DK228682A - Fremgangsmaade til fremstilling af et farmaceutisk middel med langvarig frigivelse - Google Patents

Fremgangsmaade til fremstilling af et farmaceutisk middel med langvarig frigivelse Download PDF

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Publication number
DK228682A
DK228682A DK228682A DK228682A DK228682A DK 228682 A DK228682 A DK 228682A DK 228682 A DK228682 A DK 228682A DK 228682 A DK228682 A DK 228682A DK 228682 A DK228682 A DK 228682A
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DK
Denmark
Prior art keywords
procedure
manufacturing
long
sustained release
term release
Prior art date
Application number
DK228682A
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English (en)
Other versions
DK154263B (da
DK154263C (da
Inventor
A S Mughal
D S Holmes
Original Assignee
Wyeth John & Brother Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth John & Brother Ltd filed Critical Wyeth John & Brother Ltd
Publication of DK228682A publication Critical patent/DK228682A/da
Publication of DK154263B publication Critical patent/DK154263B/da
Application granted granted Critical
Publication of DK154263C publication Critical patent/DK154263C/da

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

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  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
DK228682A 1981-05-21 1982-05-19 Fremgangsmaade til fremstilling af et farmaceutisk indoraminpraeparat med langvarig frigivelse og indeholdende et vandkanaldannelsesmiddel DK154263C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8115678 1981-05-21
GB8115678 1981-05-21

Publications (3)

Publication Number Publication Date
DK228682A true DK228682A (da) 1982-11-22
DK154263B DK154263B (da) 1988-10-31
DK154263C DK154263C (da) 1989-03-28

Family

ID=10521980

Family Applications (1)

Application Number Title Priority Date Filing Date
DK228682A DK154263C (da) 1981-05-21 1982-05-19 Fremgangsmaade til fremstilling af et farmaceutisk indoraminpraeparat med langvarig frigivelse og indeholdende et vandkanaldannelsesmiddel

Country Status (16)

Country Link
US (1) US4524060A (da)
EP (1) EP0067539B1 (da)
JP (1) JPS57197212A (da)
AT (1) ATE15599T1 (da)
AU (1) AU556241B2 (da)
CA (1) CA1165246A (da)
DE (1) DE3266332D1 (da)
DK (1) DK154263C (da)
ES (1) ES512393A0 (da)
GR (1) GR76391B (da)
IE (1) IE53118B1 (da)
IL (1) IL65706A (da)
NZ (1) NZ200519A (da)
PH (1) PH19109A (da)
PT (1) PT74946B (da)
ZA (1) ZA822995B (da)

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US20040013613A1 (en) * 2001-05-18 2004-01-22 Jain Rajeev A Rapidly disintegrating solid oral dosage form
US8236352B2 (en) * 1998-10-01 2012-08-07 Alkermes Pharma Ireland Limited Glipizide compositions
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US20080213378A1 (en) * 1998-10-01 2008-09-04 Elan Pharma International, Ltd. Nanoparticulate statin formulations and novel statin combinations
US8293277B2 (en) * 1998-10-01 2012-10-23 Alkermes Pharma Ireland Limited Controlled-release nanoparticulate compositions
US20040141925A1 (en) * 1998-11-12 2004-07-22 Elan Pharma International Ltd. Novel triamcinolone compositions
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US20040115134A1 (en) * 1999-06-22 2004-06-17 Elan Pharma International Ltd. Novel nifedipine compositions
US20040258750A1 (en) * 1999-06-28 2004-12-23 Gerard Alaux Timed dual release dosage forms comprising a short acting hypnotic or a salt thereof
EP1064938A1 (en) * 1999-06-28 2001-01-03 Sanofi-Synthelabo Pharmaceutical dosage forms for controlled release producing at least a timed pulse
CN1422156A (zh) * 2000-02-14 2003-06-04 法马西亚公司 N-取代的-1,5-二脱氧-1,5-亚氨基-d-葡萄糖醇化合物在治疗肝炎病毒感染中的用途
US20040156872A1 (en) * 2000-05-18 2004-08-12 Elan Pharma International Ltd. Novel nimesulide compositions
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JP4598399B2 (ja) * 2002-02-04 2010-12-15 エラン ファーマ インターナショナル,リミティド 表面安定剤としてリゾチームを有するナノ粒子組成物
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US7632521B2 (en) * 2003-07-15 2009-12-15 Eurand, Inc. Controlled release potassium chloride tablets
US20060020044A1 (en) * 2004-07-26 2006-01-26 Roger Berlin Methods and compositions for treating or preventing macular-degeneration related disorders
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Also Published As

Publication number Publication date
PT74946A (en) 1982-06-01
ZA822995B (en) 1983-12-28
EP0067539A3 (en) 1983-04-27
ES8302456A1 (es) 1983-02-01
GR76391B (da) 1984-08-10
CA1165246A (en) 1984-04-10
EP0067539B1 (en) 1985-09-18
ATE15599T1 (de) 1985-10-15
IE821213L (en) 1982-11-21
EP0067539A2 (en) 1982-12-22
AU8355482A (en) 1982-11-25
DK154263B (da) 1988-10-31
DK154263C (da) 1989-03-28
PH19109A (en) 1986-01-06
ES512393A0 (es) 1983-02-01
IE53118B1 (en) 1988-07-06
US4524060A (en) 1985-06-18
NZ200519A (en) 1985-08-30
PT74946B (en) 1983-12-23
JPS57197212A (en) 1982-12-03
IL65706A (en) 1985-07-31
AU556241B2 (en) 1986-10-30
DE3266332D1 (en) 1985-10-24
JPH0237327B2 (da) 1990-08-23

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