DK175126B1 - Peptid-aminoalkylamider, deres fremstilling og anvendelse til fremstilling af peptid-hydrazider - Google Patents

Peptid-aminoalkylamider, deres fremstilling og anvendelse til fremstilling af peptid-hydrazider Download PDF

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Publication number
DK175126B1
DK175126B1 DK198705482A DK548287A DK175126B1 DK 175126 B1 DK175126 B1 DK 175126B1 DK 198705482 A DK198705482 A DK 198705482A DK 548287 A DK548287 A DK 548287A DK 175126 B1 DK175126 B1 DK 175126B1
Authority
DK
Denmark
Prior art keywords
formula
compound
hydrogen
peptide
labile
Prior art date
Application number
DK198705482A
Other languages
Danish (da)
English (en)
Other versions
DK548287A (da
DK548287D0 (da
Inventor
Gerhard Breipohl
Jochen Knolle
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of DK548287D0 publication Critical patent/DK548287D0/da
Publication of DK548287A publication Critical patent/DK548287A/da
Application granted granted Critical
Publication of DK175126B1 publication Critical patent/DK175126B1/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/58—Atrial natriuretic factor complex; Atriopeptin; Atrial natriuretic peptide [ANP]; Cardionatrin; Cardiodilatin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
    • C07K1/042—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers characterised by the nature of the carrier
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Toxicology (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Analytical Chemistry (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pyrane Compounds (AREA)
DK198705482A 1986-10-21 1987-10-20 Peptid-aminoalkylamider, deres fremstilling og anvendelse til fremstilling af peptid-hydrazider DK175126B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3635670 1986-10-21
DE19863635670 DE3635670A1 (de) 1986-10-21 1986-10-21 Synthese von peptid-aminoalkylamiden und peptidhydraziden mittels festphasenmethode

Publications (3)

Publication Number Publication Date
DK548287D0 DK548287D0 (da) 1987-10-20
DK548287A DK548287A (da) 1988-04-22
DK175126B1 true DK175126B1 (da) 2004-06-07

Family

ID=6312082

Family Applications (1)

Application Number Title Priority Date Filing Date
DK198705482A DK175126B1 (da) 1986-10-21 1987-10-20 Peptid-aminoalkylamider, deres fremstilling og anvendelse til fremstilling af peptid-hydrazider

Country Status (18)

Country Link
EP (1) EP0264802B1 (fr)
JP (1) JP2540564B2 (fr)
KR (1) KR960013073B1 (fr)
AT (1) ATE83244T1 (fr)
AU (1) AU595390B2 (fr)
CA (1) CA1340421C (fr)
DE (2) DE3635670A1 (fr)
DK (1) DK175126B1 (fr)
ES (1) ES2052535T3 (fr)
FI (1) FI88031C (fr)
GR (1) GR3007231T3 (fr)
HU (1) HU197719B (fr)
IE (1) IE60864B1 (fr)
IL (1) IL84195A (fr)
NO (1) NO172895C (fr)
NZ (1) NZ222204A (fr)
PT (1) PT85952B (fr)
ZA (1) ZA877862B (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3926822A1 (de) 1989-08-14 1991-02-21 Hoechst Ag Peptide mit bradykinin-antagonistischer wirkung
EP0376218B1 (fr) * 1988-12-27 1999-02-24 Perseptive Biosystems, Inc. Rattachement sans racémisation des acides aminés aux phases solides
DE4408533A1 (de) 1994-03-14 1995-09-28 Hoechst Ag PNA-Synthese unter Verwendung einer basenlabilen Amino-Schutzgruppe
SI0946478T1 (sl) * 1996-12-19 2007-06-30 Aventis Pharma Inc Postopek za sintezo v trdni fazi aldehidov, ketonov in spojin hidroksamske kisline
GB9727123D0 (en) * 1997-12-22 1998-02-25 Int Centre Genetic Eng & Bio Synthesis of diamines
US6852789B2 (en) * 2002-02-15 2005-02-08 Degussa - Ag Glycols starting materials containing dispersed superfine ceramic powder coagulates capable of forming polyester molded bodies having high mechanical strength and transparency

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4108846A (en) * 1977-02-01 1978-08-22 Hoffmann-La Roche Inc. Solid phase synthesis with base N alpha-protecting group cleavage

Also Published As

Publication number Publication date
NO874374D0 (no) 1987-10-20
NO172895B (no) 1993-06-14
IE60864B1 (en) 1994-08-24
NO172895C (no) 1993-09-22
HUT46706A (en) 1988-11-28
EP0264802B1 (fr) 1992-12-09
EP0264802A3 (en) 1989-07-26
JP2540564B2 (ja) 1996-10-02
FI874586A (fi) 1988-04-22
EP0264802A2 (fr) 1988-04-27
IL84195A0 (en) 1988-03-31
FI88031B (fi) 1992-12-15
ATE83244T1 (de) 1992-12-15
FI88031C (fi) 1993-03-25
PT85952A (de) 1987-11-01
DE3635670A1 (de) 1988-04-28
KR880005147A (ko) 1988-06-28
DK548287A (da) 1988-04-22
GR3007231T3 (fr) 1993-07-30
FI874586A0 (fi) 1987-10-19
ZA877862B (en) 1988-04-22
IE872821L (en) 1988-04-21
ES2052535T3 (es) 1994-07-16
AU7993587A (en) 1988-04-28
HU197719B (en) 1989-05-29
JPS63104951A (ja) 1988-05-10
KR960013073B1 (ko) 1996-09-30
DK548287D0 (da) 1987-10-20
NZ222204A (en) 1989-10-27
NO874374L (no) 1988-04-22
AU595390B2 (en) 1990-03-29
PT85952B (pt) 1990-07-31
CA1340421C (fr) 1999-03-09
IL84195A (en) 1992-08-18
DE3783009D1 (fr) 1993-01-21

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