DK443589D0 - Heterocykliske forbindelser, deres fremstilling og anvendelse - Google Patents
Heterocykliske forbindelser, deres fremstilling og anvendelseInfo
- Publication number
- DK443589D0 DK443589D0 DK443589A DK443589A DK443589D0 DK 443589 D0 DK443589 D0 DK 443589D0 DK 443589 A DK443589 A DK 443589A DK 443589 A DK443589 A DK 443589A DK 443589 D0 DK443589 D0 DK 443589D0
- Authority
- DK
- Denmark
- Prior art keywords
- alkyl
- hydrogen
- chem
- halogen
- independently
- Prior art date
Links
- 238000002360 preparation method Methods 0.000 title abstract 2
- 150000002391 heterocyclic compounds Chemical class 0.000 title 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 4
- 239000001257 hydrogen Substances 0.000 abstract 4
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 3
- 229910052736 halogen Inorganic materials 0.000 abstract 3
- 150000002431 hydrogen Chemical class 0.000 abstract 3
- 150000002367 halogens Chemical class 0.000 abstract 2
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 2
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 1
- 125000006272 (C3-C7) cycloalkyl group Chemical group 0.000 abstract 1
- KJMFQJFNQYWQAV-UHFFFAOYSA-N 3h-imidazo[4,5-h]quinazoline Chemical class C1=NC=NC2=C(NC=N3)C3=CC=C21 KJMFQJFNQYWQAV-UHFFFAOYSA-N 0.000 abstract 1
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 abstract 1
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 241000124008 Mammalia Species 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000003277 amino group Chemical group 0.000 abstract 1
- 230000003474 anti-emetic effect Effects 0.000 abstract 1
- 229940125681 anticonvulsant agent Drugs 0.000 abstract 1
- 239000001961 anticonvulsive agent Substances 0.000 abstract 1
- 229940125683 antiemetic agent Drugs 0.000 abstract 1
- 239000002111 antiemetic agent Substances 0.000 abstract 1
- 239000000164 antipsychotic agent Substances 0.000 abstract 1
- 229940005529 antipsychotics Drugs 0.000 abstract 1
- 239000002249 anxiolytic agent Substances 0.000 abstract 1
- 230000000949 anxiolytic effect Effects 0.000 abstract 1
- 229940005530 anxiolytics Drugs 0.000 abstract 1
- -1 aralkoxy Chemical group 0.000 abstract 1
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 125000004104 aryloxy group Chemical group 0.000 abstract 1
- 210000004556 brain Anatomy 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 150000001721 carbon Chemical group 0.000 abstract 1
- 230000003920 cognitive function Effects 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 1
- 125000004122 cyclic group Chemical group 0.000 abstract 1
- 125000004984 dialkylaminoalkoxy group Chemical group 0.000 abstract 1
- 239000003326 hypnotic agent Substances 0.000 abstract 1
- 230000000147 hypnotic effect Effects 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
- C07D487/14—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Priority Applications (23)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DK443589A DK443589D0 (da) | 1989-09-08 | 1989-09-08 | Heterocykliske forbindelser, deres fremstilling og anvendelse |
| IE308390A IE76298B1 (en) | 1989-09-08 | 1990-08-24 | Tetracyclic Imidazoquinazoline Derivatives Preparation and Pharmaceutical Compositions |
| IL9549090A IL95490A (en) | 1989-09-08 | 1990-08-27 | History of Diamidazo] A: (1, (2-C-5, 1 [Coinazoline and Imidazo] A-5, 1 [Pyrimido] C-2, 1 [Converted Coinazoline, Preparation and Pharmaceutical Preparations Containing or |
| NZ235116A NZ235116A (en) | 1989-09-08 | 1990-08-31 | Tetracyclic imidazoquinazoline derivatives, preparation and pharmaceutical compositions thereof |
| US07/578,054 US5100895A (en) | 1989-09-08 | 1990-09-05 | Heterocyclic compounds and their preparation and use |
| AT90914139T ATE131168T1 (de) | 1989-09-08 | 1990-09-06 | Tetrazyklische imidazochinazolinderivate, deren herstellung und pharmazeutische zusammensetzungen. |
| ZA907112A ZA907112B (en) | 1989-09-08 | 1990-09-06 | Heterocyclic compounds and their preparation and use |
