ES2093694T3 - Nuevos derivados de dihidro-isoquinoleina. - Google Patents

Nuevos derivados de dihidro-isoquinoleina.

Info

Publication number
ES2093694T3
ES2093694T3 ES91810954T ES91810954T ES2093694T3 ES 2093694 T3 ES2093694 T3 ES 2093694T3 ES 91810954 T ES91810954 T ES 91810954T ES 91810954 T ES91810954 T ES 91810954T ES 2093694 T3 ES2093694 T3 ES 2093694T3
Authority
ES
Spain
Prior art keywords
isoquinolein
dihydro
new derivatives
alcoxi
esters
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES91810954T
Other languages
English (en)
Inventor
Reto Naef
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sandoz AG
Original Assignee
Sandoz AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz AG filed Critical Sandoz AG
Application granted granted Critical
Publication of ES2093694T3 publication Critical patent/ES2093694T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/02Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/12Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring
    • C07D217/14Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals
    • C07D217/16Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals substituted by oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators

Abstract

6,7-DI(C SUB 1-4ALCOXI)-1-[3,5-DI(C SUB 1-4 ALCOXI)FENIL]-3,4-DIHIDRO-3 -HIDROXI-METIL-ISOQUINOLINAS, SIENDO NOVEDOSOS SUS ESTERES HIDROLIZABLES Y ACEPTABLES FISIOLOGICAMENTE Y SALES ACIDAS DE ADICION DE LO MISMO. LOS MENCIONADOS COMPUESTOS, ESTERES Y SALES ACIDAS DE ADICION FARMACEUTICAMENTE ACEPTABLES DE LO MISMO SON UTILES COMO FARMACOS, E. J. EN EL TRATAMIENTO DEL ASMA.
ES91810954T 1990-12-13 1991-12-09 Nuevos derivados de dihidro-isoquinoleina. Expired - Lifetime ES2093694T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB909027055A GB9027055D0 (en) 1990-12-13 1990-12-13 Organic compounds

Publications (1)

Publication Number Publication Date
ES2093694T3 true ES2093694T3 (es) 1997-01-01

Family

ID=10686945

Family Applications (1)

Application Number Title Priority Date Filing Date
ES91810954T Expired - Lifetime ES2093694T3 (es) 1990-12-13 1991-12-09 Nuevos derivados de dihidro-isoquinoleina.

Country Status (25)

Country Link
US (1) US5177085A (es)
EP (1) EP0490823B1 (es)
JP (1) JPH0764820B2 (es)
KR (1) KR920012040A (es)
AT (1) ATE145201T1 (es)
AU (1) AU643575B2 (es)
CA (1) CA2057524A1 (es)
CZ (1) CZ281669B6 (es)
DE (1) DE69123124T2 (es)
DK (1) DK0490823T3 (es)
ES (1) ES2093694T3 (es)
FI (1) FI915844A (es)
GB (1) GB9027055D0 (es)
GR (1) GR3022034T3 (es)
HU (1) HUT61729A (es)
IE (1) IE914325A1 (es)
IL (1) IL100328A (es)
MX (1) MX9102502A (es)
MY (1) MY129941A (es)
NZ (1) NZ240936A (es)
PL (1) PL168329B1 (es)
PT (1) PT99775B (es)
RU (1) RU2060992C1 (es)
TW (1) TW201736B (es)
ZA (1) ZA919858B (es)

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IT1296985B1 (it) 1997-12-19 1999-08-03 Zambon Spa Derivati benzazinici inibitori della fosfodiesterasi 4
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Also Published As

Publication number Publication date
PL292738A1 (en) 1992-12-14
US5177085A (en) 1993-01-05
MX9102502A (es) 1992-06-01
ZA919858B (en) 1993-06-14
HUT61729A (en) 1993-03-01
GB9027055D0 (en) 1991-02-06
JPH0764820B2 (ja) 1995-07-12
AU8898591A (en) 1992-06-18
DK0490823T3 (es) 1997-02-17
AU643575B2 (en) 1993-11-18
ATE145201T1 (de) 1996-11-15
HU913760D0 (en) 1992-02-28
TW201736B (es) 1993-03-11
JPH04275276A (ja) 1992-09-30
IL100328A (en) 1995-12-08
GR3022034T3 (en) 1997-03-31
CA2057524A1 (en) 1992-06-14
EP0490823B1 (en) 1996-11-13
PT99775B (pt) 1999-05-31
CZ281669B6 (cs) 1996-12-11
DE69123124T2 (de) 1997-05-15
MY129941A (en) 2007-05-31
KR920012040A (ko) 1992-07-25
FI915844A (fi) 1992-06-14
NZ240936A (en) 1993-09-27
RU2060992C1 (ru) 1996-05-27
CS375791A3 (en) 1992-06-17
EP0490823A1 (en) 1992-06-17
PL168329B1 (pl) 1996-02-29
FI915844A0 (fi) 1991-12-11
IL100328A0 (en) 1992-09-06
PT99775A (pt) 1992-11-30
IE914325A1 (en) 1992-06-17
DE69123124D1 (de) 1996-12-19

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