DOP2008000053A - Inhibidores de akt(proteinas cinasa b) - Google Patents
Inhibidores de akt(proteinas cinasa b)Info
- Publication number
- DOP2008000053A DOP2008000053A DO2008000053A DO2008000053A DOP2008000053A DO P2008000053 A DOP2008000053 A DO P2008000053A DO 2008000053 A DO2008000053 A DO 2008000053A DO 2008000053 A DO2008000053 A DO 2008000053A DO P2008000053 A DOP2008000053 A DO P2008000053A
- Authority
- DO
- Dominican Republic
- Prior art keywords
- cinasa
- proteinas
- akt inhibitors
- compounds
- salt
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/02—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/045—Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
- A61K31/05—Phenols
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/472—Non-condensed isoquinolines, e.g. papaverine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
La presente invención se refiere a 4-[5-(2-amino-etanosulfonil)-isoquinolin-7-il]-fenol o una sal farmacéuticamente aceptable o un hidrato del compuesto o la sal del mismo, como inhibidores de AKt, que son agentes antineoplásicos y/o antivirales, así como también a composiciones que comprende estos compuestos y a métodos para usar estos compuestos.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US80526006P | 2006-06-20 | 2006-06-20 | |
US88576507P | 2007-01-19 | 2007-01-19 |
Publications (1)
Publication Number | Publication Date |
---|---|
DOP2008000053A true DOP2008000053A (es) | 2009-01-15 |
Family
ID=38834248
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DO2008000053A DOP2008000053A (es) | 2006-06-20 | 2008-10-24 | Inhibidores de akt(proteinas cinasa b) |
Country Status (28)
Country | Link |
---|---|
US (1) | US7998977B2 (es) |
EP (1) | EP2035385B1 (es) |
JP (1) | JP2009541335A (es) |
KR (1) | KR101067551B1 (es) |
AR (1) | AR061240A1 (es) |
AT (1) | ATE455102T1 (es) |
AU (1) | AU2007261120A1 (es) |
BR (1) | BRPI0713136A2 (es) |
CA (1) | CA2652612A1 (es) |
CL (1) | CL2007001752A1 (es) |
DE (1) | DE602007004333D1 (es) |
DK (1) | DK2035385T3 (es) |
DO (1) | DOP2008000053A (es) |
EA (1) | EA015712B1 (es) |
EC (1) | ECSP088992A (es) |
ES (1) | ES2336630T3 (es) |
HR (1) | HRP20100147T1 (es) |
IL (1) | IL195005A0 (es) |
MA (1) | MA30757B1 (es) |
MX (1) | MX2008015904A (es) |
NO (1) | NO20090289L (es) |
PE (1) | PE20080338A1 (es) |
PL (1) | PL2035385T3 (es) |
PT (1) | PT2035385E (es) |
SI (1) | SI2035385T1 (es) |
TN (1) | TNSN08529A1 (es) |
TW (1) | TW200812970A (es) |
WO (1) | WO2007149730A2 (es) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP5856843B2 (ja) | 2008-05-27 | 2016-02-10 | アンピオ ファーマシューティカルズ,インコーポレイテッド | ジケトピペラジンを用いた医薬組成物 |
EP2613786A4 (en) | 2010-09-07 | 2013-10-23 | Dmi Acquisition Corp | TREATMENT OF DISEASES |
WO2013055749A1 (en) | 2011-10-10 | 2013-04-18 | Ampio Pharmaceuticals, Inc. | Implantable medical devices with increased immune tolerance, and methods for making and implanting |
KR102032400B1 (ko) | 2011-10-10 | 2019-10-15 | 앰피오 파마슈티컬스 인코퍼레이티드 | 퇴행성 관절 질환의 치료 |
SG10201605205VA (en) | 2011-10-28 | 2016-08-30 | Ampio Pharmaceuticals Inc | Treatment of rhinitis |
