EE200400024A - Kolesterüülestri ülekandevalgu inhibiitorite iseemulgeeruvad formulatsioonid - Google Patents

Kolesterüülestri ülekandevalgu inhibiitorite iseemulgeeruvad formulatsioonid

Info

Publication number
EE200400024A
EE200400024A EEP200400024A EEP200400024A EE200400024A EE 200400024 A EE200400024 A EE 200400024A EE P200400024 A EEP200400024 A EE P200400024A EE P200400024 A EEP200400024 A EE P200400024A EE 200400024 A EE200400024 A EE 200400024A
Authority
EE
Estonia
Prior art keywords
self
transfer protein
cholesteryl ester
protein inhibitors
ester transfer
Prior art date
Application number
EEP200400024A
Other languages
English (en)
Estonian (et)
Inventor
Jon Gumkowski Michael
Balasaheb Murdande Sharad
Ellis Perlman Michael
Lombardo Franco
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of EE200400024A publication Critical patent/EE200400024A/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/44Oils, fats or waxes according to two or more groups of A61K47/02-A61K47/42; Natural or modified natural oils, fats or waxes, e.g. castor oil, polyethoxylated castor oil, montan wax, lignite, shellac, rosin, beeswax or lanolin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4418Non condensed pyridines; Hydrogenated derivatives thereof having a carbocyclic group directly attached to the heterocyclic ring, e.g. cyproheptadine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/255Esters, e.g. nitroglycerine, selenocyanates of sulfoxy acids or sulfur analogues thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41961,2,4-Triazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/47064-Aminoquinolines; 8-Aminoquinolines, e.g. chloroquine, primaquine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biophysics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Emergency Medicine (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Cosmetics (AREA)
  • Emulsifying, Dispersing, Foam-Producing Or Wetting Agents (AREA)
  • Colloid Chemistry (AREA)
  • Quinoline Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pyridine Compounds (AREA)
  • Peptides Or Proteins (AREA)
EEP200400024A 2001-06-21 2002-05-03 Kolesterüülestri ülekandevalgu inhibiitorite iseemulgeeruvad formulatsioonid EE200400024A (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US30002801P 2001-06-21 2001-06-21
PCT/IB2002/001571 WO2003000295A2 (en) 2001-06-21 2002-05-03 Self-emulsifying formulations of cholesteryl ester transfer protein inhibitors

Publications (1)

Publication Number Publication Date
EE200400024A true EE200400024A (et) 2004-06-15

Family

ID=23157363

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200400024A EE200400024A (et) 2001-06-21 2002-05-03 Kolesterüülestri ülekandevalgu inhibiitorite iseemulgeeruvad formulatsioonid

Country Status (33)

Country Link
US (2) US6962931B2 (pt)
EP (1) EP1453544A2 (pt)
JP (1) JP2005500314A (pt)
KR (1) KR20040015746A (pt)
CN (1) CN1635911A (pt)
AP (1) AP2002002559A0 (pt)
AR (1) AR034599A1 (pt)
BG (1) BG108486A (pt)
BR (1) BR0210505A (pt)
CA (1) CA2455288A1 (pt)
CR (1) CR7163A (pt)
CZ (1) CZ20033341A3 (pt)
EA (1) EA200301139A1 (pt)
EC (1) ECSP034875A (pt)
EE (1) EE200400024A (pt)
GT (1) GT200200124A (pt)
HN (1) HN2002000153A (pt)
HU (1) HUP0400263A2 (pt)
IL (1) IL158765A0 (pt)
IS (1) IS7014A (pt)
MA (1) MA27034A1 (pt)
MX (1) MXPA04000014A (pt)
NO (1) NO20035632L (pt)
OA (1) OA12619A (pt)
PA (1) PA8548601A1 (pt)
PE (1) PE20030128A1 (pt)
PL (1) PL368850A1 (pt)
SK (1) SK15172003A3 (pt)
SV (1) SV2003001103A (pt)
TN (1) TNSN03139A1 (pt)
UY (1) UY27344A1 (pt)
WO (1) WO2003000295A2 (pt)
ZA (1) ZA200308561B (pt)

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BR0210505A (pt) 2004-05-18
AR034599A1 (es) 2004-03-03
NO20035632D0 (no) 2003-12-17
IS7014A (is) 2003-10-31
US20060014788A1 (en) 2006-01-19
PA8548601A1 (es) 2003-09-05
ECSP034875A (es) 2004-01-28
CN1635911A (zh) 2005-07-06
ZA200308561B (en) 2004-11-17
TNSN03139A1 (fr) 2005-12-23
PL368850A1 (en) 2005-04-04
NO20035632L (no) 2004-02-18
KR20040015746A (ko) 2004-02-19
SK15172003A3 (en) 2004-11-03
CA2455288A1 (en) 2003-01-03
BG108486A (bg) 2005-03-31
JP2005500314A (ja) 2005-01-06
AP2002002559A0 (en) 2002-06-30
SV2003001103A (es) 2003-03-18
US20030022944A1 (en) 2003-01-30
WO2003000295A2 (en) 2003-01-03
EA200301139A1 (ru) 2004-12-30
GT200200124A (es) 2003-09-22
OA12619A (en) 2006-06-12
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US6962931B2 (en) 2005-11-08
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MA27034A1 (fr) 2004-12-20
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