ES2428543T3 - Compuestos de tiofenopirazolopirimidina - Google Patents
Compuestos de tiofenopirazolopirimidina Download PDFInfo
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- ES2428543T3 ES2428543T3 ES07814842T ES07814842T ES2428543T3 ES 2428543 T3 ES2428543 T3 ES 2428543T3 ES 07814842 T ES07814842 T ES 07814842T ES 07814842 T ES07814842 T ES 07814842T ES 2428543 T3 ES2428543 T3 ES 2428543T3
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Classifications
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- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
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- Public Health (AREA)
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- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
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- Pulmonology (AREA)
- Cardiology (AREA)
- Pregnancy & Childbirth (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US82627306P | 2006-09-20 | 2006-09-20 | |
| US826273P | 2006-09-20 | ||
| PCT/US2007/078352 WO2008036541A1 (en) | 2006-09-20 | 2007-09-13 | Thiophene pyrazolopyrimidine compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2428543T3 true ES2428543T3 (es) | 2013-11-08 |
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| ES07814842T Active ES2428543T3 (es) | 2006-09-20 | 2007-09-13 | Compuestos de tiofenopirazolopirimidina |
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| EP (1) | EP2076515B1 (cg-RX-API-DMAC7.html) |
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| BR (1) | BRPI0717070A2 (cg-RX-API-DMAC7.html) |
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| EP2025674A1 (de) | 2007-08-15 | 2009-02-18 | sanofi-aventis | Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| US9029411B2 (en) | 2008-01-25 | 2015-05-12 | Millennium Pharmaceuticals, Inc. | Thiophenes and uses thereof |
| US8796314B2 (en) | 2009-01-30 | 2014-08-05 | Millennium Pharmaceuticals, Inc. | Heteroaryls and uses thereof |
| US9090601B2 (en) | 2009-01-30 | 2015-07-28 | Millennium Pharmaceuticals, Inc. | Thiazole derivatives |
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Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR0173172B1 (ko) | 1992-12-17 | 1999-02-01 | 알렌 제이. 스피겔 | Crf 길항제로서의 피롤로피리미딘 |
| KR100421626B1 (ko) * | 1996-02-07 | 2004-05-20 | 뉴로크린 바이오사이언시즈 인코퍼레이티드 | Crf수용체에대한길항제로서의피라졸로피리미딘 |
| DK0915880T3 (da) | 1996-07-24 | 2008-02-11 | Bristol Myers Squibb Pharma Co | Azolotriaziner og pyrimidiner |
| JP3621706B2 (ja) | 1996-08-28 | 2005-02-16 | ファイザー・インク | 置換された６，５―ヘテロ―二環式誘導体 |
| US6476038B1 (en) * | 1999-09-30 | 2002-11-05 | Neurogen Corporation | Amino substituted pyrazolo[1,5,-a]-1,5-pyrimidines and pyrazolo[1,5-a]-1,3,5-triazines |
| EP1697374B1 (en) * | 2003-12-22 | 2012-08-29 | SmithKline Beecham (Cork) Limited | Crf receptor antagonists and methods relating thereto |
| CN101142217B (zh) * | 2005-03-21 | 2010-12-08 | 伊莱利利公司 | 咪唑并哒嗪化合物 |
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- 2007-09-13 CA CA2662000A patent/CA2662000C/en not_active Expired - Fee Related
- 2007-09-13 KR KR1020097005694A patent/KR101088196B1/ko not_active Expired - Fee Related
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- 2007-09-13 BR BRPI0717070-0A2A patent/BRPI0717070A2/pt not_active IP Right Cessation
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| US8110580B2 (en) | 2012-02-07 |
| KR20090053921A (ko) | 2009-05-28 |
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| EA200970302A1 (ru) | 2009-10-30 |
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| AU2007297481A1 (en) | 2008-03-27 |
| JP5184536B2 (ja) | 2013-04-17 |
| EA016056B1 (ru) | 2012-01-30 |
| WO2008036541A1 (en) | 2008-03-27 |
| BRPI0717070A2 (pt) | 2013-09-24 |
| EP2076515A1 (en) | 2009-07-08 |
| US20100022560A1 (en) | 2010-01-28 |
| CA2662000C (en) | 2013-01-08 |
| CN101516886A (zh) | 2009-08-26 |
| CA2662000A1 (en) | 2008-03-27 |
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