EP2445907A1 - Dérivés de thiazolylpipéridine comme fongicides - Google Patents

Dérivés de thiazolylpipéridine comme fongicides

Info

Publication number
EP2445907A1
EP2445907A1 EP10725040A EP10725040A EP2445907A1 EP 2445907 A1 EP2445907 A1 EP 2445907A1 EP 10725040 A EP10725040 A EP 10725040A EP 10725040 A EP10725040 A EP 10725040A EP 2445907 A1 EP2445907 A1 EP 2445907A1
Authority
EP
European Patent Office
Prior art keywords
substituents
alkyl
methyl
phenyl
haloalkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
EP10725040A
Other languages
German (de)
English (en)
Inventor
Pierre Cristau
Nicola Rahn
Tomoki Tsuchiya
Ulrike Wachendorff-Neumann
Jürgen BENTING
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer Intellectual Property GmbH
Original Assignee
Bayer CropScience AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41203840&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EP2445907(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer CropScience AG filed Critical Bayer CropScience AG
Priority to EP10725040A priority Critical patent/EP2445907A1/fr
Publication of EP2445907A1 publication Critical patent/EP2445907A1/fr
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/78—1,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

L'invention concerne des dérivés de thiazolylpipéridine de la formule (I), dans laquelle les symboles A, G, Y, n, R1, R2, R3, R4, et R5 ont la signification indiquée dans la description ainsi que des sels de ceux-ci agrochimiquement efficaces et leur utilisation dans la lutte contre des champignons parasites pathogènes ainsi qu'un procédé de fabrication de composés de la formule (I).
EP10725040A 2009-06-23 2010-06-10 Dérivés de thiazolylpipéridine comme fongicides Withdrawn EP2445907A1 (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
EP10725040A EP2445907A1 (fr) 2009-06-23 2010-06-10 Dérivés de thiazolylpipéridine comme fongicides

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP09163473A EP2272846A1 (fr) 2009-06-23 2009-06-23 Dérivés de thiazolylpipéridine en tant que fongicide
EP10725040A EP2445907A1 (fr) 2009-06-23 2010-06-10 Dérivés de thiazolylpipéridine comme fongicides
PCT/EP2010/003499 WO2010149275A1 (fr) 2009-06-23 2010-06-10 Dérivés de thiazolylpipéridine comme fongicides

Publications (1)

Publication Number Publication Date
EP2445907A1 true EP2445907A1 (fr) 2012-05-02

Family

ID=41203840

Family Applications (2)

Application Number Title Priority Date Filing Date
EP09163473A Withdrawn EP2272846A1 (fr) 2009-06-23 2009-06-23 Dérivés de thiazolylpipéridine en tant que fongicide
EP10725040A Withdrawn EP2445907A1 (fr) 2009-06-23 2010-06-10 Dérivés de thiazolylpipéridine comme fongicides

Family Applications Before (1)

Application Number Title Priority Date Filing Date
EP09163473A Withdrawn EP2272846A1 (fr) 2009-06-23 2009-06-23 Dérivés de thiazolylpipéridine en tant que fongicide

Country Status (17)

