DK220485D0 - Nye oxadiazolylimidazobenzodiazepinderivater samt fremgangsmaade tilfremstilling heraf - Google Patents

Nye oxadiazolylimidazobenzodiazepinderivater samt fremgangsmaade tilfremstilling heraf

Info

Publication number
DK220485D0
DK220485D0 DK220485A DK220485A DK220485D0 DK 220485 D0 DK220485 D0 DK 220485D0 DK 220485 A DK220485 A DK 220485A DK 220485 A DK220485 A DK 220485A DK 220485 D0 DK220485 D0 DK 220485D0
Authority
DK
Denmark
Prior art keywords
oxadiazolylimidazobenzodiazepine
derivatives
new
procedures prepared
procedures
Prior art date
Application number
DK220485A
Other languages
English (en)
Inventor
Frank Waetjen
Mogens Engelstoft
John Bondo Hansen
Leif Helth Jensen
Original Assignee
Frank Waetjen
Mogens Engelstoft
John Bondo Hansen
Leif Helth Jensen
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Frank Waetjen, Mogens Engelstoft, John Bondo Hansen, Leif Helth Jensen filed Critical Frank Waetjen
Priority to DK220485A priority Critical patent/DK220485D0/da
Publication of DK220485D0 publication Critical patent/DK220485D0/da
Priority to US06/816,732 priority patent/US4622320A/en
Priority to US06/816,731 priority patent/US4622321A/en
Priority to AU54013/86A priority patent/AU587802B2/en
Priority to DE198686102535T priority patent/DE197282T1/de
Priority to EP86102535A priority patent/EP0197282A1/en
Priority to DK094686A priority patent/DK157319C/da
Priority to PT82115A priority patent/PT82115B/pt
Priority to FI860894A priority patent/FI860894A/fi
Priority to CA000503329A priority patent/CA1261322A/en
Priority to AT86102951T priority patent/ATE35266T1/de
Priority to EP86102951A priority patent/EP0201678B1/en
Priority to US06/837,100 priority patent/US4670433A/en
Priority to DE8686102951T priority patent/DE3660331D1/de
Priority to DE198686102951T priority patent/DE201678T1/de
Priority to NZ227855A priority patent/NZ227855A/xx
Priority to NO860857A priority patent/NO165545C/no
Priority to ES552803A priority patent/ES8800216A1/es
Priority to GR860639A priority patent/GR860639B/el
Priority to JP61076422A priority patent/JPS6293289A/ja
Priority to AT86104605T priority patent/ATE38671T1/de
Priority to DE8686104605T priority patent/DE3661197D1/de
Priority to EP86104605A priority patent/EP0202441B1/en
Priority to DE198686104605T priority patent/DE202441T1/de
Priority to JP8788386A priority patent/JPS61263979A/ja
Priority to US06/856,945 priority patent/US4745112A/en
Priority to CA000507957A priority patent/CA1256865A/en
Priority to CA000507955A priority patent/CA1256863A/en
Priority to CA000507956A priority patent/CA1256864A/en
Priority to ZA863573A priority patent/ZA863573B/xx
Priority to ZA863574A priority patent/ZA863574B/xx
Priority to AU57428/86A priority patent/AU594676B2/en
Priority to AU57429/86A priority patent/AU590273B2/en
Priority to GR861261A priority patent/GR861261B/el
Priority to GR861260A priority patent/GR861260B/el
Priority to IL78790A priority patent/IL78790A/xx
Priority to IL78791A priority patent/IL78791A/xx
Priority to FI862062A priority patent/FI83325C/fi
Priority to NO861954A priority patent/NO163228C/no
Priority to FI862061A priority patent/FI82049C/fi
Priority to NZ216203A priority patent/NZ216203A/xx
Priority to NZ216202A priority patent/NZ216202A/xx
Priority to ES555035A priority patent/ES8707205A1/es
Priority to IE130686A priority patent/IE59494B1/en
Priority to NZ227983A priority patent/NZ227983A/en
Priority to PT82593A priority patent/PT82593B/pt
Priority to NO86861953A priority patent/NO162859C/no
Priority to IE130786A priority patent/IE59495B1/en
Priority to PT82594A priority patent/PT82594B/pt
Priority to DK231586A priority patent/DK154837C/da
Priority to ES555036A priority patent/ES8707206A1/es
Priority to DK231686A priority patent/DK157194C/da
Priority to IL90183A priority patent/IL90183A/xx
Priority to US06/912,775 priority patent/US4771051A/en
Priority to US06/942,162 priority patent/US4772696A/en
Priority to US06/942,200 priority patent/US4727153A/en
Priority to US07/143,364 priority patent/US4780539A/en
Priority to DK063288A priority patent/DK160097C/da
Priority to DK063388A priority patent/DK159150C/da
Priority to CA000590382A priority patent/CA1266671A/en
Priority to NO890989A priority patent/NO890989D0/no
Priority to JP1065783A priority patent/JPH01279877A/ja
Priority to IL90183A priority patent/IL90183A0/xx
Priority to NO892008A priority patent/NO169228C/no
Priority to FI892920A priority patent/FI892920A/fi
Priority to FI893143A priority patent/FI893143A0/fi
Priority to AU39333/89A priority patent/AU614407B2/en
Priority to IL93355A priority patent/IL93355A0/xx

