragments with extraordinary potency |
| US5731408A (en) * | 1995-04-10 | 1998-03-24 | Arizona Board Of Regents On Behalf Of The University Of Arizona | Peptides having potent antagonist and agonist bioactivities at melanocortin receptors |
| GB9827500D0 (en) * | 1998-12-14 | 1999-02-10 | Wapharm Ab | Compounds for control of eating, growth and body weight |
| US7176279B2 (en) * | 2000-06-28 | 2007-02-13 | Palatin Technologies, Inc. | Cyclic peptide compositions and methods for treatment of sexual dysfunction |
| PT1315750E (pt) * | 2000-08-30 | 2007-05-31 | Hoffmann La Roche | Péptidos cíclicos com actividade agonista para o receptor 4 de melanocortina |
| AU2002322466B2 (en) * | 2001-07-11 | 2007-08-30 | Palatin Technologies, Inc. | Linear and cyclic melanocortin receptor-specific peptides |
| US7345144B2 (en) * | 2001-07-11 | 2008-03-18 | Palatin Technologies, Inc. | Cyclic peptides for treatment of cachexia |
| US7342089B2 (en) * | 2001-07-11 | 2008-03-11 | Palatin Technologies, Inc. | Cyclic peptides for treatment for cachexia |
| US7034004B2 (en) * | 2002-05-07 | 2006-04-25 | University Of Florida | Peptides and methods for the control of obesity |
| FR2851563B1 (fr) | 2003-02-26 | 2005-04-22 | Sod Conseils Rech Applic | Nouveaux derives de benzimidazole et d'imidazo-pyridine et leur utilisation en tant que medicament |
| FR2852957B1 (fr) | 2003-03-31 | 2005-06-10 | Sod Conseils Rech Applic | Nouveaux derives d'imidazo-pyridine et leur utilisation en tant que medicament |
| EA200600055A1 (ru) * | 2003-06-19 | 2006-08-25 | Эли Лилли Энд Компани | Агонисты рецептора меланокортина 4 (мк4 ) и их применение |
| WO2005000338A1 (en) * | 2003-06-19 | 2005-01-06 | Eli Lilly And Company | Uses of melanocortin-3 receptor (mc3r) agonist peptides |
| FR2862971B1 (fr) | 2003-11-28 | 2006-03-24 | Sod Conseils Rech Applic | Nouveaux derives de benzimidazole et d'imidazo-pyridine et leur utilisation en tant que medicament |
| US8343031B2 (en) * | 2004-03-23 | 2013-01-01 | Michael Gertner | Obesity treatment systems |
| FR2872165B1 (fr) | 2004-06-24 | 2006-09-22 | Sod Conseils Rech Applic | Nouveaux derives de pyrimido-benzimidazole |
| EP1915168A4 (en) | 2005-07-08 | 2010-03-31 | Ipsen Pharma | LIGANDS OF MELANOCORTIN RECEPTORS |
| ES2663916T3 (es) | 2005-07-08 | 2018-04-17 | Ipsen Pharma | Ligandos de los receptores de la melanocortina |
| CA2689016C (en) | 2007-05-25 | 2014-08-12 | Ipsen Pharma S.A.S. | Melanocortin receptor ligands modified with hydantoin |
| EP2167112A4 (en) | 2007-06-15 | 2012-01-25 | Ipsen Pharma Sas | CYCLIC PEPTIDE MELANOCORTIN RECEPTOR LIGANDS |
| EP2979703B1 (en) | 2007-11-05 | 2018-07-18 | Ipsen Pharma S.A.S. | Use of melanocortins to treat insulin sensitivity |
| AR072072A1 (es) * | 2008-06-09 | 2010-08-04 | Palatin Technologies Inc | Peptidos especificos del receptor de melanocortina para el tratamiento de la obesidad / 669 |
| BRPI1009644B1 (pt) * | 2009-06-08 | 2022-02-08 | Palatin Technologies, Inc | Peptídeo cíclico ou um sal farmaceuticamente aceitável do mesmo, composição farmacêutica e uso da composição farmacêutica |