| ES90914139T ES2080159T3 (es) | 1989-09-08 | 1990-09-06 | Derivados de imidazoquinazolina tetraciclicos, preparacion y composiciones farmaceuticas. |
| JP2513237A JPH05504945A (ja) | 1989-09-08 | 1990-09-06 | 四環状イミダゾキナゾリン誘導体、その製法及び製薬組成物 |
| PCT/DK1990/000231 WO1991003478A1 (en) | 1989-09-08 | 1990-09-06 | Tetracyclic imidazoquinazoline derivatives, preparation and pharmaceutical compositions |
| EP90610057A EP0417027A1 (en) | 1989-09-08 | 1990-09-06 | Tetracyclic imidazoquinazoline derivatives, process for their preparation and pharmaceutical compositions containing them |
| AU64297/90A AU638758B2 (en) | 1989-09-08 | 1990-09-06 | Tetracyclic imidazoquinazoline derivatives, preparation and pharmaceutical compositions |
| HU92774A HUT63423A (en) | 1989-09-08 | 1990-09-06 | Process for producing tetracyclic diimidazo- and imidazopyrimido quinazoline derivatives and pharmaceutical compositions comprising same |
| CA002066695A CA2066695A1 (en) | 1989-09-08 | 1990-09-06 | Tetracyclic imidazoquinazoline derivatives, preparation and pharmaceutical compositions |
| KR1019920700516A KR927003598A (ko) | 1989-09-08 | 1990-09-06 | 테트라사이클릭 이미다조퀴나졸린 유도체, 이의 제조방법 및 약제학적 조성물 |
| DE69024058T DE69024058T2 (de) | 1989-09-08 | 1990-09-06 | Tetrazyklische imidazochinazolinderivate, deren herstellung und pharmazeutische zusammensetzungen. |
| DK90914139.2T DK0491814T3 (da) | 1989-09-08 | 1990-09-06 | Tetracycliske imidazoquinazolinderivater, fremgangsmåde til fremstilling af og farmaceutiske præparater indeholdende samme |
| EP90914139A EP0491814B1 (en) | 1989-09-08 | 1990-09-06 | Tetracyclic imidazoquinazoline derivatives, preparation and pharmaceutical compositions |
| PT95249A PT95249B (pt) | 1989-09-08 | 1990-09-07 | Processo de preparacao de compostos de imidazoquinazolina e de composicoes farmaceuticas |
| HU9200774A HU9200774D0 (en) | 1989-09-08 | 1992-03-06 | Process for the production of tetracyclic imidazo-kinoline derivatives and medical preparations containing them |
| NO920910A NO180635C (no) | 1989-09-08 | 1992-03-06 | Analogifremgangsmåte for fremstilling av en terapeutisk aktiv tetracyklisk imidazolinforbindelse |
| FI921004A FI97137C (fi) | 1989-09-08 | 1992-03-06 | Menetelmä farmaseuttisesti aktiivisten tetrasyklisten di-imidatso/1,5-a:1',2'-c/kinatsoliiniyhdisteiden valmistamiseksi |
| GR960400173T GR3018774T3 (en) | 1989-09-08 | 1996-01-24 | Tetracyclic imidazoquinazoline derivatives, preparation and pharmaceutical compositions. |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DK443589A DK443589D0 (da) | 1989-09-08 | 1989-09-08 | Heterocykliske forbindelser, deres fremstilling og anvendelse |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK443589D0 true DK443589D0 (da) | 1989-09-08 |
Family
ID=8133490
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK443589A DK443589D0 (da) | 1989-09-08 | 1989-09-08 | Heterocykliske forbindelser, deres fremstilling og anvendelse |
| DK90914139.2T DK0491814T3 (da) | 1989-09-08 | 1990-09-06 | Tetracycliske imidazoquinazolinderivater, fremgangsmåde til fremstilling af og farmaceutiske præparater indeholdende samme |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK90914139.2T DK0491814T3 (da) | 1989-09-08 | 1990-09-06 | Tetracycliske imidazoquinazolinderivater, fremgangsmåde til fremstilling af og farmaceutiske præparater indeholdende samme |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US5100895A (da) |
| EP (2) | EP0417027A1 (da) |
| JP (1) | JPH05504945A (da) |
| KR (1) | KR927003598A (da) |
| AT (1) | ATE131168T1 (da) |
| AU (1) | AU638758B2 (da) |
| CA (1) | CA2066695A1 (da) |
| DE (1) | DE69024058T2 (da) |
| DK (2) | DK443589D0 (da) |
| ES (1) | ES2080159T3 (da) |
| FI (1) | FI97137C (da) |
| GR (1) | GR3018774T3 (da) |
| HU (2) | HUT63423A (da) |
| IE (1) | IE76298B1 (da) |
| IL (1) | IL95490A (da) |
| NO (1) | NO180635C (da) |
| NZ (1) | NZ235116A (da) |
| PT (1) | PT95249B (da) |
| WO (1) | WO1991003478A1 (da) |
| ZA (1) | ZA907112B (da) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK204291D0 (da) * | 1991-12-20 | 1991-12-20 | Novo Nordisk As | Heterocykliske forbindelser deres fremstilling og anvendelse |
