ES2589558T3 - Derivados de pirimidin pirazolilo - Google Patents

Derivados de pirimidin pirazolilo Download PDF

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Publication number
ES2589558T3
ES2589558T3 ES13737134.0T ES13737134T ES2589558T3 ES 2589558 T3 ES2589558 T3 ES 2589558T3 ES 13737134 T ES13737134 T ES 13737134T ES 2589558 T3 ES2589558 T3 ES 2589558T3
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Stefano Crosignani
Catherine Jorand-Lebrun
Patrick Gerber
Mathilde Muzerelle
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Ares Trading SA
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Ares Trading SA
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    • C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
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    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
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