Links

DK220485A 1985-03-08 1985-05-17 Nye oxadiazolylimidazobenzodiazepinderivater samt fremgangsmaade tilfremstilling heraf DK220485D0 (da)

Priority Applications (68)

Application Number Priority Date Filing Date Title
DK220485A DK220485D0 (da) 1985-05-17 1985-05-17 Nye oxadiazolylimidazobenzodiazepinderivater samt fremgangsmaade tilfremstilling heraf
US06/816,732 US4622320A (en) 1985-05-17 1986-01-06 Oxadiazolylimidazobenzodiazepine, compositions, and method
US06/816,731 US4622321A (en) 1985-05-17 1986-01-06 Oxadiazolylimidazobenzodiazepine, compositions, and method
AU54013/86A AU587802B2 (en) 1985-03-08 1986-02-24 Novel oxadiazolyl imidazobenzodiazepine derivatives and methods of preparing such compounds
DE198686102535T DE197282T1 (de) 1985-03-08 1986-02-27 Oxadiazolyl-imidazobenzodiazepinderivate und methoden zu ihrer herstellung.
EP86102535A EP0197282A1 (en) 1985-03-08 1986-02-27 Novel oxadiazolyl imidazobenzodiazepine derivatives and methods of preparing such compounds
DK094686A DK157319C (da) 1985-03-08 1986-02-28 Oxadiazolylimidazobenzodiazepinderivater
PT82115A PT82115B (pt) 1985-03-08 1986-02-28 Processo de preparacao de derivados de oxadiazolilimidazobenzodiazepina e dos seus intermediarios
FI860894A FI860894A (fi) 1985-03-08 1986-03-03 Nya oxadiazolyl -imidazobensodiazepinderivat och foerfarande foer framstaellning av dylika foereningar.
CA000503329A CA1261322A (en) 1985-03-08 1986-03-05 OXADIAZOLYLIMIDABENZODIAZEPINE DERIVATIVES; METHOD OF PREPARATION; PHARMACEUTICAL COMPOSITIONS AND TREATMENT BASED ON THESE DERIVATIVES
AT86102951T ATE35266T1 (de) 1985-05-17 1986-03-06 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6dihydro-5-methyl-6-oxo-4h-imidazo(1,5a)(1,4)benzodiazepin, verfahren zu seiner herstellung und pharmazeutische zubereitungen.
EP86102951A EP0201678B1 (en) 1985-05-17 1986-03-06 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl-6-oxo-4h-imidazo(1,5-a)(1,4)benzodiazepine, a process for its preparation and pharmaceutical compositions
US06/837,100 US4670433A (en) 1985-03-08 1986-03-06 Oxadiazolyl imidazobenzodiazepine derivatives pharmaceutical compositions thereof, and method of treating therewith
DE8686102951T DE3660331D1 (en) 1985-05-17 1986-03-06 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl-6-oxo-4h-imidazo(1,5-a)(1,4)benzodiazepine, a process for its preparation and pharmaceutical compositions
DE198686102951T DE201678T1 (de) 1985-05-17 1986-03-06 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl-6-oxo-4h-imidazo(1,5-a)(1,4)benzodiazepin, verfahren zu seiner herstellung und pharmazeutische zubereitungen.
NZ227855A NZ227855A (en) 1985-03-08 1986-03-07 Isocyanomethyl derivatives of oxadiazoles
NO860857A NO165545C (no) 1985-03-08 1986-03-07 Analogifremgangsmaate for fremstilling av terapeutisk aktive nye oksadiazolimidazo-benzodiazepinderivater.
ES552803A ES8800216A1 (es) 1985-03-08 1986-03-07 Procedimiento para preparar derivados de oxadiazol imidazobenzodiazepina
GR860639A GR860639B (en) 1985-03-08 1986-03-07 Novel oxadiazolyl imidazobenzodiazepine derivates and methods of preaparing such compounds
JP61076422A JPS6293289A (ja) 1985-05-17 1986-04-02 オキサジアゾリルイミダゾベンゾジアゼピン及びその合成法,並びに抗けいれん及び抗不安剤
AT86104605T ATE38671T1 (de) 1985-05-17 1986-04-04 Oxadiazolylimidazobenzodiazepine, verfahren zu ihrer herstellung und pharmazeutische zubereitungen.
DE8686104605T DE3661197D1 (en) 1985-05-17 1986-04-04 Oxadiazolylimidazobenzodiazepines, process for their preparation and pharmaceutical compositions
