EA201890738A1 - Комбинированная терапия, включающая канаглифлозин и фентермин, для лечения ожирения и связанных с ожирением расстройств - Google Patents

Комбинированная терапия, включающая канаглифлозин и фентермин, для лечения ожирения и связанных с ожирением расстройств

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Publication number
EA201890738A1
EA201890738A1 EA201890738A EA201890738A EA201890738A1 EA 201890738 A1 EA201890738 A1 EA 201890738A1 EA 201890738 A EA201890738 A EA 201890738A EA 201890738 A EA201890738 A EA 201890738A EA 201890738 A1 EA201890738 A1 EA 201890738A1
Authority
EA
Eurasian Patent Office
Prior art keywords
progression
disorders
obesity
treating
cardiovascular
Prior art date
Application number
EA201890738A
Other languages
English (en)
Russian (ru)
Inventor
Норман Р. Розенталь
Пол Ротенберг
Дэвид К. Полидори
Дуглас К. Вэйс
Питер П. Стейн
Original Assignee
Янссен Фармацевтика Нв
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Янссен Фармацевтика Нв filed Critical Янссен Фармацевтика Нв
Publication of EA201890738A1 publication Critical patent/EA201890738A1/ru

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Emergency Medicine (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Child & Adolescent Psychology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
EA201890738A 2015-09-15 2016-09-13 Комбинированная терапия, включающая канаглифлозин и фентермин, для лечения ожирения и связанных с ожирением расстройств EA201890738A1 (ru)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201562218842P 2015-09-15 2015-09-15
US201662306110P 2016-03-10 2016-03-10
US15/262,038 US20170071970A1 (en) 2015-09-15 2016-09-12 Co-therapy comprising canagliflozin and phentermine for the treatment of obesity and obesity related disorders
PCT/US2016/051435 WO2017048670A1 (en) 2015-09-15 2016-09-13 Co-therapy comprising canagliflozin and phentermine for the treatment of obesity and obesity related disorders

Publications (1)

Publication Number Publication Date
EA201890738A1 true EA201890738A1 (ru) 2018-10-31

Family

ID=58236464

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201890738A EA201890738A1 (ru) 2015-09-15 2016-09-13 Комбинированная терапия, включающая канаглифлозин и фентермин, для лечения ожирения и связанных с ожирением расстройств

Country Status (18)

Country Link
US (3) US20170071970A1 (https=)
EP (1) EP3349740B1 (https=)
JP (1) JP2018527374A (https=)
KR (1) KR20180051560A (https=)
CN (1) CN108024977A (https=)
AU (1) AU2016322537B2 (https=)
CA (1) CA2998730A1 (https=)
CO (1) CO2018002708A2 (https=)
EA (1) EA201890738A1 (https=)
ES (1) ES2873117T3 (https=)
HK (1) HK1248124A1 (https=)
IL (1) IL257876A (https=)
MX (1) MX383002B (https=)
PH (1) PH12018500501A1 (https=)
TW (1) TW201722413A (https=)
UA (1) UA122974C2 (https=)
WO (1) WO2017048670A1 (https=)
ZA (1) ZA201802448B (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI835735B (zh) * 2017-06-12 2024-03-21 比利時商健生藥品公司 減少或預防第ii型糖尿病患者中心血管事件之方法
CN110038009B (zh) * 2019-05-13 2021-01-08 浙江大学 卡格列净在制备抗肿瘤药物中的应用
PE20230819A1 (es) 2020-02-18 2023-05-19 Novo Nordisk As Composiciones y usos de glp-1
CN112716940A (zh) * 2021-02-18 2021-04-30 苏州大学 卡格列净在制备治疗与stat6蛋白相关疾病的药物中的应用
CN113812378B (zh) * 2021-09-29 2023-02-03 湖北天勤生物技术研究院有限公司 一种食蟹猴肥胖症模型的建立方法及其应用
CN113893349B (zh) * 2021-12-13 2022-07-22 北京大学第三医院(北京大学第三临床医学院) 达格列净及其类似物在制备防治雄性生殖功能障碍的药物中的用途

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EP3349740A1 (en) 2018-07-25
US20200215090A1 (en) 2020-07-09
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