Country Link
US (3) US20110046178A1 (fr)
EP (2) EP2272846A1 (fr)
JP (1) JP2012530734A (fr)
KR (1) KR20120050434A (fr)
CN (2) CN102459254A (fr)
AR (1) AR077066A1 (fr)
BR (1) BRPI1014077A8 (fr)
CA (1) CA2766199A1 (fr)
CL (1) CL2011003180A1 (fr)
CO (1) CO6480909A2 (fr)
EA (1) EA201270059A1 (fr)
IL (1) IL216344A0 (fr)
MX (1) MX2011013706A (fr)
PE (1) PE20121047A1 (fr)
TW (1) TW201111377A (fr)
WO (1) WO2010149275A1 (fr)
ZA (1) ZA201109365B (fr)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL2516426T3 (pl) 2009-12-21 2016-03-31 Bayer Cropscience Ag Bis(difluorometylo)pirazole jako fungicydy
BR112012027762B1 (pt) 2010-04-28 2018-06-05 Bayer Intellectual Property Gmbh Derivados de cetoheteroarilpiperidina e - piperazina como fungicidas
JP2013528169A (ja) 2010-05-27 2013-07-08 バイエル・クロップサイエンス・アーゲー 殺菌剤としてのピリジニルカルボン酸誘導体
CA2815716C (fr) 2010-10-27 2019-06-11 Bayer Intellectual Property Gmbh Heteroarylpiperidine et derives d'heteroarylpiperidine comme fongicide
JP6326231B2 (ja) 2011-02-01 2018-05-16 バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングＢａｙｅｒ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ ＧｍｂＨ 殺菌剤としてのヘテロアリールピペリジン誘導体及びヘテロアリールピペラジン誘導体
US10004232B2 (en) 2011-09-15 2018-06-26 Bayer Intellectual Property Gmbh Piperidine pyrazoles as fungicides
CN104093715B (zh) 2012-02-02 2017-04-26 埃科特莱茵药品有限公司 4‑(苯并咪唑‑2‑基)‑噻唑化合物及相关氮杂衍生物
JP5931291B2 (ja) 2012-08-30 2016-06-08 バイエル・クロップサイエンス・アクチェンゲゼルシャフト ３，５−ビス（ハロアルキル）−ピラゾール−４−カルボン酸誘導体の脱カルボキシル化手順
WO2015011099A1 (fr) 2013-07-22 2015-01-29 Actelion Pharmaceuticals Ltd Dérivés de 1-(pipérazin-1-yl)-2-([1,2,4]triazol-1-yl)-éthanone
AR099789A1 (es) 2014-03-24 2016-08-17 Actelion Pharmaceuticals Ltd Derivados de 8-(piperazin-1-il)-1,2,3,4-tetrahidro-isoquinolina
WO2016024350A1 (fr) 2014-08-13 2016-02-18 株式会社エス・ディー・エス バイオテック Composés cycliques à 11 éléments condensés et fongicides pour l'agriculture et l'horticulture les contenant
TR201900680T4 (tr) 2015-01-15 2019-02-21 Idorsia Pharmaceuticals Ltd CXCR3 Reseptör modülatörleri olarak hidroksialkil- piperazin türevleri.
AR103399A1 (es) 2015-01-15 2017-05-10 Actelion Pharmaceuticals Ltd Derivados de (r)-2-metil-piperazina como moduladores del receptor cxcr3
JP6407457B2 (ja) 2016-02-08 2018-10-17 株式会社エス・ディー・エス バイオテック １，２−ベンゼンジメタノール化合物の製造方法
US11903387B2 (en) 2016-02-08 2024-02-20 Gowan Company, L.L.C. Fungicidal composition
CN106083707B (zh) * 2016-06-01 2018-10-26 温州大学 一种非对称杂芳基硫醚的合成方法
CN107646855B (zh) * 2017-08-02 2020-07-07 浙江工业大学 一种含哌啶噻唑类化合物在制备杀菌剂中的应用及其制备方法
CN114502551B (zh) 2019-11-01 2023-08-22 优迈特株式会社 含氟嘧啶化合物及其制备方法

