EA031488B1 - Способ лечения гинекологических заболеваний - Google Patents
Способ лечения гинекологических заболеваний Download PDFInfo
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- EA031488B1 EA031488B1 EA201491614A EA201491614A EA031488B1 EA 031488 B1 EA031488 B1 EA 031488B1 EA 201491614 A EA201491614 A EA 201491614A EA 201491614 A EA201491614 A EA 201491614A EA 031488 B1 EA031488 B1 EA 031488B1
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- Eurasian Patent Office
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0034—Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/02—Drugs for genital or sexual disorders; Contraceptives for disorders of the vagina
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/36—Antigestagens
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/04—Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Reproductive Health (AREA)
- Endocrinology (AREA)
- Gynecology & Obstetrics (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Diabetes (AREA)
- Urology & Nephrology (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261614785P | 2012-03-23 | 2012-03-23 | |
| EP12160956.4A EP2641602A1 (en) | 2012-03-23 | 2012-03-23 | Method for treating gynecological diseases |
| PCT/IB2013/052274 WO2013140372A1 (en) | 2012-03-23 | 2013-03-22 | Method for treating gynecological diseases |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| EA201491614A1 EA201491614A1 (ru) | 2015-01-30 |
| EA031488B1 true EA031488B1 (ru) | 2019-01-31 |
Family
ID=45976689
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EA201491614A EA031488B1 (ru) | 2012-03-23 | 2013-03-22 | Способ лечения гинекологических заболеваний |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US10441534B2 (https=) |
| EP (3) | EP2641602A1 (https=) |
| JP (2) | JP2015514700A (https=) |
| KR (1) | KR20140138824A (https=) |
| CN (1) | CN104203246A (https=) |
| AU (1) | AU2013236960B2 (https=) |
| CA (1) | CA2864073A1 (https=) |
| CO (1) | CO7111317A2 (https=) |
| EA (1) | EA031488B1 (https=) |
| GE (1) | GEP201706696B (https=) |
| HK (1) | HK1199827A1 (https=) |
| MX (1) | MX369520B (https=) |
| MY (1) | MY172530A (https=) |
| NZ (1) | NZ630011A (https=) |
| SG (1) | SG11201404921QA (https=) |
| TW (2) | TW201832767A (https=) |
| WO (1) | WO2013140372A1 (https=) |
| ZA (1) | ZA201407575B (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP6995757B2 (ja) | 2015-12-23 | 2022-01-17 | オリック ファーマシューティカルズ，インク． | グルココルチコイド受容体の阻害剤 |
| WO2017112904A1 (en) | 2015-12-23 | 2017-06-29 | Oric Pharmaceuticals, Inc. | Inhibitors of glucocorticoid receptor |
| EP3394078A4 (en) | 2015-12-23 | 2019-11-27 | Oric Pharmaceuticals, Inc. | INHIBITORS OF THE GLUCOCORTICIDE RECEPTOR |
| WO2017165707A1 (en) * | 2016-03-24 | 2017-09-28 | Juniper Pharmaceuticals, Inc. | Vaginal administration of agents for treating and preventing pain associated with gynecological medical procedures |
| NZ753142A (en) | 2016-10-07 | 2020-08-28 | Oric Pharmaceuticals Inc | Inhibitors of glucocorticoid receptor |
| WO2022174074A1 (en) * | 2021-02-12 | 2022-08-18 | The Regents Of The University Of California | Endometriosis-related methods and compositions |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2009095418A1 (en) * | 2008-01-29 | 2009-08-06 | Erin Gainer | Use of ulipristal for treating uterine fibroids |
Family Cites Families (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3545439A (en) | 1968-01-04 | 1970-12-08 | Upjohn Co | Medicated devices and methods |
| US3920805A (en) | 1971-12-09 | 1975-11-18 | Upjohn Co | Pharmaceutical devices and method |
| US4155991A (en) | 1974-10-18 | 1979-05-22 | Schering Aktiengesellschaft | Vaginal ring |
| IL48277A (en) | 1974-10-18 | 1978-03-10 | Schering Ag | Vaginal ring |
| US3995633A (en) | 1975-12-02 | 1976-12-07 | The Procter & Gamble Company | Vaginal Medicament dispensing device |
| US3995634A (en) | 1975-12-02 | 1976-12-07 | The Procter & Gamble Company | Vaginal cavity dispensing means and method |
| US3991760A (en) | 1975-12-02 | 1976-11-16 | The Procter & Gamble Company | Vaginal medicament dispensing means |
| US4286587A (en) | 1978-10-11 | 1981-09-01 | Alza Corporation | Vaginal drug delivery system made from polymer |
| US4292965A (en) | 1978-12-29 | 1981-10-06 | The Population Council, Inc. | Intravaginal ring |
| US4250611A (en) | 1979-04-19 | 1981-02-17 | Alza Corporation | Process for making drug delivery device with reservoir |
| US4596576A (en) | 1984-10-12 | 1986-06-24 | Akzo N.V. | Release system for two or more active substances |
| NL8500470A (nl) | 1985-02-19 | 1986-09-16 | Achel Homesteel Pvba | Intravaginaal orgaan. |
| US4954490A (en) | 1988-06-23 | 1990-09-04 | Research Triangle Institute | 11 β-substituted progesterone analogs |
| FI95768C (fi) | 1993-06-17 | 1996-03-25 | Leiras Oy | Emättimensisäinen antosysteemi |
