ATE244704T1 - Verfahren zur herstellung von substituierten pyrazolen - Google Patents
Verfahren zur herstellung von substituierten pyrazolenInfo
- Publication number
- ATE244704T1 ATE244704T1 AT00976715T AT00976715T ATE244704T1 AT E244704 T1 ATE244704 T1 AT E244704T1 AT 00976715 T AT00976715 T AT 00976715T AT 00976715 T AT00976715 T AT 00976715T AT E244704 T1 ATE244704 T1 AT E244704T1
- Authority
- AT
- Austria
- Prior art keywords
- substituted pyrazoles
- producing substituted
- formula
- making
- pyrazoles
- Prior art date
Links
- 150000003217 pyrazoles Chemical class 0.000 title abstract 3
- 238000004519 manufacturing process Methods 0.000 title 1
- QYCSNMDOZNUZIT-UHFFFAOYSA-N benzhydrylidenehydrazine Chemical class C=1C=CC=CC=1C(=NN)C1=CC=CC=C1 QYCSNMDOZNUZIT-UHFFFAOYSA-N 0.000 abstract 2
- 239000002253 acid Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
- 239000000758 substrate Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Urology & Nephrology (AREA)
- Heart & Thoracic Surgery (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US16247699P | 1999-10-29 | 1999-10-29 | |
| US19265100P | 2000-03-28 | 2000-03-28 | |
| PCT/US2000/029891 WO2001032627A1 (en) | 1999-10-29 | 2000-10-27 | Process of making substituted pyrazoles |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE244704T1 true ATE244704T1 (de) | 2003-07-15 |
Family
ID=26858795
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT00976715T ATE244704T1 (de) | 1999-10-29 | 2000-10-27 | Verfahren zur herstellung von substituierten pyrazolen |
Country Status (11)
| Country | Link |
|---|---|
| EP (1) | EP1235810B1 (enExample) |
| JP (1) | JP4861585B2 (enExample) |
| AT (1) | ATE244704T1 (enExample) |
| AU (1) | AU1445001A (enExample) |
| CA (1) | CA2387762C (enExample) |
| DE (1) | DE60003846T2 (enExample) |
| DK (1) | DK1235810T3 (enExample) |
| ES (1) | ES2202189T3 (enExample) |
| MX (1) | MXPA02004004A (enExample) |
| PT (1) | PT1235810E (enExample) |
| WO (1) | WO2001032627A1 (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6407238B1 (en) | 1999-10-29 | 2002-06-18 | Boehringer Ingelheim Pharmaceuticals, Inc. | Process of making substituted pyrazoles |
| US6492529B1 (en) | 2000-01-18 | 2002-12-10 | Boehringer Ingelheim Pharmaceuticals, Inc. | Bis pyrazole-1H-pyrazole intermediates and their synthesis |
| MXPA03006749A (es) | 2001-02-15 | 2004-05-31 | Boehringer Ingelheim Pharma | Proceso para la sintesis de compuestos de urea sustituidos con heteroarilo, utiles como agentes antiinflamatorios. |
| DE10315573A1 (de) | 2003-04-05 | 2004-10-14 | Merck Patent Gmbh | Substituierte Pyrazole |
| DE10315571A1 (de) | 2003-04-05 | 2004-10-14 | Merck Patent Gmbh | Pyrazolverbindungen |
| DE10315569A1 (de) * | 2003-04-05 | 2004-10-14 | Merck Patent Gmbh | Substituierte Pyrazolverbindungen |
| US7714127B2 (en) | 2005-10-06 | 2010-05-11 | Boehringer Ingelheim Pharmaceuticals, Inc. | Process for making heteroaryl amine intermediate compounds |
| EP2135865A1 (de) | 2008-06-17 | 2009-12-23 | Bayer CropScience AG | Substituierte 1-(Diazinyl) pyrazol-4-yl-essigsäuren, Verfahren zu deren Herstellung und deren Verwendung als Herbizide und Pflanzenwachstumsregulatoren |
| EP2194052A1 (de) | 2008-12-06 | 2010-06-09 | Bayer CropScience AG | Substituierte 1-(Thiazolyl)- und 1-(Isothiazolyl)pyrazol-4-yl-essigsäuren, Verfahren zu deren Herstellung und deren Verwendung als Herbizide und Pflanzenwachstumsregulatoren |
| WO2011073098A1 (de) | 2009-12-15 | 2011-06-23 | Bayer Cropscience Ag | 1-(heteroaryl)-pyrazol-4-yl-essigsäuren, verfahren zu deren herstellung und deren verwendung als herbizide und pflanzenwachstumsregulatoren |
| AU2019387370A1 (en) | 2018-11-30 | 2021-06-10 | Nuvation Bio Inc. | Pyrrole and pyrazole compounds and methods of use thereof |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4314851A1 (de) * | 1993-05-05 | 1994-11-10 | Huels Chemische Werke Ag | Verfahren zur Herstellung von 3-Amino-5-methylpyrazol |
| US5698708A (en) * | 1996-06-20 | 1997-12-16 | Monsanto Company | Preparation of substituted 3-aryl-5-haloalkyl-pyrazoles having herbicidal activity |
