EE9400348A - Aminoalküülguanidiinide valmistamise protsess ja selliselt saadud ühendid - Google Patents

Aminoalküülguanidiinide valmistamise protsess ja selliselt saadud ühendid

Info

Publication number
EE9400348A
EE9400348A EE9400348A EE9400348A EE9400348A EE 9400348 A EE9400348 A EE 9400348A EE 9400348 A EE9400348 A EE 9400348A EE 9400348 A EE9400348 A EE 9400348A EE 9400348 A EE9400348 A EE 9400348A
Authority
EE
Estonia
Prior art keywords
pct
compounds
date
sec
jun
Prior art date
Application number
EE9400348A
Other languages
English (en)
Estonian (et)
Inventor
Frederik Sj�bom Hans
Erik Nystr�m Jan-
Original Assignee
Astra Aktiebolag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astra Aktiebolag filed Critical Astra Aktiebolag
Publication of EE9400348A publication Critical patent/EE9400348A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C277/00Preparation of guanidine or its derivatives, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C277/08Preparation of guanidine or its derivatives, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups of substituted guanidines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/20Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups containing any of the groups, X being a hetero atom, Y being any atom, e.g. acylguanidines
    • C07C279/24Y being a hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Treatments For Attaching Organic Compounds To Fibrous Goods (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
EE9400348A 1993-06-03 1994-11-17 Aminoalküülguanidiinide valmistamise protsess ja selliselt saadud ühendid EE9400348A (et)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE19939301912A SE9301912D0 (sv) 1993-06-03 1993-06-03 Process for the production of aminoalkylguandines

Publications (1)

Publication Number Publication Date
EE9400348A true EE9400348A (et) 1996-04-15

Family

ID=20390162

Family Applications (1)

Application Number Title Priority Date Filing Date
EE9400348A EE9400348A (et) 1993-06-03 1994-11-17 Aminoalküülguanidiinide valmistamise protsess ja selliselt saadud ühendid

Country Status (27)

Country Link
US (1) US5659071A (sh)
EP (1) EP0701550B1 (sh)
JP (1) JP3662925B2 (sh)
CN (1) CN1124956A (sh)
AT (1) ATE178316T1 (sh)
AU (1) AU674970B2 (sh)
BR (1) BR9406713A (sh)
CA (1) CA2162920C (sh)
CZ (1) CZ320095A3 (sh)
DE (1) DE69417554T2 (sh)
DK (1) DK0701550T3 (sh)
EE (1) EE9400348A (sh)
ES (1) ES2131688T3 (sh)
FI (1) FI120093B (sh)
GR (1) GR3030501T3 (sh)
HR (1) HRP940317A2 (sh)
HU (1) HUT74293A (sh)
IL (1) IL109683A0 (sh)
IS (1) IS4165A (sh)
LT (1) LT3309B (sh)
NO (1) NO305514B1 (sh)
NZ (1) NZ267192A (sh)
PL (1) PL311760A1 (sh)
SE (1) SE9301912D0 (sh)
SK (1) SK151895A3 (sh)
WO (1) WO1994029269A1 (sh)
YU (1) YU33594A (sh)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5610308A (en) * 1995-05-18 1997-03-11 Bristol-Myers Squibb Company Process for preparing intermediates for thrombin inhibitors
JP2000502078A (ja) * 1995-12-09 2000-02-22 ベーリンガー マンハイム ゲゼルシャフト ミット ベシュレンクテル ハフツング 擬似アルギニン特性を有する3―アミノエチル―n―アミジノ―2,5―ジヒドロピロール誘導体
AR035216A1 (es) * 2000-12-01 2004-05-05 Astrazeneca Ab Derivados de acido mandelico ,derivados farmaceuticamente aceptables, uso de estos derivados para la fabricacion de medicamentos, metodos de tratamiento ,procesos para la preparacion de estos derivados, y compuestos intermediarios
US7129233B2 (en) * 2000-12-01 2006-10-31 Astrazeneca Ab Mandelic acid derivatives and their use as thrombin inhibitors
FR2822463B1 (fr) 2001-03-21 2004-07-30 Lipha Derives bicycliques de guanidines et leurs applications en therapeutique
AR034517A1 (es) 2001-06-21 2004-02-25 Astrazeneca Ab Formulacion farmaceutica
SE0201661D0 (sv) 2002-05-31 2002-05-31 Astrazeneca Ab New salts
SE0201659D0 (sv) 2002-05-31 2002-05-31 Astrazeneca Ab Modified release pharmaceutical formulation
US7781424B2 (en) * 2003-05-27 2010-08-24 Astrazeneca Ab Modified release pharmaceutical formulation
US7524354B2 (en) * 2005-07-07 2009-04-28 Research Foundation Of State University Of New York Controlled synthesis of highly monodispersed gold nanoparticles
CN101489655A (zh) 2006-07-14 2009-07-22 威斯康星旧生研究基金会 捕获病毒用吸附膜
TW200827336A (en) * 2006-12-06 2008-07-01 Astrazeneca Ab New crystalline forms
US20090061000A1 (en) * 2007-08-31 2009-03-05 Astrazeneca Ab Pharmaceutical formulation use 030
JP6006634B2 (ja) * 2011-12-28 2016-10-12 東和薬品株式会社 イソウレア化合物を用いるエピナスチンの製造方法
CN106132926B (zh) * 2014-03-28 2019-05-21 株式会社钟化 三苄氧羰基精氨酸的制造方法
US20220002238A1 (en) * 2018-11-07 2022-01-06 Regents Of The University Of Minnesota Analgesic and anti-addictive compositions for treatment of chronic pain and opioid addiction

