EA007741B1 - Способ получения 2-(замещенный фенил)-2-гидроксиэтилкарбаматов - Google Patents

Способ получения 2-(замещенный фенил)-2-гидроксиэтилкарбаматов Download PDF

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Publication number
EA007741B1
EA007741B1 EA200400850A EA200400850A EA007741B1 EA 007741 B1 EA007741 B1 EA 007741B1 EA 200400850 A EA200400850 A EA 200400850A EA 200400850 A EA200400850 A EA 200400850A EA 007741 B1 EA007741 B1 EA 007741B1
Authority
EA
Eurasian Patent Office
Prior art keywords
formula
compound
ethers
alcohol
ester
Prior art date
Application number
EA200400850A
Other languages
English (en)
Russian (ru)
Other versions
EA200400850A1 (ru
Inventor
Макс Рей
Томас Оттен
Дэниел Коури
Original Assignee
Орто-Макнейл Фармасьютикал, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Орто-Макнейл Фармасьютикал, Инк. filed Critical Орто-Макнейл Фармасьютикал, Инк.
Priority claimed from PCT/EP2002/014843 external-priority patent/WO2003053916A1/en
Publication of EA200400850A1 publication Critical patent/EA200400850A1/ru
Publication of EA007741B1 publication Critical patent/EA007741B1/ru

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C269/04—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups from amines with formation of carbamate groups
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/325—Carbamic acids; Thiocarbamic acids; Anhydrides or salts thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06—Esters of carbamic acids
    • C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/12—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
EA200400850A 2001-12-21 2002-12-19 Способ получения 2-(замещенный фенил)-2-гидроксиэтилкарбаматов EA007741B1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP01205097 2001-12-21
US41808402P 2002-10-11 2002-10-11
PCT/EP2002/014843 WO2003053916A1 (en) 2001-12-21 2002-12-19 Process for preparing 2-(substituted phenyl) - 2 - hydroxy-ethyl carbamates

Publications (2)

Publication Number Publication Date
EA200400850A1 EA200400850A1 (ru) 2004-10-28
EA007741B1 true EA007741B1 (ru) 2006-12-29

Family

ID=35519523

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200400850A EA007741B1 (ru) 2001-12-21 2002-12-19 Способ получения 2-(замещенный фенил)-2-гидроксиэтилкарбаматов

Country Status (5)

Country Link
KR (2) KR100945720B1 (ko)
CN (1) CN101343243A (ko)
CA (1) CA2752518A1 (ko)
EA (1) EA007741B1 (ko)
ZA (1) ZA200405782B (ko)

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0459455A2 (en) * 1990-05-31 1991-12-04 Chisso Corporation Process for producing optically active alpha-hydroxyesters
US5504108A (en) * 1990-01-12 1996-04-02 The Ohio State University Research Foundation Optically pure 4-aryl-2-hydroxytetronic acids
WO1997026241A1 (en) * 1996-01-16 1997-07-24 Sk Corporation Halogen substituted carbamate compounds from 2-phenyl-1,2-ethanediol
WO2001040168A1 (fr) * 1999-11-29 2001-06-07 Mitsubishi Rayon Co., Ltd. Derive d'acetalsulfonate, son procede de fabrication et obtention d'un derive d'oxyde styrene

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5504108A (en) * 1990-01-12 1996-04-02 The Ohio State University Research Foundation Optically pure 4-aryl-2-hydroxytetronic acids
EP0459455A2 (en) * 1990-05-31 1991-12-04 Chisso Corporation Process for producing optically active alpha-hydroxyesters
WO1997026241A1 (en) * 1996-01-16 1997-07-24 Sk Corporation Halogen substituted carbamate compounds from 2-phenyl-1,2-ethanediol
WO2001040168A1 (fr) * 1999-11-29 2001-06-07 Mitsubishi Rayon Co., Ltd. Derive d'acetalsulfonate, son procede de fabrication et obtention d'un derive d'oxyde styrene

Also Published As

Publication number Publication date
ZA200405782B (en) 2005-08-29
KR20100134082A (ko) 2010-12-22
CN101343243A (zh) 2009-01-14
EA200400850A1 (ru) 2004-10-28
CA2752518A1 (en) 2003-07-03
KR100945720B1 (ko) 2010-03-05
KR20040068588A (ko) 2004-07-31

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MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM

PD4A Registration of transfer of a eurasian patent in accordance with the succession in title
TC4A Change in name of a patent proprietor in a eurasian patent
PC4A Registration of transfer of a eurasian patent by assignment