FI913699A0 - Menetelmä farmaseuttisesti käyttökelpoisten 4'-epi-4'-aminoantrasykliinien valmistamiseksi sekä menetelmässä käytettävät välituotteet - Google Patents

Menetelmä farmaseuttisesti käyttökelpoisten 4'-epi-4'-aminoantrasykliinien valmistamiseksi sekä menetelmässä käytettävät välituotteet

Info

Publication number
FI913699A0
FI913699A0 FI913699A FI913699A FI913699A0 FI 913699 A0 FI913699 A0 FI 913699A0 FI 913699 A FI913699 A FI 913699A FI 913699 A FI913699 A FI 913699A FI 913699 A0 FI913699 A0 FI 913699A0
Authority
FI
Finland
Prior art keywords
aminoanthracyclines
epi
intermediates
preparation
pharmaceutically useful
Prior art date
Application number
FI913699A
Other languages
English (en)
Swedish (sv)
Other versions
FI96605C (fi
FI96605B (fi
Inventor
Francesco Angelucci
Alberto Bargiotti
Daniela Faiardi
Stefania Stefanelli
Antonino Suarato
Original Assignee
Erba Carlo Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Carlo Spa filed Critical Erba Carlo Spa
Publication of FI913699A0 publication Critical patent/FI913699A0/fi
Application granted granted Critical
Publication of FI96605B publication Critical patent/FI96605B/fi
Publication of FI96605C publication Critical patent/FI96605C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/24Condensed ring systems having three or more rings
    • C07H15/252Naphthacene radicals, e.g. daunomycins, adriamycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Pyridine Compounds (AREA)
FI913699A 1989-02-07 1991-08-02 Menetelmä farmaseuttisesti käyttökelpoisten 4'-epi-4'-aminoantrasykliinien valmistamiseksi sekä menetelmässä käytettävät välituotteet FI96605C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB8902709 1989-02-07
GB898902709A GB8902709D0 (en) 1989-02-07 1989-02-07 New 4'-epi-4'-amino anthracyclines
PCT/EP1990/000183 WO1990009392A1 (en) 1989-02-07 1990-02-02 New 4'-epi-4'-amino anthracyclines
EP9000183 1990-02-02

Publications (3)

Publication Number Publication Date
FI913699A0 true FI913699A0 (fi) 1991-08-02
FI96605B FI96605B (fi) 1996-04-15
FI96605C FI96605C (fi) 1996-07-25

Family

ID=10651266

Family Applications (1)

Application Number Title Priority Date Filing Date
FI913699A FI96605C (fi) 1989-02-07 1991-08-02 Menetelmä farmaseuttisesti käyttökelpoisten 4'-epi-4'-aminoantrasykliinien valmistamiseksi sekä menetelmässä käytettävät välituotteet

Country Status (21)

Country Link
EP (1) EP0381989B1 (fi)
JP (1) JP3000562B2 (fi)
KR (1) KR920701227A (fi)
AT (1) ATE72445T1 (fi)
AU (1) AU628478B2 (fi)
CA (1) CA2046645A1 (fi)
DE (1) DE69000019D1 (fi)
DK (1) DK0381989T3 (fi)
ES (1) ES2041050T3 (fi)
FI (1) FI96605C (fi)
GB (1) GB8902709D0 (fi)
GR (1) GR3003873T3 (fi)
HU (1) HU206700B (fi)
IE (1) IE62307B1 (fi)
IL (1) IL93258A (fi)
MY (1) MY105541A (fi)
NZ (1) NZ232305A (fi)
PT (1) PT93071B (fi)
RU (1) RU2073681C1 (fi)
WO (1) WO1990009392A1 (fi)
ZA (1) ZA90835B (fi)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1241927B (it) * 1990-05-14 1994-02-01 Menarini Farma Ind 3'-deamino-4'-deossi-4'-amino-8-fluoroantra- cicline processi per la loro preparazione e composizioni farmaceutiche che le contengono
CN1089071C (zh) * 1999-10-11 2002-08-14 葛水生 铁路列车卫星电视系统
JP5105403B2 (ja) 2006-12-06 2012-12-26 日本サーモスタット株式会社 感温インジケータ
PT2917195T (pt) * 2012-11-05 2018-02-09 Pfizer Análogos de spliceostatina
US9828405B2 (en) 2013-04-29 2017-11-28 Nerviano Medical Sciences S.R.L. Morpholinyl anthracycline derivatives
EP3215513B1 (en) 2014-11-05 2019-05-08 Nerviano Medical Sciences S.r.l. Functionalized morpholinyl anthracycline derivatives

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE8401T1 (de) * 1980-11-01 1984-07-15 Farmitalia Carlo Erba S.P.A. Anthracyclin-glycoside, verfahren zu ihrer herstellung, zwischenprodukte und ihre herstellung und arzneimittel.
GB2091243B (en) * 1981-01-21 1984-06-20 Erba Farmitalia Anthracycline glycosides
GB8803076D0 (en) * 1988-02-10 1988-03-09 Erba Carlo Spa 3'-deamino-4'-deoxy-4'-amino anthracyclines

Also Published As

Publication number Publication date
HUT58065A (en) 1992-01-28
GR3003873T3 (fi) 1993-03-16
EP0381989A1 (en) 1990-08-16
JP3000562B2 (ja) 2000-01-17
FI96605C (fi) 1996-07-25
ATE72445T1 (de) 1992-02-15
AU4951090A (en) 1990-09-05
IE62307B1 (en) 1995-01-25
IE900403L (en) 1990-08-07
DE69000019D1 (en) 1992-03-19
MY105541A (en) 1994-10-31
GB8902709D0 (en) 1989-03-30
HU901678D0 (en) 1991-11-28
RU2073681C1 (ru) 1997-02-20
NZ232305A (en) 1991-11-26
WO1990009392A1 (en) 1990-08-23
IL93258A0 (en) 1990-11-29
PT93071B (pt) 1996-01-31
ZA90835B (en) 1990-11-28
FI96605B (fi) 1996-04-15
PT93071A (pt) 1990-08-31
IL93258A (en) 1994-05-30
KR920701227A (ko) 1992-08-11
ES2041050T3 (es) 1993-11-01
CA2046645A1 (en) 1990-08-08
DK0381989T3 (da) 1992-03-23
EP0381989B1 (en) 1992-02-05
AU628478B2 (en) 1992-09-17
JPH04503210A (ja) 1992-06-11
HU206700B (en) 1992-12-28

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