EA028385B1 - Опосредуемое dcc сочетание для получения галофената - Google Patents

Опосредуемое dcc сочетание для получения галофената Download PDF

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Publication number
EA028385B1
EA028385B1 EA201591348A EA201591348A EA028385B1 EA 028385 B1 EA028385 B1 EA 028385B1 EA 201591348 A EA201591348 A EA 201591348A EA 201591348 A EA201591348 A EA 201591348A EA 028385 B1 EA028385 B1 EA 028385B1
Authority
EA
Eurasian Patent Office
Prior art keywords
halofenate
formula
compound
toluene
solution
Prior art date
Application number
EA201591348A
Other languages
English (en)
Russian (ru)
Other versions
EA201591348A1 (ru
Inventor
Цзяньгао Сун
Original Assignee
Саймабэй Терапьютикс, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Саймабэй Терапьютикс, Инк. filed Critical Саймабэй Терапьютикс, Инк.
Publication of EA201591348A1 publication Critical patent/EA201591348A1/ru
Publication of EA028385B1 publication Critical patent/EA028385B1/ru

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
EA201591348A 2013-01-18 2013-01-18 Опосредуемое dcc сочетание для получения галофената EA028385B1 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US2013/022213 WO2014113022A1 (fr) 2013-01-18 2013-01-18 Couplage médié par dcc pour la fabrication d'halofénate

Publications (2)

Publication Number Publication Date
EA201591348A1 EA201591348A1 (ru) 2016-01-29
EA028385B1 true EA028385B1 (ru) 2017-11-30

Family

ID=51209969

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201591348A EA028385B1 (ru) 2013-01-18 2013-01-18 Опосредуемое dcc сочетание для получения галофената

Country Status (9)

Country Link
EP (1) EP2945926A4 (fr)
CN (1) CN105143172B (fr)
AU (1) AU2013374358B2 (fr)
CA (1) CA2901353A1 (fr)
EA (1) EA028385B1 (fr)
HK (1) HK1211020A1 (fr)
NZ (1) NZ711096A (fr)
WO (1) WO2014113022A1 (fr)
ZA (1) ZA201505919B (fr)

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7432394B2 (en) * 2005-09-23 2008-10-07 Metabolex, Inc. Resolution of α-(phenoxy) phenylacetic acid derivatives with naphthyl-alkylamines
US20100093854A1 (en) * 2008-04-03 2010-04-15 Diego Broggini Process for the preparation of (-)-(4-chloro-phenyl)-(3-trifluoromethyl-phenoxy)-acetic acid 2-acetylamino-ethyl ester

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3517050A (en) * 1966-10-03 1970-06-23 Merck & Co Inc Ester and amide derivative of (3-trifluoromethylphenoxy) (4 - halophenyl)acetic acid

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7432394B2 (en) * 2005-09-23 2008-10-07 Metabolex, Inc. Resolution of α-(phenoxy) phenylacetic acid derivatives with naphthyl-alkylamines
US20100093854A1 (en) * 2008-04-03 2010-04-15 Diego Broggini Process for the preparation of (-)-(4-chloro-phenyl)-(3-trifluoromethyl-phenoxy)-acetic acid 2-acetylamino-ethyl ester

Also Published As

Publication number Publication date
AU2013374358B2 (en) 2017-06-08
EP2945926A4 (fr) 2016-09-14
EP2945926A1 (fr) 2015-11-25
NZ711096A (en) 2016-10-28
ZA201505919B (en) 2017-05-31
EA201591348A1 (ru) 2016-01-29
AU2013374358A1 (en) 2015-09-03
CA2901353A1 (fr) 2014-07-24
CN105143172B (zh) 2016-12-14
CN105143172A (zh) 2015-12-09
WO2014113022A1 (fr) 2014-07-24
HK1211020A1 (en) 2016-05-13

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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG TJ TM RU