NO163228C - Analogifremgangsmaate til fremstilling av terapeutisk aktive oksadiazolylimidazobenzodiazepinforbindelse. - Google Patents

Analogifremgangsmaate til fremstilling av terapeutisk aktive oksadiazolylimidazobenzodiazepinforbindelse.

Info

Publication number
NO163228C
NO163228C NO861954A NO861954A NO163228C NO 163228 C NO163228 C NO 163228C NO 861954 A NO861954 A NO 861954A NO 861954 A NO861954 A NO 861954A NO 163228 C NO163228 C NO 163228C
Authority
NO
Norway
Prior art keywords
oxadiazolylimidazobenzodiazepin
preparation
connection
therapeutic active
analogue procedure
Prior art date
Application number
NO861954A
Other languages
English (en)
Norwegian (no)
Other versions
NO163228B (no
NO861954L (no
Inventor
Frank Waetjen
Mogens Engelstoft
John Bondo Hansen
Leif Helth Jensen
Original Assignee
Ferrosan As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DK220485A external-priority patent/DK220485D0/da
Priority claimed from DK365985A external-priority patent/DK365985D0/da
Priority claimed from DK476985A external-priority patent/DK476985D0/da
Application filed by Ferrosan As filed Critical Ferrosan As
Publication of NO861954L publication Critical patent/NO861954L/no
Priority to NO892008A priority Critical patent/NO169228C/no
Publication of NO163228B publication Critical patent/NO163228B/no
Publication of NO163228C publication Critical patent/NO163228C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/061,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Diaphragms For Electromechanical Transducers (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Polyethers (AREA)
  • Phenolic Resins Or Amino Resins (AREA)
  • Polyesters Or Polycarbonates (AREA)
NO861954A 1985-05-17 1986-05-16 Analogifremgangsmaate til fremstilling av terapeutisk aktive oksadiazolylimidazobenzodiazepinforbindelse. NO163228C (no)

Priority Applications (1)

Application Number Priority Date Filing Date Title
NO892008A NO169228C (no) 1985-05-17 1989-05-19 5-cyklopropyl-3-isocyanometyl-1,2,4-oksadiazol

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DK220485A DK220485D0 (da) 1985-05-17 1985-05-17 Nye oxadiazolylimidazobenzodiazepinderivater samt fremgangsmaade tilfremstilling heraf
DK365985A DK365985D0 (da) 1985-08-12 1985-08-12 Nye oxadiazolylimidazobenzodiazepinderivater samt fremgangsmaade tilfremstilling heraf
DK476985A DK476985D0 (da) 1985-10-17 1985-10-17 Fremgangsmaade til fremstilling af oxadiazolylderivater af imidazobenzodiazepiner og mellemprodukt til brug ved fremgangsmaaden

Publications (3)

Publication Number Publication Date
NO861954L NO861954L (no) 1986-11-18
NO163228B NO163228B (no) 1990-01-15
NO163228C true NO163228C (no) 1990-04-25

Family

ID=27221528

Family Applications (1)

Application Number Title Priority Date Filing Date
NO861954A NO163228C (no) 1985-05-17 1986-05-16 Analogifremgangsmaate til fremstilling av terapeutisk aktive oksadiazolylimidazobenzodiazepinforbindelse.

Country Status (16)