EP86104605A EP0202441B1 (en) 1985-05-17 1986-04-04 Oxadiazolylimidazobenzodiazepines, process for their preparation and pharmaceutical compositions
DE198686104605T DE202441T1 (de) 1985-05-17 1986-04-04 Oxadiazolylimidazobenzodiazepine, verfahren zu ihrer herstellung und pharmazeutische zubereitungen.
JP8788386A JPS61263979A (ja) 1985-05-17 1986-04-16 オキサジアゾリルイミダゾベンゾジアゼピン、並びに抗けいれん及び抗不安剤
US06/856,945 US4745112A (en) 1985-05-17 1986-04-28 Oxadiazolylimidazobenzodiazepine, compositions, and method III
CA000507957A CA1256865A (en) 1985-05-17 1986-04-30 Oxadiazolylimidazobenzodiazepine, compositions, and method iii
CA000507955A CA1256863A (en) 1985-05-17 1986-04-30 Oxadiazolylimidazobenzodiazepine, compositions, and method i
CA000507956A CA1256864A (en) 1985-05-17 1986-04-30 Oxadiazolylimidazobenzodiazepine, compositions, and method ii
ZA863573A ZA863573B (en) 1985-05-17 1986-05-14 Oxadiazolyl imidazobenzodiazepine compound,pharmaceutical composition containing said compound and method of preparing said compound
ZA863574A ZA863574B (en) 1985-05-17 1986-05-14 Oxadiazolyl imidazobenzodiazepine compound,pharmaceutical composition containing said compound and method of preparing said compound
AU57428/86A AU594676B2 (en) 1985-05-17 1986-05-14 Oxadiazolyl imidazobenaodiazepine compound, pharmaceutical composition containing said compound, method of preparing said compound and method of treating a central nervous system ailment
AU57429/86A AU590273B2 (en) 1985-05-17 1986-05-14 Oxydiazolyl imidazobenzodiazepine compound, pharmaceutical composition containing said compound, method of preparing said compound and method of treating a central nervous system ailment
GR861261A GR861261B (en) 1985-05-17 1986-05-14 Oxadiazolyl imidazobenzodiazepine compound pharmaceutical composition containing said compound method of preparing said compound and method of treating a central nervous system ailment
GR861260A GR861260B (en) 1985-05-17 1986-05-14 Oxadiazolyl imidazobenzodiazepine compound pharmaceutial composition containing said compound method of preparing said compound and method of treating a central nervous system ailment
IL78790A IL78790A (en) 1985-05-17 1986-05-15 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl 6-oxo-4h-imidazo(1,5-a)(1,4)benzodiazepine,a pharmaceutical composition containing it and a method of preparing it
IL78791A IL78791A (en) 1985-05-17 1986-05-15 7-substituted-3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl-6-oxo-4h-imidazo(1,5-a)-(1,4)-benzodiazepines,pharmaceutical compositions containing them and method of preparing them
FI862062A FI83325C (fi) 1985-05-17 1986-05-16 Foerfarande foer framstaellning av 7- substituerade 3-(5-cyklopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-metyl -6-oxo-4h-imidazo(1,5-a)(1,4) bensodiazepiner.
NO861954A NO163228C (no) 1985-05-17 1986-05-16 Analogifremgangsmaate til fremstilling av terapeutisk aktive oksadiazolylimidazobenzodiazepinforbindelse.
FI862061A FI82049C (fi) 1985-05-17 1986-05-16 Foerfarande foer framstaellning av saosom laekemedel anvaendbar 3-(5-cyklopropyl-1,2,4-oxadiazol-3-yl) 5,6-dihydro-5-metyl-6-oxo-4h-imidazo-(1,5-a)(1,4)bensodiazepin.
NZ216203A NZ216203A (en) 1985-05-17 1986-05-16 Oxydiazolyl imidazobenzodiazepines and pharmaceutical compositions
NZ216202A NZ216202A (en) 1985-05-17 1986-05-16 An oxadiazolyl imidazobenzodiazepine compound and pharmaceutical compositions thereof
ES555035A ES8707205A1 (es) 1985-05-17 1986-05-16 Procedimiento para preparar un derivado de oxadiazolilimidazobenzodiazepina