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE463576C (de) * 1924-08-06 1928-07-31 Schering Kahlbaum Akt Ges Verfahren zur Darstellung von Aminoguanidinen oder deren Salzen
FR2294699A1 (fr) * 1974-12-19 1976-07-16 Bottu Nouveaux derives du pyrazole et compositions pharmaceutiques les renfermant
HU178398B (en) * 1979-06-12 1982-04-28 Gyogyszerkutato Intezet Process for producing new agmatine derivatives of activity against haemagglutination
US4387049A (en) 1982-02-22 1983-06-07 Smithkline Beckman Corporation Adamantyl containing peptides
DE3222342A1 (de) * 1982-06-14 1983-12-15 Hoechst Ag, 6230 Frankfurt 6-aryl-1,2,4-triazolo (4,3-b) pyridazin-3-carbaminate, ihre herstellung und sie enthaltende arzneimittel
US4914189A (en) * 1987-02-05 1990-04-03 The Adminstrators Of The Tulane Educational Fund Synthetic GHRH analogs
AU2306592A (en) * 1991-07-03 1993-02-11 E.I. Du Pont De Nemours And Company Azeotropic or azeotrope-like compositions of pentafluoroethane and propane or isobutane
US5498724A (en) * 1994-06-28 1996-03-12 Aktiebolaget Astra Pyrazoleamidine compounds

