DK387889A - Makrolider, og farmaceutiske praeparater med indhold af saadanne forbindelser - Google Patents

Makrolider, og farmaceutiske praeparater med indhold af saadanne forbindelser Download PDF

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Publication number
DK387889A
DK387889A DK387889A DK387889A DK387889A DK 387889 A DK387889 A DK 387889A DK 387889 A DK387889 A DK 387889A DK 387889 A DK387889 A DK 387889A DK 387889 A DK387889 A DK 387889A
Authority
DK
Denmark
Prior art keywords
represent
compounds
alkyl
macrolides
groups including
Prior art date
Application number
DK387889A
Other languages
Danish (da)
English (en)
Other versions
DK387889D0 (da
Inventor
Martin Edward Cooper
David Keith Donald
David Norman Hardern
Original Assignee
Fisons Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB878728821A external-priority patent/GB8728821D0/en
Priority claimed from GB878728820A external-priority patent/GB8728820D0/en
Priority claimed from GB888803370A external-priority patent/GB8803370D0/en
Priority claimed from GB888803375A external-priority patent/GB8803375D0/en
Priority claimed from GB888803373A external-priority patent/GB8803373D0/en
Priority claimed from GB888803371A external-priority patent/GB8803371D0/en
Priority claimed from GB888803374A external-priority patent/GB8803374D0/en
Priority claimed from GB888803372A external-priority patent/GB8803372D0/en
Priority claimed from GB888803377A external-priority patent/GB8803377D0/en
Priority claimed from GB888809174A external-priority patent/GB8809174D0/en
Priority claimed from GB888817624A external-priority patent/GB8817624D0/en
Priority claimed from GB888818426A external-priority patent/GB8818426D0/en
Publication of DK387889A publication Critical patent/DK387889A/da
Publication of DK387889D0 publication Critical patent/DK387889D0/da
Application filed by Fisons Plc filed Critical Fisons Plc

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Immunology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Steroid Compounds (AREA)
DK387889A 1987-12-09 1989-08-08 Makrolider, og farmaceutiske praeparater med indhold af saadanne forbindelser DK387889A (da)

Applications Claiming Priority (13)

Application Number Priority Date Filing Date Title
GB878728821A GB8728821D0 (en) 1987-12-09 1987-12-09 Compounds
GB878728820A GB8728820D0 (en) 1987-12-09 1987-12-09 Compounds
GB888803375A GB8803375D0 (en) 1988-02-13 1988-02-13 Compound
GB888803370A GB8803370D0 (en) 1988-02-13 1988-02-13 Compound
GB888803373A GB8803373D0 (en) 1988-02-13 1988-02-13 Compound
GB888803371A GB8803371D0 (en) 1988-02-13 1988-02-13 Compound
GB888803374A GB8803374D0 (en) 1988-02-13 1988-02-13 Compound
GB888803372A GB8803372D0 (en) 1988-02-13 1988-02-13 Compound
GB888803377A GB8803377D0 (en) 1988-02-13 1988-02-13 Compound
GB888809174A GB8809174D0 (en) 1988-04-19 1988-04-19 Compounds
GB888817624A GB8817624D0 (en) 1988-07-23 1988-07-23 Compounds
GB888818426A GB8818426D0 (en) 1988-08-03 1988-08-03 Compounds
PCT/GB1988/001093 WO1989005304A1 (en) 1987-12-09 1988-12-02 Macrocyclic compounds

Publications (2)

Publication Number Publication Date
DK387889D0 DK387889D0 (da) 1989-08-08
DK387889A true DK387889A (da) 1989-08-08

Family

ID=27583057

Family Applications (1)

Application Number Title Priority Date Filing Date
DK387889A DK387889A (da) 1987-12-09 1989-08-08 Makrolider, og farmaceutiske praeparater med indhold af saadanne forbindelser

Country Status (16)

Country Link
EP (2) EP0323042A1 (ko)
JP (1) JP2799208B2 (ko)
KR (1) KR900700494A (ko)
CN (1) CN1033458A (ko)
AT (1) ATE120466T1 (ko)
AU (1) AU630866B2 (ko)
CA (1) CA1339128C (ko)
DE (1) DE3853477T2 (ko)
DK (1) DK387889A (ko)
ES (1) ES2071681T3 (ko)
FI (1) FI90550C (ko)
IE (1) IE66163B1 (ko)
IL (1) IL88629A (ko)
NO (1) NO893166D0 (ko)
NZ (1) NZ227251A (ko)
WO (1) WO1989005304A1 (ko)

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US4650803A (en) * 1985-12-06 1987-03-17 University Of Kansas Prodrugs of rapamycin
EP0349061B1 (en) * 1988-06-29 1995-03-29 Merck & Co. Inc. Immunosuppressant agent
ATE131536T1 (de) * 1988-08-01 1995-12-15 Fujisawa Pharmaceutical Co Fr-901154- und fr-901155-derivate, verfahren zu ihrer herstellung
EP0356399A3 (en) * 1988-08-26 1991-03-20 Sandoz Ag Substituted 4-azatricyclo (22.3.1.04.9) octacos-18-ene derivatives, their preparation and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
EP0346427B1 (en) 1995-03-29
JPH02502463A (ja) 1990-08-09
WO1989005304A1 (en) 1989-06-15
NZ227251A (en) 1990-02-26
FI90550C (fi) 1994-02-25
DK387889D0 (da) 1989-08-08
EP0346427A1 (en) 1989-12-20
AU2822889A (en) 1989-07-05
EP0323042A1 (en) 1989-07-05
FI893750A0 (fi) 1989-08-09
ATE120466T1 (de) 1995-04-15
IL88629A (en) 1994-04-12
ES2071681T3 (es) 1995-07-01
IE66163B1 (en) 1995-12-13
CA1339128C (en) 1997-07-29
KR900700494A (ko) 1990-08-13
NO893166L (no) 1989-08-04
FI90550B (fi) 1993-11-15
JP2799208B2 (ja) 1998-09-17
CN1033458A (zh) 1989-06-21
IE883662L (en) 1989-06-09
DE3853477T2 (de) 1995-11-09
NO893166D0 (no) 1989-08-04
DE3853477D1 (de) 1995-05-04
AU630866B2 (en) 1992-11-12

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