CA2878621C - Pyrimidine pyrazolyl derivatives - Google Patents

Pyrimidine pyrazolyl derivatives Download PDF

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Publication number
CA2878621C
CA2878621C CA2878621A CA2878621A CA2878621C CA 2878621 C CA2878621 C CA 2878621C CA 2878621 A CA2878621 A CA 2878621A CA 2878621 A CA2878621 A CA 2878621A CA 2878621 C CA2878621 C CA 2878621C
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pyrazol
mmol
hplc
esi
denotes
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French (fr)
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CA2878621A1 (en
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Stefano Crosignani
Catherine Jorand-Lebrun
Patrick Gerber
Mathilde Muzerelle
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Ares Trading SA
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Ares Trading SA
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    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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