WO2014145729A2 (en) | 2013-03-15 | 2014-09-18 | Ampio Pharmaceuticals, Inc. | Compositions for the mobilization, homing, expansion and differentiation of stem cells and methods of using the same |
KR20160104612A (ko) | 2013-07-26 | 2016-09-05 | 업데이트 파마 인코포레이트 | 비산트렌의 치료 효과 개선용 조성물 |
RU2020136589A (ru) | 2014-08-18 | 2020-12-24 | Ампио Фармасьютикалз, Инк. | Лечение дегенеративных заболеваний суставов |
US10123997B2 (en) * | 2015-06-15 | 2018-11-13 | Yong Liao | Target for treating hepatitis B virus |
US11389512B2 (en) | 2015-06-22 | 2022-07-19 | Ampio Pharmaceuticals, Inc. | Use of low molecular weight fractions of human serum albumin in treating diseases |
US10722484B2 (en) | 2016-03-09 | 2020-07-28 | K-Gen, Inc. | Methods of cancer treatment |
CN115843298B (zh) * | 2020-07-22 | 2024-03-29 | 南京正大天晴制药有限公司 | 一种二氢吡啶并[2,3-d]嘧啶酮衍生物的盐及晶型 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL136458A0 (en) | 2000-05-30 | 2001-06-14 | Peptor Ltd | Protein kinase inhibitors |
JP2006521382A (ja) | 2003-03-28 | 2006-09-21 | イーライ リリー アンド カンパニー | Akt(プロテインキナーゼb)阻害剤 |
GB0317315D0 (en) | 2003-07-24 | 2003-08-27 | Astex Technology Ltd | Pharmaceutical compounds |
WO2005054202A1 (en) * | 2003-11-25 | 2005-06-16 | Eli Lilly And Company | 7-phenyl-isoquinoline-5-sulfonylamino derivatives as inhibitors of akt (proteinkinase b) |
-
2007
- 2007-06-06 AR ARP070102429A patent/AR061240A1/es unknown
- 2007-06-12 PL PL07798410T patent/PL2035385T3/pl unknown
- 2007-06-12 DE DE602007004333T patent/DE602007004333D1/de active Active
- 2007-06-12 EA EA200970041A patent/EA015712B1/ru not_active IP Right Cessation
- 2007-06-12 AU AU2007261120A patent/AU2007261120A1/en not_active Abandoned
- 2007-06-12 BR BRPI0713136-4A patent/BRPI0713136A2/pt not_active IP Right Cessation
- 2007-06-12 EP EP07798410A patent/EP2035385B1/en active Active
- 2007-06-12 MX MX2008015904A patent/MX2008015904A/es active IP Right Grant
- 2007-06-12 SI SI200730212T patent/SI2035385T1/sl unknown
- 2007-06-12 JP JP2009516633A patent/JP2009541335A/ja not_active Ceased
- 2007-06-12 CA CA002652612A patent/CA2652612A1/en not_active Abandoned
- 2007-06-12 US US12/300,358 patent/US7998977B2/en not_active Expired - Fee Related
- 2007-06-12 ES ES07798410T patent/ES2336630T3/es active Active
- 2007-06-12 WO PCT/US2007/070945 patent/WO2007149730A2/en active Application Filing
- 2007-06-12 DK DK07798410.2T patent/DK2035385T3/da active
- 2007-06-12 AT AT07798410T patent/ATE455102T1/de active
- 2007-06-12 KR KR1020087030916A patent/KR101067551B1/ko not_active IP Right Cessation
- 2007-06-12 PT PT07798410T patent/PT2035385E/pt unknown
- 2007-06-15 CL CL2007001752A patent/CL2007001752A1/es unknown
- 2007-06-18 PE PE2007000768A patent/PE20080338A1/es not_active Application Discontinuation
- 2007-06-20 TW TW096122142A patent/TW200812970A/zh unknown
-
2008
- 2008-10-24 DO DO2008000053A patent/DOP2008000053A/es unknown
- 2008-10-30 IL IL195005A patent/IL195005A0/en unknown
- 2008-12-18 EC EC2008008992A patent/ECSP088992A/es unknown
- 2008-12-19 TN TNP2008000529A patent/TNSN08529A1/en unknown
-
2009
- 2009-01-19 NO NO20090289A patent/NO20090289L/no not_active Application Discontinuation
- 2009-01-19 MA MA31573A patent/MA30757B1/fr unknown
-
2010
- 2010-03-15 HR HR20100147T patent/HRP20100147T1/hr unknown
