DK63288A - Fremgangsmaade til fremstilling af 3-(5-cyclopropyl-1,2,4-oxadiazol-3yl)-5,6-dihydro-5-methyl-6-oxo-4h-imidazo(1,5-a)(1,4)benzodiazepin samt 3-cyclopropyl-3-isocyanomethyl-1,2,4-oxadiazol til anvendelse som udgangsmateriale ved fremgangsmaaden - Google Patents

Fremgangsmaade til fremstilling af 3-(5-cyclopropyl-1,2,4-oxadiazol-3yl)-5,6-dihydro-5-methyl-6-oxo-4h-imidazo(1,5-a)(1,4)benzodiazepin samt 3-cyclopropyl-3-isocyanomethyl-1,2,4-oxadiazol til anvendelse som udgangsmateriale ved fremgangsmaaden

Info

Publication number
DK63288A
DK63288A DK063288A DK63288A DK63288A DK 63288 A DK63288 A DK 63288A DK 063288 A DK063288 A DK 063288A DK 63288 A DK63288 A DK 63288A DK 63288 A DK63288 A DK 63288A
Authority
DK
Denmark
Prior art keywords
cyclopropyl
oxadiazol
isocyanomethyl
benzodiazepine
imidazo
Prior art date
Application number
DK063288A
Other languages
English (en)
Other versions
DK160097C (da
DK63288D0 (da
DK160097B (da
Inventor
Frank Waetjen
Mogens Engelstoft
John Bondo Hansen
Leif Helth Jensen
Original Assignee
Ferrosan As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DK220485A external-priority patent/DK220485D0/da
Priority claimed from DK365985A external-priority patent/DK365985D0/da
Priority claimed from DK476985A external-priority patent/DK476985D0/da
Application filed by Ferrosan As filed Critical Ferrosan As
Priority to DK063288A priority Critical patent/DK160097C/da
Publication of DK63288D0 publication Critical patent/DK63288D0/da
Publication of DK63288A publication Critical patent/DK63288A/da
Publication of DK160097B publication Critical patent/DK160097B/da
Application granted granted Critical
Publication of DK160097C publication Critical patent/DK160097C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Diaphragms For Electromechanical Transducers (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Polyethers (AREA)
  • Phenolic Resins Or Amino Resins (AREA)
  • Polyesters Or Polycarbonates (AREA)
DK063288A 1985-05-17 1988-02-08 Fremgangsmaade til fremstilling af 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl-6-oxo-4h-imidazo(1,5-a)(1,4)benzodiazepin samt 3-cyclopropyl-3-isocyanomethyl-1,2,4-oxadiazol til anvendelse som udgangsmateriale ved fremgangsmaaden DK160097C (da)

Priority Applications (1)

Application Number Priority Date Filing Date Title
DK063288A DK160097C (da) 1985-05-17 1988-02-08 Fremgangsmaade til fremstilling af 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl-6-oxo-4h-imidazo(1,5-a)(1,4)benzodiazepin samt 3-cyclopropyl-3-isocyanomethyl-1,2,4-oxadiazol til anvendelse som udgangsmateriale ved fremgangsmaaden

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
DK220485 1985-05-17
DK220485A DK220485D0 (da) 1985-05-17 1985-05-17 Nye oxadiazolylimidazobenzodiazepinderivater samt fremgangsmaade tilfremstilling heraf
DK365985A DK365985D0 (da) 1985-08-12 1985-08-12 Nye oxadiazolylimidazobenzodiazepinderivater samt fremgangsmaade tilfremstilling heraf
DK365985 1985-08-12
DK476985A DK476985D0 (da) 1985-10-17 1985-10-17 Fremgangsmaade til fremstilling af oxadiazolylderivater af imidazobenzodiazepiner og mellemprodukt til brug ved fremgangsmaaden
DK476985 1985-10-17
DK63288 1988-02-08
DK063288A DK160097C (da) 1985-05-17 1988-02-08 Fremgangsmaade til fremstilling af 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl-6-oxo-4h-imidazo(1,5-a)(1,4)benzodiazepin samt 3-cyclopropyl-3-isocyanomethyl-1,2,4-oxadiazol til anvendelse som udgangsmateriale ved fremgangsmaaden

Publications (4)

Publication Number Publication Date
DK63288D0 DK63288D0 (da) 1988-02-08
DK63288A true DK63288A (da) 1988-02-08
DK160097B DK160097B (da) 1991-01-28
DK160097C DK160097C (da) 1991-06-24

Family

ID=27221528

Family Applications (2)

Application Number Title Priority Date Filing Date
DK231686A DK157194C (da) 1985-05-17 1986-05-16 Oxadiazolylimidazobenzodiazepinforbindelse og farmaceutisk praeparat indeholdende samme
DK063288A DK160097C (da) 1985-05-17 1988-02-08 Fremgangsmaade til fremstilling af 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl-6-oxo-4h-imidazo(1,5-a)(1,4)benzodiazepin samt 3-cyclopropyl-3-isocyanomethyl-1,2,4-oxadiazol til anvendelse som udgangsmateriale ved fremgangsmaaden

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK231686A DK157194C (da) 1985-05-17 1986-05-16 Oxadiazolylimidazobenzodiazepinforbindelse og farmaceutisk praeparat indeholdende samme

Country Status (16)

