ES2060980T3 - Nuevos inhibidores de alfa-glucosidasa. - Google Patents
Nuevos inhibidores de alfa-glucosidasa.Info
- Publication number
- ES2060980T3 ES2060980T3 ES90402613T ES90402613T ES2060980T3 ES 2060980 T3 ES2060980 T3 ES 2060980T3 ES 90402613 T ES90402613 T ES 90402613T ES 90402613 T ES90402613 T ES 90402613T ES 2060980 T3 ES2060980 T3 ES 2060980T3
- Authority
- ES
- Spain
- Prior art keywords
- glycosyl
- radical
- glucosidase inhibitors
- new alpha
- new
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 229940077274 Alpha glucosidase inhibitor Drugs 0.000 title 1
- 239000003888 alpha glucosidase inhibitor Substances 0.000 title 1
- 208000030507 AIDS Diseases 0.000 abstract 2
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 1
- -1 HYDROXYL PART Chemical group 0.000 abstract 1
- 208000008589 Obesity Diseases 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 238000001311 chemical methods and process Methods 0.000 abstract 1
- 206010012601 diabetes mellitus Diseases 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 235000020824 obesity Nutrition 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/044—Pyrrole radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/26—Acyclic or carbocyclic radicals, substituted by hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Molecular Biology (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Biochemistry (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Emergency Medicine (AREA)
- Virology (AREA)
- Endocrinology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- AIDS & HIV (AREA)
- Child & Adolescent Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP89402794A EP0422307A1 (en) | 1989-10-10 | 1989-10-10 | Novel alpha-glucosidase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2060980T3 true ES2060980T3 (es) | 1994-12-01 |
Family
ID=8202997
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES90402613T Expired - Lifetime ES2060980T3 (es) | 1989-10-10 | 1990-09-21 | Nuevos inhibidores de alfa-glucosidasa. |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US5097023A (enExample) |
| EP (2) | EP0422307A1 (enExample) |
| JP (1) | JP3032266B2 (enExample) |
| KR (1) | KR0183012B1 (enExample) |
| CN (1) | CN1029974C (enExample) |
| AR (1) | AR246745A1 (enExample) |
| AT (1) | ATE109153T1 (enExample) |
| AU (1) | AU632855B2 (enExample) |
| CA (1) | CA2027276C (enExample) |
| DE (1) | DE69011033T2 (enExample) |
| DK (1) | DK0422975T3 (enExample) |
| ES (1) | ES2060980T3 (enExample) |
| FI (1) | FI101796B1 (enExample) |
| HU (1) | HU209724B (enExample) |
| IE (1) | IE64079B1 (enExample) |
| IL (1) | IL95928A (enExample) |
| NO (1) | NO174203C (enExample) |
| NZ (1) | NZ235578A (enExample) |
| PT (1) | PT95547B (enExample) |
| TW (1) | TW225539B (enExample) |
| ZA (1) | ZA907936B (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5504078A (en) * | 1990-06-08 | 1996-04-02 | Merrell Dow Pharmaceuticals Inc. | α-glucosidase inhibitors |
| US5268364A (en) * | 1991-12-12 | 1993-12-07 | The Biomembrane Institute | Method for inhibiting selectin-dependent adhesion of leukocytes and platelets by O-glycosylation modification |
| US5605893A (en) * | 1994-03-15 | 1997-02-25 | Children's Hospital Of Los Angeles | Method of using a therapeutic food composition to diminish blood sugar fluctuations in diabetic patients |
| US5843921A (en) * | 1994-03-15 | 1998-12-01 | Childrens Hospital Of Los Angeles | Therapeutic food composition and method to diminish blood sugar fluctuations |
| JP3580900B2 (ja) * | 1995-04-20 | 2004-10-27 | ホクレン農業協同組合連合会 | α−グルコシダーゼ阻害剤を含む糖を主体とする組成物を有効成分とする食品及び飼料 |
| US5929037A (en) * | 1995-06-07 | 1999-07-27 | Alberta Research Council | Modified α-D-Glcρ-(1-2)-α-D-Glcρ-(1-3)-α-D-Glcρ-analogues |
| CZ120398A3 (cs) * | 1995-09-08 | 1998-12-16 | Novo Nordisk A/S | Použití 2-alkylpyrrolidinových derivátů pro přípravu léčiva pro léčbu diabetu, 2-alkylpyrrolidiné deriváty |
| AU4335997A (en) * | 1996-09-09 | 1998-03-26 | Wisconsin Alumni Research Foundation | Human salivary proteins and fragments thereof having alpha-glucosidase inhibitory activity |
| US6534487B1 (en) | 1999-08-03 | 2003-03-18 | Childrens Hospital Los Angeles | Methods for suppressing appetite and enhancing exercise and recovery |
| KR20020070996A (ko) * | 1999-12-21 | 2002-09-11 | 아지노모토 가부시키가이샤 | 질소 함유 카복실산 셀룰로스 부분 에스테르 및 이의제조방법 |
| JP4486792B2 (ja) * | 2003-06-12 | 2010-06-23 | 学校法人近畿大学 | 環状オニウム化合物およびグルコシダーゼ阻害剤 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NO154918C (no) * | 1977-08-27 | 1987-01-14 | Bayer Ag | Analogifremgangsmaate til fremstilling av terapeutisk aktive derivater av 3,4,5-trihydroksypiperidin. |
-
1989
- 1989-10-10 EP EP89402794A patent/EP0422307A1/en not_active Withdrawn
-
1990
- 1990-09-17 US US07/583,545 patent/US5097023A/en not_active Expired - Fee Related
- 1990-09-21 DK DK90402613.5T patent/DK0422975T3/da active
- 1990-09-21 EP EP90402613A patent/EP0422975B1/en not_active Expired - Lifetime
- 1990-09-21 DE DE69011033T patent/DE69011033T2/de not_active Expired - Fee Related
- 1990-09-21 AT AT90402613T patent/ATE109153T1/de not_active IP Right Cessation
- 1990-09-21 ES ES90402613T patent/ES2060980T3/es not_active Expired - Lifetime
- 1990-10-04 AU AU63756/90A patent/AU632855B2/en not_active Ceased
- 1990-10-04 ZA ZA907936A patent/ZA907936B/xx unknown
- 1990-10-05 TW TW079108368A patent/TW225539B/zh active
- 1990-10-05 NZ NZ235578A patent/NZ235578A/en unknown
- 1990-10-09 FI FI904965A patent/FI101796B1/fi not_active IP Right Cessation
- 1990-10-09 JP JP2269667A patent/JP3032266B2/ja not_active Expired - Fee Related
- 1990-10-09 IL IL9592890A patent/IL95928A/en not_active IP Right Cessation
- 1990-10-09 PT PT95547A patent/PT95547B/pt not_active IP Right Cessation
- 1990-10-09 AR AR90318034A patent/AR246745A1/es active
- 1990-10-09 IE IE361390A patent/IE64079B1/en not_active IP Right Cessation
- 1990-10-09 NO NO904372A patent/NO174203C/no not_active IP Right Cessation
- 1990-10-09 HU HU906389A patent/HU209724B/hu not_active IP Right Cessation
- 1990-10-10 KR KR1019900016003A patent/KR0183012B1/ko not_active Expired - Fee Related
- 1990-10-10 CN CN90108284A patent/CN1029974C/zh not_active Expired - Fee Related
- 1990-10-10 CA CA002027276A patent/CA2027276C/en not_active Expired - Fee Related
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG2A | Definitive protection |
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