IE130686A IE59494B1 (en) 1985-05-17 1986-05-16 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5--methyl-6-oxo-4h-imidazo(1,4-a)(1,4)benzodiazepine, a process for its preparation and pharmaceutical compositions
NZ227983A NZ227983A (en) 1985-05-17 1986-05-16 5 cyclopropyl-3-isocyanomethyl-1,2,4-oxidiazole
PT82593A PT82593B (pt) 1985-05-17 1986-05-16 Processo de preparacao da oxadiazolil-imidazobenzodiazepina e das composicoes farmaceuticas que a contem
NO86861953A NO162859C (no) 1985-05-17 1986-05-16 Analogifremgangsmaate for fremstilling av terapeutisk aktive oksadiazolylimidazobenzodiazepinforbindelser.
IE130786A IE59495B1 (en) 1985-05-17 1986-05-16 Oxadiazolylimidazobenzodiazepines, process for their preparation and pharmaceutical compositions
PT82594A PT82594B (pt) 1985-05-17 1986-05-16 Processo de preparacao da oxadiazolil-imidazobenzodiazepina e das composicoes farmaceuticas que a contem
DK231586A DK154837C (da) 1985-05-17 1986-05-16 Oxadiazolylimidazobenzodiazepinforbindelse og farmaceutisk praeparat indeholdende samme
ES555036A ES8707206A1 (es) 1985-05-17 1986-05-16 Procedimiento para preparar derivados de oxadiazolilimidazobenzodiazepina
DK231686A DK157194C (da) 1985-05-17 1986-05-16 Oxadiazolylimidazobenzodiazepinforbindelse og farmaceutisk praeparat indeholdende samme
IL90183A IL90183A (en) 1985-05-17 1986-05-18 5-cyclopropyl-3-isocyanomethyl-1,2,4-oxadiazole
US06/912,775 US4771051A (en) 1985-05-17 1986-09-26 3-substituted-4,5-dihydro-5-oxo imidazoquinazolines, their preparation, and their use in treating benzodiazepin receptor-related ailments
US06/942,162 US4772696A (en) 1985-03-08 1986-12-16 Oxadiazolyl imidazobenzodiazepine process
US06/942,200 US4727153A (en) 1985-03-08 1986-12-16 Oxadiazolyl intermediates
US07/143,364 US4780539A (en) 1985-05-17 1988-01-12 3-substituted-4,5-dihydro-5-oxo imidazoquinazolines, their preparation, and their use in treating benzodiazepin receptor-related ailments
DK063288A DK160097C (da) 1985-05-17 1988-02-08 Fremgangsmaade til fremstilling af 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl-6-oxo-4h-imidazo(1,5-a)(1,4)benzodiazepin samt 3-cyclopropyl-3-isocyanomethyl-1,2,4-oxadiazol til anvendelse som udgangsmateriale ved fremgangsmaaden
DK063388A DK159150C (da) 1985-03-08 1988-02-08 Isocyanomethylforbindelse samt fremgangsmaade til fremstilling af et oxadiazolimidazobenzodiazepinderivat
CA000590382A CA1266671A (en) 1985-03-08 1989-02-07 Oxadiazolyl imidazobenzodiazepine derivatives, a method of preparing the same, pharmaceutical compositions thereof, and method of treating therewith
NO890989A NO890989D0 (no) 1985-03-08 1989-03-08 Isocyanometylforbindelse samt fremgangsmaate for fremstilling av et oksadiazolimidazobenzodiazepinderivat.
JP1065783A JPH01279877A (ja) 1985-05-17 1989-03-17 5―シクロプロピル―3―イソシアノメチル―1,2,4―オキサジアゾール
IL90183A IL90183A0 (en) 1985-05-17 1989-05-04 Substituted 1,2,4-oxadiazole
NO892008A NO169228C (no) 1985-05-17 1989-05-19 5-cyklopropyl-3-isocyanometyl-1,2,4-oksadiazol
FI892920A FI892920A (fi) 1985-05-17 1989-06-14 Substituerad 1,2,4-oxadiazol.
FI893143A FI893143A0 (fi) 1985-03-08 1989-06-28 Isocyanometylfoerening samt foerfarande foer framstaellning av oxadiazolylimidazobensodiazepin -derivat.
AU39333/89A AU614407B2 (en) 1985-05-17 1989-08-04 Oxadiazolyl imidazobenzodiazepine compound, pharmaceutical composition containing said compound, method of preparing said compound and method of treating a central nervous system ailment
IL93355A IL93355A0 (en) 1985-03-08 1990-02-12 Isocyanomethyl derivatives