| DK41191D0 (da) * | 1991-03-07 | 1991-03-07 | Novo Nordisk As | Heterocycliske forbindelser, deres fremstilling og anvendelse |
| NZ243065A (en) * | 1991-06-13 | 1995-07-26 | Lundbeck & Co As H | Piperidine derivatives and pharmaceutical compositions |
| TW201311B (da) * | 1991-06-17 | 1993-03-01 | Hoffmann La Roche | |
| WO1993017025A1 (en) * | 1992-02-19 | 1993-09-02 | The Upjohn Company | 3-substituted imidazo(1,5-a)quinoxalines and quinazolines with cns activity |
| US7915410B2 (en) * | 2005-09-09 | 2011-03-29 | Bristol-Myers Squibb Company | Acyclic IKur inhibitors |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3847918A (en) * | 1973-05-17 | 1974-11-12 | Sandoz Ag | S-triazolo(1,5-c)quinazolin-7(6h)-ones |
| DK476885D0 (da) * | 1985-10-17 | 1985-10-17 | Ferrosan As | Heterocycliske forbindelser og fremgangsmaader til fremstilling heraf |
| DE3686723T2 (de) * | 1985-10-17 | 1993-04-01 | Novonordisk As | Oxadiazolylacetonitrile, ihre herstellung und anwendung. |
| DE3730718A1 (de) * | 1987-09-12 | 1989-03-23 | Basf Ag | Tetracyclische chinazolinderivate, herstellung und verwendung |
-
1989
- 1989-09-08 DK DK443589A patent/DK443589D0/da not_active Application Discontinuation
-
1990
- 1990-08-24 IE IE308390A patent/IE76298B1/en not_active IP Right Cessation
- 1990-08-27 IL IL9549090A patent/IL95490A/en not_active IP Right Cessation
- 1990-08-31 NZ NZ235116A patent/NZ235116A/en unknown
- 1990-09-05 US US07/578,054 patent/US5100895A/en not_active Expired - Fee Related
- 1990-09-06 DE DE69024058T patent/DE69024058T2/de not_active Expired - Fee Related
- 1990-09-06 ZA ZA907112A patent/ZA907112B/xx unknown
- 1990-09-06 WO PCT/DK1990/000231 patent/WO1991003478A1/en not_active Ceased
- 1990-09-06 EP EP90610057A patent/EP0417027A1/en active Pending
- 1990-09-06 EP EP90914139A patent/EP0491814B1/en not_active Expired - Lifetime
- 1990-09-06 ES ES90914139T patent/ES2080159T3/es not_active Expired - Lifetime
- 1990-09-06 DK DK90914139.2T patent/DK0491814T3/da active
- 1990-09-06 JP JP2513237A patent/JPH05504945A/ja active Pending
- 1990-09-06 CA CA002066695A patent/CA2066695A1/en not_active Abandoned
- 1990-09-06 HU HU92774A patent/HUT63423A/hu unknown
- 1990-09-06 AU AU64297/90A patent/AU638758B2/en not_active Ceased
- 1990-09-06 KR KR1019920700516A patent/KR927003598A/ko not_active Ceased
- 1990-09-06 AT AT90914139T patent/ATE131168T1/de not_active IP Right Cessation
- 1990-09-07 PT PT95249A patent/PT95249B/pt not_active IP Right Cessation
-
1992
- 1992-03-06 FI FI921004A patent/FI97137C/fi not_active IP Right Cessation
- 1992-03-06 NO NO920910A patent/NO180635C/no unknown
- 1992-03-06 HU HU9200774A patent/HU9200774D0/hu unknown
-
1996
- 1996-01-24 GR GR960400173T patent/GR3018774T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR927003598A (ko) | 1992-12-18 |
| HU9200774D0 (en) | 1992-05-28 |
| IE903083A1 (en) | 1991-03-13 |
| DE69024058T2 (de) | 1996-08-29 |
| JPH05504945A (ja) | 1993-07-29 |
| ATE131168T1 (de) | 1995-12-15 |
| US5100895A (en) | 1992-03-31 |
| FI921004A0 (fi) | 1992-03-06 |
| NO180635C (no) | 1997-05-21 |
| IL95490A (en) | 1994-04-12 |
| NO920910D0 (no) | 1992-03-06 |
| PT95249A (pt) | 1991-05-22 |
| HUT63423A (en) | 1993-08-30 |
| NO920910L (no) | 1992-03-06 |
| DE69024058D1 (de) | 1996-01-18 |
| FI97137B (fi) | 1996-07-15 |
| NO180635B (no) | 1997-02-10 |
| AU638758B2 (en) | 1993-07-08 |
| CA2066695A1 (en) | 1991-03-09 |
| EP0491814B1 (en) | 1995-12-06 |
| WO1991003478A1 (en) | 1991-03-21 |
| PT95249B (pt) | 1997-06-30 |
| EP0491814A1 (en) | 1992-07-01 |
| ZA907112B (en) | 1991-07-31 |
| NZ235116A (en) | 1992-08-26 |
| IL95490A0 (en) | 1991-06-30 |
| ES2080159T3 (es) | 1996-02-01 |
| GR3018774T3 (en) | 1996-04-30 |
| FI97137C (fi) | 1996-10-25 |
| IE76298B1 (en) | 1997-10-08 |
| DK0491814T3 (da) | 1996-04-09 |
| EP0417027A1 (en) | 1991-03-13 |
| AU6429790A (en) | 1991-04-08 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHS | Application shelved for other reasons than non-payment |