Also Published As
Publication number | Publication date |
---|---|
BRPI0713136A2 (pt) | 2012-04-17 |
WO2007149730A2 (en) | 2007-12-27 |
EP2035385B1 (en) | 2010-01-13 |
CL2007001752A1 (es) | 2008-01-18 |
KR101067551B1 (ko) | 2011-09-27 |
DE602007004333D1 (de) | 2010-03-04 |
US7998977B2 (en) | 2011-08-16 |
US20090221633A1 (en) | 2009-09-03 |
AU2007261120A1 (en) | 2007-12-27 |
EP2035385A2 (en) | 2009-03-18 |
ES2336630T3 (es) | 2010-04-14 |
SI2035385T1 (sl) | 2010-05-31 |
JP2009541335A (ja) | 2009-11-26 |
EA015712B1 (ru) | 2011-10-31 |
CA2652612A1 (en) | 2007-12-27 |
PE20080338A1 (es) | 2008-04-25 |
ATE455102T1 (de) | 2010-01-15 |
TW200812970A (en) | 2008-03-16 |
KR20090015978A (ko) | 2009-02-12 |
PT2035385E (pt) | 2010-03-01 |
NO20090289L (no) | 2009-01-19 |
WO2007149730A3 (en) | 2008-04-24 |
PL2035385T3 (pl) | 2010-06-30 |
EA200970041A1 (ru) | 2009-06-30 |
DK2035385T3 (da) | 2010-03-22 |
HRP20100147T1 (hr) | 2010-04-30 |
MX2008015904A (es) | 2009-01-12 |
IL195005A0 (en) | 2009-08-03 |
AR061240A1 (es) | 2008-08-13 |
MA30757B1 (fr) | 2009-10-01 |
ECSP088992A (es) | 2009-01-30 |
TNSN08529A1 (en) | 2010-04-14 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DOP2008000053A (es) | Inhibidores de akt(proteinas cinasa b) | |
CR20110339A (es) | Compuestos útiles para inhibir chk1 | |
EA200970856A1 (ru) | Ингибиторы пути хеджхога | |
CL2011000504A1 (es) | Compuestos derivados de piridin-4-il-tiazol-2il-amida 2-amida-pirrolidin-1,2-dicarboxilico, inhibidores de quinasa de fosfatidil-inositol-3; composicion farmaceutica que comprende a uno de los compuestos; y uso de los compuestos en la preparacion de un medicamento para el tratamiento del cancer. | |
PA8828201A1 (es) | Compuestos triazina como inhibidores mtor y quinasa p13 | |
UY32730A (es) | Inhibidores de cyp17 | |
ATE479687T1 (de) | Kinaseinhibitoren | |
ECSP055867A (es) | Derivados de pirrolopirimidina | |
CR10277A (es) | Pirazolquinolonas como potentes inhibidores de parp | |
CR11510A (es) | Uso de un inhibidor de la gamma-secretasa para tratamiento del cancer | |
CR20140036A (es) | Compuesto inhibidor de la señalización de la trayectoria notch | |
DOP2011000113A (es) | Pirazolilaminopiridinas como inhibidores de fak | |
CL2009000914A1 (es) | Compuestos derivados de 1-ciano-3-pirrolidinil-n-sustituidas-sulfonamidas, inhibidores de catepsina c; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para el tratamiento de una enfermedad pulmonar obstructiva cronica. | |
TN2010000038A1 (en) | Organic compounds | |
EA200900631A1 (ru) | Замещённые пиразолы и триазолы, как ингибиторы кбв (кинезин-белок веретена) | |
CO6440548A2 (es) | 1-/arilsulfonil)-4-(piperazin-1-il)-1h-benzimidazoles como ligandos de 5-hidroxitriptamina-6. | |
CR10199A (es) | Derivados de benzimidazol | |
NI201100035A (es) | Agentes antifúngicos. | |
AR057403A1 (es) | 4- anilino-3-quinolincarbonitrilos para el tratamiento del cancer | |
MX2009003793A (es) | Inhibidores de cinasa. | |
GT200600132A (es) | Una oxindoloxazolidinona como agente antibacteriano | |
CL2009000386A1 (es) | Compuestos derivados de oxazolidinona; composición farmacéutica que contiene dichos compuestos; y su uso para prevenir o tratar una infección bacteriana. |