Also Published As

Publication number Publication date
HUT74293A (en) 1996-11-28
LTIP1940A (en) 1994-12-27
SK151895A3 (en) 1996-04-03
AU6940494A (en) 1995-01-03
IS4165A (is) 1994-12-04
NO954835D0 (no) 1995-11-28
NO954835L (no) 1995-11-28
LT3309B (en) 1995-06-26
ATE178316T1 (de) 1999-04-15
FI120093B (fi) 2009-06-30
DK0701550T3 (da) 1999-10-11
FI955800A0 (fi) 1995-12-01
SE9301912D0 (sv) 1993-06-03
FI955800A (fi) 1995-12-01
CA2162920C (en) 2005-08-09
CZ320095A3 (en) 1996-07-17
EP0701550B1 (en) 1999-03-31
CA2162920A1 (en) 1994-12-22
CN1124956A (zh) 1996-06-19
HRP940317A2 (en) 1996-10-31
NO305514B1 (no) 1999-06-14
HU9503444D0 (en) 1996-01-29
DE69417554T2 (de) 1999-09-02
ES2131688T3 (es) 1999-08-01
AU674970B2 (en) 1997-01-16
NZ267192A (en) 1997-03-24
JPH08511016A (ja) 1996-11-19
WO1994029269A1 (en) 1994-12-22
IL109683A0 (en) 1994-08-26
BR9406713A (pt) 1996-03-19
JP3662925B2 (ja) 2005-06-22
YU33594A (sh) 1997-05-28
PL311760A1 (en) 1996-03-18
EP0701550A1 (en) 1996-03-20
GR3030501T3 (en) 1999-10-29
DE69417554D1 (de) 1999-05-06
US5659071A (en) 1997-08-19

Similar Documents

Publication Publication Date Title
EE9400348A (et) Aminoalküülguanidiinide valmistamise protsess ja selliselt saadud ühendid
HK1013283A1 (en) Nitrato amino acid disulphides for use in the therapy of disorders of the cardiovasculary system
BR0307351A (pt) Composto, composição farmacêutica, método para tratar uma condição ou estado de doença mediados pela atividade de p38 quinase ou mediados por citocinas produzidas pela atividade de p38 quinase, uso de um composto, e, processo para preparar um composto
BG103250A (en) Modified amino acids, medicamentous forms containing them, and method for their preparation
IL126610A0 (en) N-(amidinophenyl)-n'-(subst.)-3h-2,4-benzodiazepin-3- one derivatives as factor xa inhibitors
ATE295346T1 (de) N-(aryl/heteroarylacetyl)aminosäureester, diese enthaltende pharmazeutische zusammensetzungen und methoden zur inhibierung der beta- amyloidfreisetzung und/oder deren synthese unter verwendung dieser verbindungen
MX9803954A (es) Derivados de aminoacidos, composiciones farmaceuticas que contienen estos compuestos y procesos para prepararlos.
ES2108882T3 (es) Procedimiento para la alquilacion de derivados de estrona.
HK1028610A1 (en) Method for preparing a substituted perhydroisoindole
PL336996A1 (en) Guanidilating compounds
NO975679L (no) Fremgangsmåte for fremstilling av N-monosubstituerte og N,N'-disubstituerte, usymmetriske, cykliske ureaer
IT1293777B1 (it) Processo per la preparazione di tetraazamacrocicli
BR0009453A (pt) Processo para a preparação de um composto
BR9608237A (pt) Processos para preparar 1-(piridil)-2-cicloexiletilamina racêmica e anantiomérica.
DE50309260D1 (de) Verfahren zur herstellung von bicalutamid
BR9610175A (pt) Composto processo de preparação do composto composição farmacêutica e utilização do composto
CO5540298A2 (es) Proceso para preparar un ligando de ppar de tiazol y polimorfos del mismo
DK1246790T3 (da) Substituerede 1- og 2-naphthol-Mannichbaser
HK1027560A1 (en) Method for producing 1,3-disubstituted 2-nitroguanidines
DK0824515T3 (da) Substitueret phenylamidiner, medikamenter indeholdende disse forbindelser og fremgangsmåder til fremstilling deraf
DE69905397T2 (de) Selektive inhibitoren des mmp-12
IT1216865B (it) Derivato argininico, procedimento per la sua preparazione e suo impiego nelle sintesi peptidiche.
NO974625L (no) Fremgangsmåte for reduktiv alkylering til fremstilling av forbindelser med minst to aminogrupper
BR0112849A (pt) Processo para a preparação de um composto quiral, e, composto quiral
HUP0102540A2 (hu) Új angiotenzin-receptor, eljárás előállítására és alkalmazása