ES2140778T3 - Procedimiento para la preparacion de compuestos de 2-cianoimidazol 1-sustituidos. - Google Patents
Procedimiento para la preparacion de compuestos de 2-cianoimidazol 1-sustituidos.Info
- Publication number
- ES2140778T3 ES2140778T3 ES96118827T ES96118827T ES2140778T3 ES 2140778 T3 ES2140778 T3 ES 2140778T3 ES 96118827 T ES96118827 T ES 96118827T ES 96118827 T ES96118827 T ES 96118827T ES 2140778 T3 ES2140778 T3 ES 2140778T3
- Authority
- ES
- Spain
- Prior art keywords
- cianoimidazole
- procedure
- preparation
- formula
- compound represented
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
- C07C251/32—Oximes
- C07C251/34—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
- C07C251/48—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atom of at least one of the oxyimino groups bound to a carbon atom of a six-membered aromatic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/63—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
Abstract
SE DESCRIBE UN PROCEDIMIENTO DE PRODUCCION DE COMPUESTOS DE 2CIANOIMIDAZOL SUSTITUIDOS EN POSICION 1, QUE COMPRENDE UNA REACCION DE SULFAMOILACION Y UNA REACCION DE ISOMERIZACION DE UN COMPUESTO 2-CIANOIMIDAZOL, REPRESENTADO POR LA FORMULA (II) Y UN COMPUESTO REPRESENTADO POR LA FORMULA (III), EN PRESENCIA DE AL MENOS UNA BASE, SELECCIONADA ENTRE CARBONATOS DE METALES ALCALINOS Y BICARBONATOS DE METALES ALCALINOS, Y DE UN SOLVENTE POLAR, PARA PRODUCIR UN COMPUESTO DE 2-CIANOIMIDAZOL SUSTITUIDO EN POSICION 1, REPRESENTADO POR LA FORMULA (I-B). LOS SUSTITUYENTES DE LAS CITADAS FORMULAS SE DEFINEN ESPECIFICAMENTE EN LA DESCRIPCION.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP24216494 | 1994-09-08 | ||
JP27032194 | 1994-10-07 | ||
JP28926794 | 1994-10-28 | ||
JP5362995 | 1995-02-16 |
Publications (1)
Publication Number | Publication Date |
---|---|
ES2140778T3 true ES2140778T3 (es) | 2000-03-01 |
Family
ID=27462936
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES96118827T Expired - Lifetime ES2140778T3 (es) | 1994-09-08 | 1995-09-06 | Procedimiento para la preparacion de compuestos de 2-cianoimidazol 1-sustituidos. |
Country Status (9)
Country | Link |
---|---|
US (1) | US5869683A (es) |
EP (2) | EP0705823A1 (es) |
KR (1) | KR100368510B1 (es) |
AT (1) | ATE187168T1 (es) |
CA (1) | CA2157753C (es) |
DE (1) | DE69513657T2 (es) |
DK (1) | DK0765872T3 (es) |
ES (1) | ES2140778T3 (es) |
GR (1) | GR3032745T3 (es) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20050203025A1 (en) * | 1998-05-05 | 2005-09-15 | Adherex Technologies, Inc. | Compounds and methods for modulating nonclassical cadherin-mediated functions |
US7481999B2 (en) * | 1998-05-05 | 2009-01-27 | Adherex Technologies, Inc. | Compounds and methods for modulating OB-cadherin-mediated function |
US6680175B2 (en) * | 1998-05-05 | 2004-01-20 | Adherex Technologies, Inc. | Methods for diagnosing and evaluating cancer |
WO2000075094A2 (en) * | 1999-06-03 | 2000-12-14 | Ishihara Sangyo Kaisha, Ltd. | Method for producing a halogenated acetophenone |
AU2003298475A1 (en) * | 2002-11-14 | 2004-06-18 | Adherex Technologies, Inc. | Compounds and methods for modulating desmosomal and atypical cadherin-mediated cell adhesion |