Country Link
US (2) US4622321A (da)
EP (1) EP0201678B1 (da)
JP (1) JPH01279877A (da)
AT (1) ATE35266T1 (da)
AU (2) AU590273B2 (da)
CA (2) CA1256864A (da)
DE (2) DE3660331D1 (da)
DK (2) DK157194C (da)
ES (1) ES8707205A1 (da)
FI (1) FI82049C (da)
GR (1) GR861260B (da)
IE (1) IE59494B1 (da)
IL (1) IL78790A (da)
NO (1) NO163228C (da)
NZ (1) NZ216202A (da)
PT (1) PT82594B (da)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1252462A (en) * 1984-01-19 1989-04-11 Walter Hunkeler Imidazodiazepine derivatives
US4745112A (en) * 1985-05-17 1988-05-17 A/S Ferrosan Oxadiazolylimidazobenzodiazepine, compositions, and method III
US4622321A (en) * 1985-05-17 1986-11-11 As Ferrosan Oxadiazolylimidazobenzodiazepine, compositions, and method
US4771051A (en) * 1985-05-17 1988-09-13 A/S Ferrosan 3-substituted-4,5-dihydro-5-oxo imidazoquinazolines, their preparation, and their use in treating benzodiazepin receptor-related ailments
DE3686723T2 (de) * 1985-10-17 1993-04-01 Novonordisk As Oxadiazolylacetonitrile, ihre herstellung und anwendung.
DK174086D0 (da) * 1986-04-16 1986-04-16 Ferrosan As Nye benzodiazepinderivater samt fremgangsmaade til fremstilling af samme
DK522187D0 (da) * 1987-10-06 1987-10-06 Ferrosan As Imidozothienopyrimidiner, deres fremstilling og anvendelse
GB8823475D0 (en) * 1988-10-06 1988-11-16 Merck Sharp & Dohme Chemical compounds
CA2143246C (en) * 1994-03-16 2000-08-22 Thierry Godel Imidazodiazepines
FI101305B (fi) * 1996-03-18 1998-05-29 Map Medical Technologies Oy Radiofarmaseuttisena aineena käyttökelpoiset radiojodatut bentsodiatse piini-johdannaiset ja niiden käyttö diagnostiikassa
US20090054412A1 (en) * 2007-08-20 2009-02-26 John Alan Kemp Treatment of Sleep Disorders
EP2190435B1 (en) * 2007-08-20 2018-05-30 Evotec International GmbH Treatment of sleep disorders

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4031029A (en) * 1975-07-02 1977-06-21 General Electric Company Process for producing uranium oxide rich compositions from uranium hexafluoride using fluid injection into the reaction zone
CA1143728A (en) * 1979-10-04 1983-03-29 Max Gerecke Imidazodiazepine derivatives
JPS57123180A (en) * 1980-12-17 1982-07-31 Schering Ag 3-substituted beta-carboline, manufacture and psychotropic drug containing same
DK151808C (da) * 1982-11-16 1988-06-20 Ferrosan As Analogifremgangsmaade til fremstilling af oxadiazolylimidazo-oe1,4aa-benzodiazepinderivater
CA1252462A (en) * 1984-01-19 1989-04-11 Walter Hunkeler Imidazodiazepine derivatives
AU587802B2 (en) * 1985-03-08 1989-08-31 Ferrosan A/S Novel oxadiazolyl imidazobenzodiazepine derivatives and methods of preparing such compounds
US4622321A (en) * 1985-05-17 1986-11-11 As Ferrosan Oxadiazolylimidazobenzodiazepine, compositions, and method
DE3686723T2 (de) * 1985-10-17 1993-04-01 Novonordisk As Oxadiazolylacetonitrile, ihre herstellung und anwendung.
DK174086D0 (da) * 1986-04-16 1986-04-16 Ferrosan As Nye benzodiazepinderivater samt fremgangsmaade til fremstilling af samme

Also Published As

Publication number Publication date
FI862061A0 (fi) 1986-05-16
DE201678T1 (de) 1987-02-26
AU614407B2 (en) 1991-08-29
DK157194C (da) 1990-04-23
DK63288D0 (da) 1988-02-08
PT82594B (pt) 1988-03-03
IL78790A0 (en) 1986-08-31
NZ216202A (en) 1989-08-29
DK63288A (da) 1988-02-08
US4622320A (en) 1986-11-11
CA1256864A (en) 1989-07-04
PT82594A (en) 1986-06-01
AU590273B2 (en) 1989-11-02
IE59494B1 (en) 1994-02-23
ATE35266T1 (de) 1988-07-15
IE861306L (en) 1986-11-17
FI82049B (fi) 1990-09-28
EP0201678B1 (en) 1988-06-22
FI862061A (fi) 1986-11-18
FI82049C (fi) 1991-01-10
AU5742986A (en) 1986-11-20
DK160097C (da) 1991-06-24
GR861260B (en) 1986-09-10
NO163228B (no) 1990-01-15
EP0201678A1 (en) 1986-11-20
NO861954L (no) 1986-11-18
CA1256863A (en) 1989-07-04
DK160097B (da) 1991-01-28
IL78790A (en) 1990-01-18
AU3933389A (en) 1989-11-23
ES8707205A1 (es) 1987-07-16
DK157194B (da) 1989-11-20
DK231686D0 (da) 1986-05-16
US4622321A (en) 1986-11-11
ES555035A0 (es) 1987-07-16
DE3660331D1 (en) 1988-07-28
DK231686A (da) 1986-11-18
JPH01279877A (ja) 1989-11-10

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