| US5929262A (en) | 1995-03-30 | 1999-07-27 | The United States Of America As Represented By The Department Of Health And Human Services | Method for preparing 17α-acetoxy-11β-(4-N, N-dimethylaminophyl)-19-Norpregna-4,9-diene-3, 20-dione, intermediates useful in the method, and methods for the preparation of such intermediates |
| US5972372A (en) | 1996-07-31 | 1999-10-26 | The Population Council, Inc. | Intravaginal rings with insertable drug-containing core |
| ES2212912B1 (es) | 2003-01-22 | 2005-10-01 | Crystal Pharma, S.A. | Procedimiento para la obtencion de 17alfa-acetoxi-11beta-(4-n,n-dimetilaminofenil)-19-norpregna-4,9-dien-3,20-diona. |
| CA2516319C (en) | 2003-02-28 | 2012-09-18 | The Government Of The United States Of America, As Represented By The Se Cretary, Department Of Health And Human Services | Method for preparing 17.alpha.-acetoxy-11.beta.-(4-n,n-dimethylaminophenyl)-19-norpregna-4,9-diene-3,20-dione, intermediates thereof, and methods for the preparation of such intermediates |
| CA2573266C (en) | 2004-07-09 | 2011-11-08 | The Population Council, Inc. | Sustained release compositions containing progesterone receptor modulators |
| SI2148681T1 (sl) * | 2007-04-20 | 2016-07-29 | Preglem S.A. | Selektivni modulatorji progesterona v zdravljenju maternične krvavitve |
| EP2359807B1 (en) * | 2008-02-04 | 2017-07-26 | Ferring B.V. | Monolithic intravaginal rings comprising progesterone and methods of making and uses thereof |
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2012
- 2012-03-23 EP EP12160956.4A patent/EP2641602A1/en not_active Withdrawn
-
2013
- 2013-03-22 CN CN201380014168.1A patent/CN104203246A/zh active Pending
- 2013-03-22 JP JP2015501044A patent/JP2015514700A/ja active Pending
- 2013-03-22 GE GEAP201313608A patent/GEP201706696B/en unknown
- 2013-03-22 NZ NZ630011A patent/NZ630011A/en not_active IP Right Cessation
- 2013-03-22 KR KR1020147027575A patent/KR20140138824A/ko not_active Ceased
- 2013-03-22 TW TW107104368A patent/TW201832767A/zh unknown
- 2013-03-22 EP EP13721095.1A patent/EP2827873A1/en not_active Ceased
- 2013-03-22 EA EA201491614A patent/EA031488B1/ru not_active IP Right Cessation
- 2013-03-22 WO PCT/IB2013/052274 patent/WO2013140372A1/en not_active Ceased
- 2013-03-22 AU AU2013236960A patent/AU2013236960B2/en not_active Ceased
- 2013-03-22 MY MYPI2014002228A patent/MY172530A/en unknown
- 2013-03-22 CA CA2864073A patent/CA2864073A1/en not_active Abandoned
- 2013-03-22 US US14/386,726 patent/US10441534B2/en not_active Expired - Fee Related
- 2013-03-22 TW TW102110291A patent/TW201400121A/zh unknown
- 2013-03-22 HK HK15100309.9A patent/HK1199827A1/xx unknown
- 2013-03-22 SG SG11201404921QA patent/SG11201404921QA/en unknown
- 2013-03-22 EP EP17192417.8A patent/EP3363500A1/en not_active Withdrawn
- 2013-03-22 MX MX2014011487A patent/MX369520B/es active IP Right Grant
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2014
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- 2014-10-20 CO CO14231832A patent/CO7111317A2/es unknown
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2018
- 2018-02-13 JP JP2018023604A patent/JP2018109025A/ja active Pending
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| WO2009095418A1 (en) * | 2008-01-29 | 2009-08-06 | Erin Gainer | Use of ulipristal for treating uterine fibroids |
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| DONNEZ J, TATARCHUK T F, BOUCHARD P, PUSCASIU L, ZAKHARENKO N F, IVANOVA T, UGOCSAI G, MARA M, JILLA M P, BESTEL E, TERRILL P, OST: "Ulipristal acetate versus placebo for fibroid treatment before surgery.", NEW ENGLAND JOURNAL OF MEDICINE, THE - NEJM, MASSACHUSETTS MEDICAL SOCIETY, US, vol. 366, no. 5, 2 February 2012 (2012-02-02), US, pages 409 - 420, XP002676689, ISSN: 1533-4406, DOI: 10.1056/NEJMoa1103182 * |
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| AU2013236960A1 (en) | 2014-09-25 |
| WO2013140372A1 (en) | 2013-09-26 |
| GEP201706696B (en) | 2017-07-10 |
| EP2641602A1 (en) | 2013-09-25 |
| JP2018109025A (ja) | 2018-07-12 |
| EP2827873A1 (en) | 2015-01-28 |
| HK1199827A1 (en) | 2015-07-24 |
| CO7111317A2 (es) | 2014-11-10 |
| US10441534B2 (en) | 2019-10-15 |
| JP2015514700A (ja) | 2015-05-21 |
| EA201491614A1 (ru) | 2015-01-30 |
| MX2014011487A (es) | 2015-01-12 |
| MX369520B (es) | 2019-11-11 |
| AU2013236960B2 (en) | 2017-11-23 |
| US20150038476A1 (en) | 2015-02-05 |
| TW201400121A (zh) | 2014-01-01 |
| TW201832767A (zh) | 2018-09-16 |
| ZA201407575B (en) | 2015-12-23 |
| NZ630011A (en) | 2016-12-23 |
| MY172530A (en) | 2019-11-29 |
| KR20140138824A (ko) | 2014-12-04 |
| CN104203246A (zh) | 2014-12-10 |
| EP3363500A1 (en) | 2018-08-22 |
| CA2864073A1 (en) | 2013-09-26 |
| SG11201404921QA (en) | 2014-10-30 |
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