| JP2000512656A (ja) * | 1996-06-20 | 2000-09-26 | モンサント・カンパニー | 除草剤活性を有する置換された3―アリール―5―ハロアルキル―ピラゾールの製法 |
| EP1028953A1 (en) * | 1997-11-03 | 2000-08-23 | Boehringer Ingelheim Pharmaceuticals Inc. | Aromatic heterocyclic compounds as anti-inflammatory agents |
-
2000
- 2000-10-27 AT AT00976715T patent/ATE244704T1/de active
- 2000-10-27 ES ES00976715T patent/ES2202189T3/es not_active Expired - Lifetime
- 2000-10-27 EP EP00976715A patent/EP1235810B1/en not_active Expired - Lifetime
- 2000-10-27 DK DK00976715T patent/DK1235810T3/da active
- 2000-10-27 WO PCT/US2000/029891 patent/WO2001032627A1/en not_active Ceased
- 2000-10-27 AU AU14450/01A patent/AU1445001A/en not_active Abandoned
- 2000-10-27 MX MXPA02004004A patent/MXPA02004004A/es active IP Right Grant
- 2000-10-27 CA CA002387762A patent/CA2387762C/en not_active Expired - Fee Related
- 2000-10-27 DE DE60003846T patent/DE60003846T2/de not_active Expired - Lifetime
- 2000-10-27 JP JP2001534779A patent/JP4861585B2/ja not_active Expired - Fee Related
- 2000-10-27 PT PT00976715T patent/PT1235810E/pt unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2001032627A8 (en) | 2002-01-24 |
| CA2387762A1 (en) | 2001-05-10 |
| DK1235810T3 (da) | 2003-11-03 |
| ES2202189T3 (es) | 2004-04-01 |
| JP2003513076A (ja) | 2003-04-08 |
| EP1235810A1 (en) | 2002-09-04 |
| WO2001032627A1 (en) | 2001-05-10 |
| CA2387762C (en) | 2008-07-29 |
| MXPA02004004A (es) | 2002-10-23 |
| DE60003846D1 (de) | 2003-08-14 |
| DE60003846T2 (de) | 2004-06-03 |
| EP1235810B1 (en) | 2003-07-09 |
| AU1445001A (en) | 2001-05-14 |
| PT1235810E (pt) | 2003-11-28 |
| JP4861585B2 (ja) | 2012-01-25 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DE69310410D1 (de) | Verfahren zur Herstellung von Innenständern für elektromagnetische Pumpen | |
| ATE501113T1 (de) | Verfahren zur herstellung von 2-halogenacyl-3- amino-acrylsäure- derivaten | |
| DE69631305D1 (de) | Verfahren zur Herstellung von Polymilchsäure | |
| DE19681532T1 (de) | Verfahren zur Herstellung von L-Glutaminsäure durch Fermentation | |
| DE69619030D1 (de) | Verfahren zur Herstellung von Essigsäure durch Carbonylierung | |
| ATE244704T1 (de) | Verfahren zur herstellung von substituierten pyrazolen | |
| DE59405805D1 (de) | Verfahren zur herstellung von pyrazol und dessen derivaten | |
| TR28332A (tr) | Arilasetik asit türevleri. | |
| ATE224379T1 (de) | Ein verfahren zur herstellung von 1,4,7,10- tetraazacyclododecan-1,4,7-triessigsäure und deren derivaten | |
| ATE359272T1 (de) | Verfahren zur herstellung von 3-hydroxy-n-1,6- | |
| ATE207883T1 (de) | Phenylessigsäurederivate, verfahren und zwischenprodukte zu ihrer herstellung und ihre verwendung als schädlingsbekämpfungsmittel und fungizide | |
| ATE197150T1 (de) | Verfahren zur herstellung von dihydroxypyrimidin- derivaten | |
| ATE206407T1 (de) | Verfahren zur herstellung von hiv proteasinhibitoren | |
| DE69808771D1 (de) | Ein verfahren zur herstellung von tetraaza makrocyclen | |
| DE69404454D1 (de) | Verfahren zur herstellung von aminomethanphosphonsäure | |
| ATE271057T1 (de) | Verfahren zur herstellung von alendron-säure | |
| DE69926223D1 (de) | Verfahren zur herstellung von zwischenprodukten | |
| ATE248141T1 (de) | Verfahren zur herstellung von (r) und (s)- aminocarnitin und deren derivative aus d- und l- aspargin säure | |
| DE69508864D1 (de) | Verfahren zur Herstellung von Pikrinsaüre | |
| DE59803194D1 (de) | Verfahren zur herstellung von 1,3-disubstituierten 2-nitroguanidinen | |
| DE60031315D1 (de) | Verfahren zur Herstellung von Derivaten von i(1,5-Diaryl)pyrazol-3-ylöpropansäure | |
| DE69821763D1 (de) | Verfahren zur herstellung von 2-alkylthio-substituierten benzoesäurederivaten | |
| DE69601277D1 (de) | Verfahren zur Herstellung von Fumarsäure | |
| DE69926642D1 (de) | Verfahren zur herstellung von n-geschützten azetidin-2-carbonsäuren | |
| DE60229261D1 (de) | Verfahren zur herstellung von säureanhydrid |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification |
Ref document number: 1235810 Country of ref document: EP |