DK3529248T3 - Farmaceutiske sammensætninger - Google Patents

Farmaceutiske sammensætninger Download PDF

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Publication number
DK3529248T3
DK3529248T3 DK17790813.4T DK17790813T DK3529248T3 DK 3529248 T3 DK3529248 T3 DK 3529248T3 DK 17790813 T DK17790813 T DK 17790813T DK 3529248 T3 DK3529248 T3 DK 3529248T3
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DK
Denmark
Prior art keywords
pharmaceutical compositions
pharmaceutical
compositions
Prior art date
Application number
DK17790813.4T
Other languages
Danish (da)
English (en)
Inventor
Neil Anthony Pegg
Stuart Thomas Onions
David Michel Adrien Taddei
Jonathan Shannon
Silvia Paoletta
Richard James Brown
Don Smyth
Gareth Harbottle
Original Assignee
Cellcentric Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cellcentric Ltd filed Critical Cellcentric Ltd
Application granted granted Critical
Publication of DK3529248T3 publication Critical patent/DK3529248T3/da

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/422Oxazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Dermatology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK17790813.4T 2016-10-18 2017-10-18 Farmaceutiske sammensætninger DK3529248T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB1617630.7A GB201617630D0 (en) 2016-10-18 2016-10-18 Pharmaceutical compounds
PCT/GB2017/053152 WO2018073586A1 (en) 2016-10-18 2017-10-18 Pharmaceutical compounds

Publications (1)

Publication Number Publication Date
DK3529248T3 true DK3529248T3 (da) 2020-09-14

Family

ID=57680668

Family Applications (1)

Application Number Title Priority Date Filing Date
DK17790813.4T DK3529248T3 (da) 2016-10-18 2017-10-18 Farmaceutiske sammensætninger

Country Status (24)

Country Link
US (2) US10696666B2 (enExample)
EP (1) EP3529248B1 (enExample)
JP (1) JP7152393B2 (enExample)
KR (1) KR102578786B1 (enExample)
CN (1) CN110049983B (enExample)
AU (1) AU2017346453B2 (enExample)
CA (1) CA3039641A1 (enExample)
CY (1) CY1123666T1 (enExample)
DK (1) DK3529248T3 (enExample)
EA (1) EA201990643A1 (enExample)
ES (1) ES2828504T3 (enExample)
GB (1) GB201617630D0 (enExample)
HR (1) HRP20201444T1 (enExample)
HU (1) HUE052443T2 (enExample)
IL (1) IL266017B (enExample)
LT (1) LT3529248T (enExample)
MX (1) MX384438B (enExample)
PT (1) PT3529248T (enExample)
RS (1) RS61007B1 (enExample)
SG (1) SG11201903155XA (enExample)
SI (1) SI3529248T1 (enExample)
SM (1) SMT202000593T1 (enExample)
WO (1) WO2018073586A1 (enExample)
ZA (1) ZA201902334B (enExample)

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GB201806320D0 (en) * 2018-04-18 2018-05-30 Cellcentric Ltd Process
CN116178369A (zh) 2018-06-29 2023-05-30 福马疗法公司 抑制creb结合蛋白(cbp)
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CN112574189B (zh) * 2019-09-27 2024-05-31 海创药业股份有限公司 一种ep300/cbp抑制剂
CN112574191B (zh) * 2019-09-29 2024-01-23 南京圣和药业股份有限公司 异噁唑杂环类化合物及其应用
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US11795168B2 (en) 2020-09-23 2023-10-24 Forma Therapeutics, Inc. Inhibiting cyclic amp-responsive element-binding protein (CREB) binding protein (CBP)
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TW202227429A (zh) * 2020-11-06 2022-07-16 大陸商貝達藥業股份有限公司 P300抑制劑、包含其的藥物組合物、其應用及製備其的方法
US20240122941A1 (en) * 2020-12-25 2024-04-18 National Cancer Center Therapy based on synthetic lethality in swi/snf complex-dysfunction cancer
CN116670129A (zh) * 2020-12-31 2023-08-29 南京明德新药研发有限公司 苯并咪唑类化合物及其应用
CN114989158A (zh) * 2021-03-02 2022-09-02 复旦大学 组蛋白乙酰转移酶p300溴结构域抑制剂及其药用组合物及其应用
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Also Published As

Publication number Publication date
EP3529248A1 (en) 2019-08-28
CA3039641A1 (en) 2018-04-26
KR20190075095A (ko) 2019-06-28
LT3529248T (lt) 2020-10-26
US20200407349A1 (en) 2020-12-31
ZA201902334B (en) 2022-10-26
CY1123666T1 (el) 2022-03-24
PT3529248T (pt) 2020-09-03
HRP20201444T1 (hr) 2020-12-11
CN110049983A (zh) 2019-07-23
KR102578786B1 (ko) 2023-09-15
US10696666B2 (en) 2020-06-30
WO2018073586A1 (en) 2018-04-26
MX2019004113A (es) 2019-09-09
BR112019007834A2 (pt) 2019-07-16
EA201990643A1 (ru) 2019-11-29
CN110049983B (zh) 2022-06-14
AU2017346453B2 (en) 2022-02-17
AU2017346453A1 (en) 2019-05-02
IL266017B (en) 2021-08-31
US11377443B2 (en) 2022-07-05
US20190375740A1 (en) 2019-12-12
IL266017A (en) 2019-06-30
EP3529248B1 (en) 2020-08-19
SI3529248T1 (sl) 2020-11-30
ES2828504T3 (es) 2021-05-26
HUE052443T2 (hu) 2021-04-28
GB201617630D0 (en) 2016-11-30
JP7152393B2 (ja) 2022-10-12
NZ752354A (en) 2025-02-28
SMT202000593T1 (it) 2020-11-10
JP2019537571A (ja) 2019-12-26
MX384438B (es) 2025-03-14
SG11201903155XA (en) 2019-05-30
RS61007B1 (sr) 2020-11-30

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