ITMI20051558A1 (it) | 2005-08-09 | 2007-02-10 | Isagro Spa | Miscele e-o composizioni sinergiche cin elevata attivita'fungicida |
CN101312649B (zh) | 2005-11-22 | 2012-03-28 | 石原产业株式会社 | 农业园艺用杀菌剂组合物以及植物病害的防除方法 |
CN102424671B (zh) * | 2011-11-04 | 2014-05-14 | 西安近代化学研究所 | 4-氯-2-氰基-1-二甲基氨基磺酰基-5-(4-甲基苯基)咪唑的合成方法 |
CN103936678B (zh) * | 2014-04-23 | 2016-04-27 | 西安近代化学研究所 | 一种4-氯-2-氰基-n,n-二甲基-5-(4’-甲基苯基)-1h-咪唑-1-磺酰胺的合成方法 |
CN104292166B (zh) * | 2014-10-14 | 2016-04-27 | 西安近代化学研究所 | 4-氯-2-氰基-n,n-二甲基-5-对甲苯基咪唑-1-磺酰胺合成方法 |
CN107118160B (zh) * | 2016-12-07 | 2019-06-28 | 盐城辉煌化工有限公司 | 一种2-氰基-4-(对甲苯基)-5-氯-1h-咪唑的制备工艺 |
US10968182B2 (en) | 2017-02-23 | 2021-04-06 | Adama Makhteshim Ltd. | Process for the preparation of 2-cyanoimidazole compounds |
CN106986830A (zh) * | 2017-05-11 | 2017-07-28 | 蚌埠中实化学技术有限公司 | 4‑氯‑2‑氰基‑1‑二甲基氨基磺酰基‑5‑(4‑甲基苯基)咪唑的合成方法 |
CN107602477A (zh) * | 2017-10-25 | 2018-01-19 | 西安近代化学研究所 | 一种氰霜唑原药的精制方法 |
CN109400534B (zh) * | 2018-10-17 | 2020-11-03 | 兰博尔开封科技有限公司 | 一种1-羟基-4-(4′-甲基苯基)-2-甲肟咪唑-3-氧化物的生产工艺 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5219B1 (es) | 1968-08-15 | 1977-01-05 | ||
US4441916A (en) * | 1981-10-19 | 1984-04-10 | Stauffer Chemical Company | Haloalkyloxime herbicidal antidotes |
CA1339133C (en) | 1987-03-13 | 1997-07-29 | Rikuo Nasu | Imidazole compounds and biocidal composition comprising the same for controlling harmful organisms |
MY129863A (en) * | 1988-03-11 | 2007-05-31 | Ishihara Sangyo Kaisha | Biocidal composition |
JP2879164B2 (ja) | 1990-06-28 | 1999-04-05 | 石原産業株式会社 | 置換2―シアノイミダゾール系化合物の製造方法 |
JPH04120063A (ja) | 1990-09-07 | 1992-04-21 | Ishihara Sangyo Kaisha Ltd | イミダゾール系化合物の分離方法 |
DE69401486T2 (de) * | 1993-11-12 | 1997-04-30 | Ishihara Sangyo Kaisha | Verfahren zur Herstellung 2-cyanoimidazol Derivate |
-
1995
- 1995-09-06 EP EP95306229A patent/EP0705823A1/en not_active Withdrawn
- 1995-09-06 AT AT96118827T patent/ATE187168T1/de active
- 1995-09-06 DK DK96118827T patent/DK0765872T3/da active
- 1995-09-06 DE DE69513657T patent/DE69513657T2/de not_active Expired - Lifetime
- 1995-09-06 EP EP96118827A patent/EP0765872B1/en not_active Expired - Lifetime
- 1995-09-06 KR KR1019950029085A patent/KR100368510B1/ko not_active IP Right Cessation
- 1995-09-06 ES ES96118827T patent/ES2140778T3/es not_active Expired - Lifetime
- 1995-09-07 CA CA002157753A patent/CA2157753C/en not_active Expired - Fee Related
-
1997
- 1997-11-03 US US08/962,648 patent/US5869683A/en not_active Expired - Lifetime
-
2000
- 2000-02-23 GR GR20000400445T patent/GR3032745T3/el unknown
Also Published As
Publication number | Publication date |
---|---|
ATE187168T1 (de) | 1999-12-15 |
KR100368510B1 (ko) | 2003-04-23 |
DK0765872T3 (da) | 2000-05-22 |
EP0705823A1 (en) | 1996-04-10 |
EP0765872A3 (es) | 1997-04-09 |
EP0765872A2 (en) | 1997-04-02 |
DE69513657D1 (de) | 2000-01-05 |
EP0765872B1 (en) | 1999-12-01 |
DE69513657T2 (de) | 2000-04-06 |
CA2157753A1 (en) | 1996-03-09 |
GR3032745T3 (en) | 2000-06-30 |
KR960010630A (ko) | 1996-04-20 |
US5869683A (en) | 1999-02-09 |
CA2157753C (en) | 2006-12-12 |
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Legal Events
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---|---|---|---|
FG2A | Definitive protection |
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