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DK220485A DK220485D0 (da) 1985-05-17 1985-05-17 Nye oxadiazolylimidazobenzodiazepinderivater samt fremgangsmaade tilfremstilling heraf

Publications (1)

Publication Number Publication Date
DK220485D0 true DK220485D0 (da) 1985-05-17

Family

ID=8110769

Family Applications (1)

Application Number Title Priority Date Filing Date
DK220485A DK220485D0 (da) 1985-03-08 1985-05-17 Nye oxadiazolylimidazobenzodiazepinderivater samt fremgangsmaade tilfremstilling heraf

Country Status (3)

Country Link
JP (2) JPS6293289A (da)
DK (1) DK220485D0 (da)
ZA (2) ZA863574B (da)

Also Published As

Publication number Publication date
JPS6293289A (ja) 1987-04-28
ZA863573B (en) 1987-01-28
JPH0329795B2 (da) 1991-04-25
JPS61263979A (ja) 1986-11-21
JPH0127074B2 (da) 1989-05-26
ZA863574B (en) 1987-01-28

Similar Documents

Publication Publication Date Title
DK312386A (da) N-aralkyl-piperidenmethanolderivater samt disses fremstilling
DK289886A (da) Substituerede 3-phenyl-4-cyanopyrrol-derivater samt deres fremstilling og anvendelse
DK165249C (da) Imidazooe4,5-baaquinolin-2-thionderivater samt fremgangsmaade til fremstilling deraf
DK149786D0 (da) Nye forbindelser
DK62586D0 (da) Nye forbindelser
DK29686A (da) 13beta-alkyl-milbemycinderivater samt deres fremstilling og anvendelse
DK499886D0 (da) Nye forbindelser
DK139286D0 (da) Inden- og naphthalenderivater
NO872778L (no) Nye 4-pyridonderivater samt fremgangsmŸte for fremstilling derav.
DK163584C (da) 7-amino-3-propenylcephalosporinsyrederivater samt fremgangsmaade til fremstilling deraf
DK109186A (da) Dihydropyridazinonderivater
DK470886D0 (da) Oxazol- og isoxazolderivater
DE3680771D1 (de) Isoxazolopyridophenoxazin- und isothiazolopyridophenoxazinderivate.
DK162186A (da) Aminoketonderivater samt laegemidler indeholdende saadanne derivater
DK491786D0 (da) Dichloranilinderivater
DK556386D0 (da) Quinilinderivater
DE3680775D1 (de) Isoxazolopyridobenzoxazin- und isothiazolopyridobenzoxazinderivate.
DK303886A (da) Secocanthinderivater
DK108085D0 (da) Nye oxadiazolylimidazobenzodiazepinderivater samt fremgangsmaade tilfremstilling heraf
DK220485D0 (da) Nye oxadiazolylimidazobenzodiazepinderivater samt fremgangsmaade tilfremstilling heraf
DK108185D0 (da) Nye oxadiazolylimidazobenzodiazepinderivater samt fremgangsmaade tilfremstilling heraf
DK365985D0 (da) Nye oxadiazolylimidazobenzodiazepinderivater samt fremgangsmaade tilfremstilling heraf
DE3662889D1 (de) Tetrahydrofurancarboxylic-acid derivatives
KR880700821A (ko) 데--데옥시테이코플라닌 유도체
FR2588259B1 (fr) Bis-acridiniques monopontes et bis-acridiniques bipontes