ES2032317T3 - Derivados de quinazolina tetraciclicos, obtencion y empleo. - Google Patents

Derivados de quinazolina tetraciclicos, obtencion y empleo.

Info

Publication number
ES2032317T3
ES2032317T3 ES198888114755T ES88114755T ES2032317T3 ES 2032317 T3 ES2032317 T3 ES 2032317T3 ES 198888114755 T ES198888114755 T ES 198888114755T ES 88114755 T ES88114755 T ES 88114755T ES 2032317 T3 ES2032317 T3 ES 2032317T3
Authority
ES
Spain
Prior art keywords
terracyclic
employment
obtaining
quinazoline derivatives
quinazoline
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES198888114755T
Other languages
English (en)
Inventor
Albrecht Dr. Franke
Bernd Dr. Ostersehlt
Rainer Dr. Schlecker
Beatrice Dr. Rendenbach
Gerda Dr. Von Philipsborn
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BASF SE
Original Assignee
BASF SE
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by BASF SE filed Critical BASF SE
Application granted granted Critical
Publication of ES2032317T3 publication Critical patent/ES2032317T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

SE DESCRIBEN DERIVADOS TETRACICLICOS DE LA QUINAZOLINA DE LA FORMULA(I) DONDE A, X Y R TIENEN LOS SIGNIFICADOS DADOS EN LA DESCRIPCION, ASI COMO SU PRODUCCION. LAS NUEVAS SUSTANCIAS SON APTAS PARA COMBATIR ENFERMEDADES.
ES198888114755T 1987-09-12 1988-09-09 Derivados de quinazolina tetraciclicos, obtencion y empleo. Expired - Lifetime ES2032317T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19873730718 DE3730718A1 (de) 1987-09-12 1987-09-12 Tetracyclische chinazolinderivate, herstellung und verwendung

Publications (1)

Publication Number Publication Date
ES2032317T3 true ES2032317T3 (es) 1993-02-01

Family

ID=6335899

Family Applications (1)

Application Number Title Priority Date Filing Date
ES198888114755T Expired - Lifetime ES2032317T3 (es) 1987-09-12 1988-09-09 Derivados de quinazolina tetraciclicos, obtencion y empleo.

Country Status (7)

Country Link
US (1) US5214047A (es)
EP (1) EP0307814B1 (es)
JP (1) JPS6471881A (es)
AT (1) ATE74605T1 (es)
CA (1) CA1331608C (es)
DE (2) DE3730718A1 (es)
ES (1) ES2032317T3 (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK443589D0 (da) * 1989-09-08 1989-09-08 Ferrosan As Heterocykliske forbindelser, deres fremstilling og anvendelse
KR100333790B1 (ko) 1993-06-25 2002-11-04 메렐 파마슈티칼스 인크. 항히스타민성4-디페닐메틸/디페닐메톡시피페리딘유도체제조용신규중간체
US6147216A (en) * 1993-06-25 2000-11-14 Merrell Pharmaceuticals Inc. Intermediates useful for the preparation of antihistaminic piperidine derivatives
US6930197B2 (en) 1998-07-02 2005-08-16 Aventis Pharmaceuticals Inc. Antihistaminic piperidine derivatives and intermediates for the preparation thereof
US6683094B2 (en) 1998-07-02 2004-01-27 Aventis Pharmaceuticals Inc. Antihistaminic piperidine derivatives and intermediates for the preparation thereof
US6538000B1 (en) 1999-11-19 2003-03-25 Abbott Laboratories Tricyclic dihydropyrimidine potassium channel openers
WO2001036422A1 (en) * 1999-11-19 2001-05-25 Abbott Laboratories Tricyclic dihydropyrimidine potassium channel openers
US6345853B1 (en) * 2000-08-25 2002-02-12 William A. Price, Jr. Self-supporting, confined space entry mobile unit
US20050107867A1 (en) * 2003-11-17 2005-05-19 Taheri Syde A. Temporary absorbable venous occlusive stent and superficial vein treatment method
US7972354B2 (en) 2005-01-25 2011-07-05 Tyco Healthcare Group Lp Method and apparatus for impeding migration of an implanted occlusive structure
US9017361B2 (en) * 2006-04-20 2015-04-28 Covidien Lp Occlusive implant and methods for hollow anatomical structure

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL126596C (es) * 1964-02-11
US3441566A (en) * 1964-11-09 1969-04-29 Sandoz Ag Substituted quinazolines
NL7116968A (es) * 1970-12-21 1972-06-23
GB1347493A (en) * 1971-02-11 1974-02-27 Aspro Nicholas Ltd Benzazine derivatives
US3743733A (en) * 1971-07-26 1973-07-03 Sandoz Ag Method of treating bronchial asthma
US3847918A (en) * 1973-05-17 1974-11-12 Sandoz Ag S-triazolo(1,5-c)quinazolin-7(6h)-ones
GR78233B (es) * 1980-08-15 1984-09-26 Ciba Geigy Ag

Also Published As

Publication number Publication date
EP0307814A3 (en) 1990-08-08
ATE74605T1 (de) 1992-04-15
EP0307814A2 (de) 1989-03-22
CA1331608C (en) 1994-08-23
EP0307814B1 (de) 1992-04-08
US5214047A (en) 1993-05-25
DE3869886D1 (de) 1992-05-14
JPS6471881A (en) 1989-03-16
DE3730718A1 (de) 1989-03-23

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