ES2435997T3 - Aminopirimidinas útiles como inhibidores de las proteínas cinasas - Google Patents
Aminopirimidinas útiles como inhibidores de las proteínas cinasas Download PDFInfo
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- ES2435997T3 ES2435997T3 ES08731830T ES08731830T ES2435997T3 ES 2435997 T3 ES2435997 T3 ES 2435997T3 ES 08731830 T ES08731830 T ES 08731830T ES 08731830 T ES08731830 T ES 08731830T ES 2435997 T3 ES2435997 T3 ES 2435997T3
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- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
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- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
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| US95302007P | 2007-07-31 | 2007-07-31 | |
| US953020P | 2007-07-31 | ||
| PCT/US2008/056423 WO2008112642A1 (en) | 2007-03-09 | 2008-03-10 | Aminopyrimidines useful as inhibitors of protein kinases |
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| AU2008257044A1 (en) | 2007-05-24 | 2008-12-04 | Vertex Pharmaceuticals Incorporated | Thiazoles and pyrazoles useful as kinase inhibitors |
| AR067762A1 (es) * | 2007-07-31 | 2009-10-21 | Vertex Pharma | Proceso para preparar 5-fluoro-1h-pirazolo (3,4-b) piridin-3-amina y derivados de la misma |
| MX384179B (es) | 2009-03-20 | 2025-03-14 | Vertex Pharma | Proceso para producir moduladores del regulador de conductancia transmembrana de fibrosis quística. |
-
2008
- 2008-03-10 WO PCT/US2008/056423 patent/WO2008112642A1/en not_active Ceased
- 2008-03-10 MX MX2009009590A patent/MX2009009590A/es active IP Right Grant
- 2008-03-10 EP EP08731830.9A patent/EP2134707B1/en not_active Not-in-force
- 2008-03-10 JP JP2009552927A patent/JP5520057B2/ja not_active Expired - Fee Related
- 2008-03-10 AU AU2008226457A patent/AU2008226457B2/en not_active Ceased
- 2008-03-10 CA CA002679884A patent/CA2679884A1/en not_active Abandoned
- 2008-03-10 CN CN200880012693.9A patent/CN101663295B/zh not_active Expired - Fee Related
- 2008-03-10 ES ES08731830T patent/ES2435997T3/es active Active
- 2008-03-10 NZ NZ579446A patent/NZ579446A/en not_active IP Right Cessation
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2010
- 2010-06-02 US US12/791,976 patent/US8664219B2/en not_active Expired - Fee Related
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2014
- 2014-01-15 US US14/155,624 patent/US20140194444A1/en not_active Abandoned
- 2014-06-18 AU AU2014203289A patent/AU2014203289A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| NZ579446A (en) | 2012-02-24 |
| AU2008226457A1 (en) | 2008-09-18 |
| CN101663295B (zh) | 2014-11-05 |
| US8664219B2 (en) | 2014-03-04 |
| JP5520057B2 (ja) | 2014-06-11 |
| US20110020376A1 (en) | 2011-01-27 |
| CA2679884A1 (en) | 2008-09-18 |
| EP2134707B1 (en) | 2013-09-11 |
| US20140194444A1 (en) | 2014-07-10 |
| AU2014203289A1 (en) | 2014-07-17 |
| CN101663295A (zh) | 2010-03-03 |
| MX2009009590A (es) | 2009-11-10 |
| WO2008112642A1 (en) | 2008-09-18 |
| EP2134707A1 (en) | 2009-12-23 |
| JP2010520886A (ja) | 2010-06-17 |
| AU2008226457B2 (en) | 2014-03-20 |
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