ES2202189T3 - Procedimiento para preparar pirazoles sustituidos. - Google Patents

Procedimiento para preparar pirazoles sustituidos.

Info

Publication number
ES2202189T3
ES2202189T3 ES00976715T ES00976715T ES2202189T3 ES 2202189 T3 ES2202189 T3 ES 2202189T3 ES 00976715 T ES00976715 T ES 00976715T ES 00976715 T ES00976715 T ES 00976715T ES 2202189 T3 ES2202189 T3 ES 2202189T3
Authority
ES
Spain
Prior art keywords
alkyl
amino
optionally
completely halogenated
chosen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES00976715T
Other languages
English (en)
Spanish (es)
Inventor
James A. Baron
Vittorio Farina
Nizar Haddad
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Pharmaceuticals Inc
Original Assignee
Boehringer Ingelheim Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharmaceuticals Inc filed Critical Boehringer Ingelheim Pharmaceuticals Inc
Application granted granted Critical
Publication of ES2202189T3 publication Critical patent/ES2202189T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ES00976715T 1999-10-29 2000-10-27 Procedimiento para preparar pirazoles sustituidos. Expired - Lifetime ES2202189T3 (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US16247699P 1999-10-29 1999-10-29
US162476P 1999-10-29
US19265100P 2000-03-28 2000-03-28
US192651P 2000-03-28

Publications (1)

Publication Number Publication Date
ES2202189T3 true ES2202189T3 (es) 2004-04-01

Family

ID=26858795

Family Applications (1)

Application Number Title Priority Date Filing Date
ES00976715T Expired - Lifetime ES2202189T3 (es) 1999-10-29 2000-10-27 Procedimiento para preparar pirazoles sustituidos.

Country Status (11)

Country Link
EP (1) EP1235810B1 (enExample)
JP (1) JP4861585B2 (enExample)
AT (1) ATE244704T1 (enExample)
AU (1) AU1445001A (enExample)
CA (1) CA2387762C (enExample)
DE (1) DE60003846T2 (enExample)
DK (1) DK1235810T3 (enExample)
ES (1) ES2202189T3 (enExample)
MX (1) MXPA02004004A (enExample)
PT (1) PT1235810E (enExample)
WO (1) WO2001032627A1 (enExample)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6407238B1 (en) 1999-10-29 2002-06-18 Boehringer Ingelheim Pharmaceuticals, Inc. Process of making substituted pyrazoles
US6492529B1 (en) 2000-01-18 2002-12-10 Boehringer Ingelheim Pharmaceuticals, Inc. Bis pyrazole-1H-pyrazole intermediates and their synthesis
MXPA03006749A (es) 2001-02-15 2004-05-31 Boehringer Ingelheim Pharma Proceso para la sintesis de compuestos de urea sustituidos con heteroarilo, utiles como agentes antiinflamatorios.
DE10315573A1 (de) 2003-04-05 2004-10-14 Merck Patent Gmbh Substituierte Pyrazole
DE10315571A1 (de) 2003-04-05 2004-10-14 Merck Patent Gmbh Pyrazolverbindungen
DE10315569A1 (de) * 2003-04-05 2004-10-14 Merck Patent Gmbh Substituierte Pyrazolverbindungen
US7714127B2 (en) 2005-10-06 2010-05-11 Boehringer Ingelheim Pharmaceuticals, Inc. Process for making heteroaryl amine intermediate compounds
EP2135865A1 (de) 2008-06-17 2009-12-23 Bayer CropScience AG Substituierte 1-(Diazinyl) pyrazol-4-yl-essigsäuren, Verfahren zu deren Herstellung und deren Verwendung als Herbizide und Pflanzenwachstumsregulatoren
EP2194052A1 (de) 2008-12-06 2010-06-09 Bayer CropScience AG Substituierte 1-(Thiazolyl)- und 1-(Isothiazolyl)pyrazol-4-yl-essigsäuren, Verfahren zu deren Herstellung und deren Verwendung als Herbizide und Pflanzenwachstumsregulatoren
WO2011073098A1 (de) 2009-12-15 2011-06-23 Bayer Cropscience Ag 1-(heteroaryl)-pyrazol-4-yl-essigsäuren, verfahren zu deren herstellung und deren verwendung als herbizide und pflanzenwachstumsregulatoren
AU2019387370A1 (en) 2018-11-30 2021-06-10 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4314851A1 (de) * 1993-05-05 1994-11-10 Huels Chemische Werke Ag Verfahren zur Herstellung von 3-Amino-5-methylpyrazol
US5698708A (en) * 1996-06-20 1997-12-16 Monsanto Company Preparation of substituted 3-aryl-5-haloalkyl-pyrazoles having herbicidal activity
JP2000512656A (ja) * 1996-06-20 2000-09-26 モンサント・カンパニー 除草剤活性を有する置換された３―アリール―５―ハロアルキル―ピラゾールの製法
EP1028953A1 (en) * 1997-11-03 2000-08-23 Boehringer Ingelheim Pharmaceuticals Inc. Aromatic heterocyclic compounds as anti-inflammatory agents

Also Published As

Publication number Publication date
WO2001032627A8 (en) 2002-01-24
ATE244704T1 (de) 2003-07-15
CA2387762A1 (en) 2001-05-10
DK1235810T3 (da) 2003-11-03
JP2003513076A (ja) 2003-04-08
EP1235810A1 (en) 2002-09-04
WO2001032627A1 (en) 2001-05-10
CA2387762C (en) 2008-07-29
MXPA02004004A (es) 2002-10-23
DE60003846D1 (de) 2003-08-14
DE60003846T2 (de) 2004-06-03
EP1235810B1 (en) 2003-07-09
AU1445001A (en) 2001-05-14
PT1235810E (pt) 2003-11-28
JP4861585B2 (ja) 2012-01-25

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