| UY32690A (es) * | 2009-06-08 | 2011-01-31 | Astrazeneca Ab | Péptidos específicos para receptores de melanocortina |
| MX2012001513A (es) | 2009-08-05 | 2012-05-22 | Ipsen Pharma Sas | Uso de melanocortinas para tratar la dislipidemia. |
| JP5486690B2 (ja) | 2009-11-16 | 2014-05-07 | イプセン ファルマ ソシエテ パール アクシオン サンプリフィエ | メラノコルチン受容体リガンドの医薬組成物 |
| WO2011060355A1 (en) | 2009-11-16 | 2011-05-19 | Ipsen Pharma S.A.S | Process for the synthesis of ac-arg-cyclo(cys-d-ala-his-d-phe-arg-trp-cys)-nh2 |
| KR102038677B1 (ko) | 2011-06-14 | 2019-10-30 | 입센 파마 에스.에이.에스 | 활성 성분으로 멜라노코르틴 수용체 리간드를 함유하는 지속-방출형 조성물 |
| EP2705835A1 (en) | 2012-06-08 | 2014-03-12 | Ipsen Pharma S.A.S. | Aqueous gelling compositions of soluble active pharmaceutical peptides providing modified release |
| JP6622690B2 (ja) * | 2013-03-15 | 2019-12-18 | リズム・ファーマシューティカルズ・インコーポレイテッド | ペプチド組成物 |
| JP6538025B2 (ja) * | 2013-03-15 | 2019-07-03 | リズム・ファーマシューティカルズ・インコーポレイテッド | 医薬組成物 |
-
2014
- 2014-03-14 JP JP2016502840A patent/JP6622690B2/ja active Active
- 2014-03-14 US US14/775,916 patent/US10196425B2/en active Active
- 2014-03-14 CA CA2906694A patent/CA2906694A1/en active Pending
- 2014-03-14 AU AU2014227712A patent/AU2014227712B2/en active Active
- 2014-03-14 CN CN202410043141.5A patent/CN118240012A/zh active Pending
- 2014-03-14 TR TR2018/15173T patent/TR201815173T4/tr unknown
- 2014-03-14 RU RU2015145593A patent/RU2725150C2/ru active
- 2014-03-14 CN CN202410043113.3A patent/CN118271400A/zh active Pending
- 2014-03-14 EP EP14719988.9A patent/EP2970388B1/en active Active
- 2014-03-14 RU RU2020120797A patent/RU2020120797A/ru unknown
- 2014-03-14 WO PCT/US2014/028590 patent/WO2014144260A1/en not_active Ceased
- 2014-03-14 EP EP18183527.3A patent/EP3450449A3/en active Pending
- 2014-03-14 ES ES14719988.9T patent/ES2693761T3/es active Active
- 2014-03-14 CN CN201480026843.7A patent/CN105492456B/zh active Active
-
2018
- 2018-10-30 AU AU2018256493A patent/AU2018256493A1/en not_active Abandoned
- 2018-12-11 US US16/216,116 patent/US10858399B2/en active Active
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2019
- 2019-06-19 JP JP2019113626A patent/JP7046871B2/ja active Active
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2020
- 2020-05-22 AU AU2020203353A patent/AU2020203353A1/en not_active Abandoned
- 2020-10-26 US US17/080,293 patent/US12077612B2/en active Active
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2021
- 2021-11-18 AU AU2021269411A patent/AU2021269411A1/en not_active Abandoned
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2022
- 2022-03-24 JP JP2022048719A patent/JP7654587B2/ja active Active
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2024
- 2024-01-29 AU AU2024200528A patent/AU2024200528A1/en not_active Abandoned
- 2024-07-24 US US18/782,986 patent/US20250188124A1/en active Pending
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2025
- 2025-03-19 JP JP2025045947A patent/JP2025102830A/ja active Pending
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2026
- 2026-05-27 AU AU2026204118A patent/AU2026204118A1/en active Pending
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