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US4272417A (en) 1979-05-22 1981-06-09 Cargill, Incorporated Stable protective seed coating
US4245432A (en) 1979-07-25 1981-01-20 Eastman Kodak Company Seed coatings
WO1987005296A1 (fr) 1986-03-07 1987-09-11 Pfizer Inc. 2-[(2-pyridyl)methylsulfinyl]thienoimidazoles et composes apparentes utilises en tant qu'agents de traitement ou de prevention des ulceres
US4808430A (en) 1987-02-27 1989-02-28 Yazaki Corporation Method of applying gel coating to plant seeds
GB8810120D0 (en) 1988-04-28 1988-06-02 Plant Genetic Systems Nv Transgenic nuclear male sterile plants
ATE342968T1 (de) 1995-04-20 2006-11-15 Basf Ag Auf basis ihrer struktur entworfene herbizid resistente produkte
US5876739A (en) 1996-06-13 1999-03-02 Novartis Ag Insecticidal seed coating
US6503904B2 (en) 1998-11-16 2003-01-07 Syngenta Crop Protection, Inc. Pesticidal composition for seed treatment
US6660690B2 (en) 2000-10-06 2003-12-09 Monsanto Technology, L.L.C. Seed treatment with combinations of insecticides
US20020134012A1 (en) 2001-03-21 2002-09-26 Monsanto Technology, L.L.C. Method of controlling the release of agricultural active ingredients from treated plant seeds
EP2277867B1 (fr) * 2002-07-15 2012-12-05 Symphony Evolution, Inc. Composés, compositions pharmaceutiques les contenants et leur utilisation pour traiter le cancer
FR2856685B1 (fr) * 2003-06-25 2005-09-23 Merck Sante Sas Derives de thiazolylpiperidine, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent
PE20060426A1 (es) 2004-06-02 2006-06-28 Schering Corp DERIVADOS DE ACIDO TARTARICO COMO INHIBIDORES DE MMPs, ADAMs, TACE Y TNF-alfa
DE102005031583A1 (de) * 2005-07-06 2007-01-25 Bayer Cropscience Gmbh Verfahren zur Herstellung von von 3-Arylmethylthio- und 3-Heteroarylmethylthio-4,5-dihydro-isoxazolin-Derivaten
TW200738701A (en) 2005-07-26 2007-10-16 Du Pont Fungicidal carboxamides
BRPI0614834A2 (pt) * 2005-08-18 2011-04-19 Hoffmann La Roche compostos, processo para a sua manufatura, composições farmacêuticas que os compreendem e usos destas
ATE544861T1 (de) 2005-08-24 2012-02-15 Pioneer Hi Bred Int Verfahren und zusammensetzungen für den ausdruck eines polynukleotid von interesse
ES2400809T3 (es) 2005-08-31 2013-04-12 Monsanto Technology Llc Secuencias de nucleótidos que codifican proteínas insecticidas
KR101130380B1 (ko) 2006-06-13 2012-04-23 상하이 인스티튜트 오브 마테리아 메디카 차이니즈 아카데미 오브 싸이언시즈 헤테로시클릭 비뉴클레오시드 화합물, 그의 제조방법, 약학적 조성물 및 항바이러스성 약제로서의 용도
DE102006031143A1 (de) * 2006-07-04 2008-01-24 Merck Patent Gmbh Fluortenside
WO2008013622A2 (fr) 2006-07-27 2008-01-31 E. I. Du Pont De Nemours And Company Amides azocycliques fongicides
US7638541B2 (en) * 2006-12-28 2009-12-29 Metabolex Inc. 5-ethyl-2-{4-[4-(4-tetrazol-1-yl-phenoxymethyl)-thiazol-2-yl]-piperidin-1-yl}-pyrimidine
WO2008091594A2 (fr) 2007-01-24 2008-07-31 E. I. Du Pont De Nemours And Company Mélanges fongicides
JP5337711B2 (ja) 2007-01-25 2013-11-06 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー 殺菌性アミド
TWI428091B (zh) 2007-10-23 2014-03-01 Du Pont 殺真菌劑混合物

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Also Published As

Publication number Publication date
US20130090476A1 (en) 2013-04-11
KR20120050434A (ko) 2012-05-18
US20110046178A1 (en) 2011-02-24
US20130090477A1 (en) 2013-04-11
BRPI1014077A2 (pt) 2015-08-25
TW201111377A (en) 2011-04-01
PE20121047A1 (es) 2012-08-02
CN104059059A (zh) 2014-09-24
IL216344A0 (en) 2012-01-31
MX2011013706A (es) 2012-02-22
CO6480909A2 (es) 2012-07-16
EP2272846A1 (fr) 2011-01-12
CL2011003180A1 (es) 2012-06-15
CN102459254A (zh) 2012-05-16
WO2010149275A1 (fr) 2010-12-29
ZA201109365B (en) 2013-02-27
CA2766199A1 (fr) 2010-12-29
AR077066A1 (es) 2011-07-27
EA201270059A1 (ru) 2012-08-30
BRPI1014077A8 (pt) 2016-05-24
JP2012530734A (ja) 2012-12-06

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Legal Events

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Effective date: 20140217

RAP1 Party data changed (applicant data changed or rights of an application transferred)

Owner name: BAYER INTELLECTUAL PROPERTY GMBH

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