Country Link
US (2) US4622320A (da)
EP (1) EP0201678B1 (da)
JP (1) JPH01279877A (da)
AT (1) ATE35266T1 (da)
AU (2) AU590273B2 (da)
CA (2) CA1256863A (da)
DE (2) DE201678T1 (da)
DK (2) DK157194C (da)
ES (1) ES8707205A1 (da)
FI (1) FI82049C (da)
GR (1) GR861260B (da)
IE (1) IE59494B1 (da)
IL (1) IL78790A (da)
NO (1) NO163228C (da)
NZ (1) NZ216202A (da)
PT (1) PT82594B (da)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3587913D1 (de) * 1984-01-19 1994-10-06 Hoffmann La Roche Imidazodiazepin-Derivate.
US4771051A (en) * 1985-05-17 1988-09-13 A/S Ferrosan 3-substituted-4,5-dihydro-5-oxo imidazoquinazolines, their preparation, and their use in treating benzodiazepin receptor-related ailments
US4622320A (en) * 1985-05-17 1986-11-11 As Ferrosan Oxadiazolylimidazobenzodiazepine, compositions, and method
US4745112A (en) * 1985-05-17 1988-05-17 A/S Ferrosan Oxadiazolylimidazobenzodiazepine, compositions, and method III
EP0274009B1 (en) 1985-10-17 1992-09-09 Novo Nordisk A/S Oxadiazolylacetonitriles, their preparation and use
DK174086D0 (da) * 1986-04-16 1986-04-16 Ferrosan As Nye benzodiazepinderivater samt fremgangsmaade til fremstilling af samme
DK522187D0 (da) * 1987-10-06 1987-10-06 Ferrosan As Imidozothienopyrimidiner, deres fremstilling og anvendelse
GB8823475D0 (en) * 1988-10-06 1988-11-16 Merck Sharp & Dohme Chemical compounds
CA2143246C (en) * 1994-03-16 2000-08-22 Thierry Godel Imidazodiazepines
FI101305B1 (fi) * 1996-03-18 1998-05-29 Map Medical Technologies Oy Radiofarmaseuttisena aineena käyttökelpoiset radiojodatut bentsodiatsepiini-johdannaiset ja niiden käyttö diagnostiikassa
US20090054412A1 (en) * 2007-08-20 2009-02-26 John Alan Kemp Treatment of Sleep Disorders
CN101827597B (zh) * 2007-08-20 2013-03-13 伊沃泰克国际有限责任公司 睡眠障碍的治疗

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4031029A (en) * 1975-07-02 1977-06-21 General Electric Company Process for producing uranium oxide rich compositions from uranium hexafluoride using fluid injection into the reaction zone
CA1143728A (en) * 1979-10-04 1983-03-29 Max Gerecke Imidazodiazepine derivatives
JPS57123180A (en) * 1980-12-17 1982-07-31 Schering Ag 3-substituted beta-carboline, manufacture and psychotropic drug containing same
DK151808C (da) * 1982-11-16 1988-06-20 Ferrosan As Analogifremgangsmaade til fremstilling af oxadiazolylimidazo-oe1,4aa-benzodiazepinderivater
DE3587913D1 (de) * 1984-01-19 1994-10-06 Hoffmann La Roche Imidazodiazepin-Derivate.
AU587802B2 (en) * 1985-03-08 1989-08-31 Ferrosan A/S Novel oxadiazolyl imidazobenzodiazepine derivatives and methods of preparing such compounds
US4622320A (en) * 1985-05-17 1986-11-11 As Ferrosan Oxadiazolylimidazobenzodiazepine, compositions, and method
EP0274009B1 (en) * 1985-10-17 1992-09-09 Novo Nordisk A/S Oxadiazolylacetonitriles, their preparation and use
DK174086D0 (da) * 1986-04-16 1986-04-16 Ferrosan As Nye benzodiazepinderivater samt fremgangsmaade til fremstilling af samme

Also Published As

Publication number Publication date
AU5742986A (en) 1986-11-20
IE861306L (en) 1986-11-17
DK157194C (da) 1990-04-23
DK160097C (da) 1991-06-24
DK231686A (da) 1986-11-18
DK157194B (da) 1989-11-20
DK231686D0 (da) 1986-05-16
JPH01279877A (ja) 1989-11-10
DE3660331D1 (en) 1988-07-28
PT82594A (en) 1986-06-01
NZ216202A (en) 1989-08-29
FI82049B (fi) 1990-09-28
NO163228C (no) 1990-04-25
CA1256864A (en) 1989-07-04
US4622321A (en) 1986-11-11
ES8707205A1 (es) 1987-07-16
DK63288D0 (da) 1988-02-08
AU590273B2 (en) 1989-11-02
AU614407B2 (en) 1991-08-29
DK160097B (da) 1991-01-28
CA1256863A (en) 1989-07-04
IL78790A (en) 1990-01-18
GR861260B (en) 1986-09-10
NO861954L (no) 1986-11-18
EP0201678B1 (en) 1988-06-22
FI862061A0 (fi) 1986-05-16
FI82049C (fi) 1991-01-10
US4622320A (en) 1986-11-11
PT82594B (pt) 1988-03-03
NO163228B (no) 1990-01-15
ES555035A0 (es) 1987-07-16
IE59494B1 (en) 1994-02-23
FI862061A (fi) 1986-11-18
EP0201678A1 (en) 1986-11-20
AU3933389A (en) 1989-11-23
DE201678T1 (de) 1987-02-26
IL78790A0 (en) 1986-08-31
ATE35266T1 (de) 1988-07-15

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