DK170100B1 - 2'-Substituerede 4-deoxytiazolo(5,4-c)rifamycin SV-derivater, fremgangsmåde til fremstilling heraf, en sådan forbindelse til anvendelse som lægemiddel, anvendelse af forbindelsen til fremstilling af et antibakterielt medikament samt farmaceutisk præparat indeholdende forbindelsen - Google Patents
2'-Substituerede 4-deoxytiazolo(5,4-c)rifamycin SV-derivater, fremgangsmåde til fremstilling heraf, en sådan forbindelse til anvendelse som lægemiddel, anvendelse af forbindelsen til fremstilling af et antibakterielt medikament samt farmaceutisk præparat indeholdende forbindelsen Download PDFInfo
- Publication number
- DK170100B1 DK170100B1 DK630686A DK630686A DK170100B1 DK 170100 B1 DK170100 B1 DK 170100B1 DK 630686 A DK630686 A DK 630686A DK 630686 A DK630686 A DK 630686A DK 170100 B1 DK170100 B1 DK 170100B1
- Authority
- DK
- Denmark
- Prior art keywords
- compound
- rifamycin
- alkyl
- group
- optionally substituted
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/10—Spiro-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
- C07D513/18—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB858531887A GB8531887D0 (en) | 1985-12-30 | 1985-12-30 | Rifamycin sv derivatives |
GB8531887 | 1985-12-30 |
Publications (3)
Publication Number | Publication Date |
---|---|
DK630686D0 DK630686D0 (da) | 1986-12-29 |
DK630686A DK630686A (da) | 1987-07-01 |
DK170100B1 true DK170100B1 (da) | 1995-05-22 |
Family
ID=10590333
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK630686A DK170100B1 (da) | 1985-12-30 | 1986-12-29 | 2'-Substituerede 4-deoxytiazolo(5,4-c)rifamycin SV-derivater, fremgangsmåde til fremstilling heraf, en sådan forbindelse til anvendelse som lægemiddel, anvendelse af forbindelsen til fremstilling af et antibakterielt medikament samt farmaceutisk præparat indeholdende forbindelsen |
Country Status (17)
Country | Link |
---|---|
US (1) | US4880789A (ja) |
EP (1) | EP0228606B1 (ja) |
JP (1) | JPH07108909B2 (ja) |
KR (1) | KR940009795B1 (ja) |
AT (1) | ATE60772T1 (ja) |
CA (1) | CA1271472A (ja) |
DE (1) | DE3677485D1 (ja) |
DK (1) | DK170100B1 (ja) |
ES (1) | ES2031815T3 (ja) |
GB (1) | GB8531887D0 (ja) |
GR (1) | GR3001543T3 (ja) |
HK (1) | HK97391A (ja) |
HU (1) | HU196812B (ja) |
IE (1) | IE59505B1 (ja) |
IL (1) | IL80447A (ja) |
SG (1) | SG67091G (ja) |
ZA (1) | ZA869453B (ja) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK0497125T3 (da) * | 1991-01-28 | 1999-08-16 | Lepetit Spa | Fremgangsmåde til fremstilling af 2'-(diethylamino)rifamycin P (P/DEA) |
US6375658B1 (en) | 2000-04-28 | 2002-04-23 | Smith & Nephew, Inc. | Cartilage grafting |
US7265107B2 (en) | 2004-03-10 | 2007-09-04 | Cumbre Pharmaceuticals Inc. | Rifamycin C-11 oxime cyclo derivatives effective against drug-resistant microbes |
US7256187B2 (en) | 2004-03-10 | 2007-08-14 | Cumbre Pharmaceuticals Inc. | Rifamycin C-11 oxime derivatives effective against drug-resistant microbes |
US20100125146A1 (en) * | 2008-11-19 | 2010-05-20 | Johnson Matthey Public Limited Company | Method for making pharmaceutical compounds |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1470426A (en) * | 1974-08-30 | 1977-04-14 | Lepetit Spa | Rifamycins |
GB1523198A (en) * | 1976-05-28 | 1978-08-31 | Lepetit Spa | Thiazolo-rifamycin derivatives |
GB1523199A (en) * | 1976-05-28 | 1978-08-31 | Lepetit Spa | Rifamycin sv derivatives |
CH629212A5 (it) * | 1976-10-18 | 1982-04-15 | Erba Farmitalia | Procedimento per la preparazione di composti di rifamicina. |
GB1594134A (en) * | 1977-11-25 | 1981-07-30 | Holco Investment Inc | Rifamycins |
IT1111173B (it) * | 1978-04-27 | 1986-01-13 | Lepetit Spa | Derivati rifamicinici |
FI812936L (fi) * | 1980-09-25 | 1982-03-26 | Ciba Geigy Ag | Nya 2-aminoimidazoler foerfaranden foer deras framstaellning dessa foereningar innehaollande farmaceutiska preparat och deras anvaendning |
-
1985
- 1985-12-30 GB GB858531887A patent/GB8531887D0/en active Pending
-
1986
- 1986-10-29 IL IL80447A patent/IL80447A/xx not_active IP Right Cessation
- 1986-12-06 EP EP19860117005 patent/EP0228606B1/en not_active Expired - Lifetime
- 1986-12-06 DE DE8686117005T patent/DE3677485D1/de not_active Expired - Fee Related
- 1986-12-06 ES ES198686117005T patent/ES2031815T3/es not_active Expired - Lifetime
- 1986-12-06 AT AT86117005T patent/ATE60772T1/de not_active IP Right Cessation
- 1986-12-16 IE IE327786A patent/IE59505B1/en not_active IP Right Cessation
- 1986-12-17 ZA ZA869453A patent/ZA869453B/xx unknown
- 1986-12-18 KR KR1019860010871A patent/KR940009795B1/ko not_active IP Right Cessation
- 1986-12-25 JP JP61308066A patent/JPH07108909B2/ja not_active Expired - Lifetime
- 1986-12-29 CA CA000526359A patent/CA1271472A/en not_active Expired - Fee Related
- 1986-12-29 HU HU865501A patent/HU196812B/hu not_active IP Right Cessation
- 1986-12-29 DK DK630686A patent/DK170100B1/da not_active IP Right Cessation
-
1988
- 1988-08-24 US US07/238,985 patent/US4880789A/en not_active Expired - Fee Related
-
1991
- 1991-03-04 GR GR91400257T patent/GR3001543T3/el unknown
- 1991-08-16 SG SG670/91A patent/SG67091G/en unknown
- 1991-12-05 HK HK973/91A patent/HK97391A/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
JPH07108909B2 (ja) | 1995-11-22 |
HUT45072A (en) | 1988-05-30 |
IE59505B1 (en) | 1994-03-09 |
IL80447A0 (en) | 1987-01-30 |
IL80447A (en) | 1990-09-17 |
ZA869453B (en) | 1987-09-30 |
DK630686D0 (da) | 1986-12-29 |
US4880789A (en) | 1989-11-14 |
ATE60772T1 (de) | 1991-02-15 |
ES2031815T3 (es) | 1993-01-01 |
GR3001543T3 (en) | 1992-11-23 |
GB8531887D0 (en) | 1986-02-05 |
CA1271472A (en) | 1990-07-10 |
JPS62158292A (ja) | 1987-07-14 |
IE863277L (en) | 1987-06-30 |
KR940009795B1 (ko) | 1994-10-17 |
EP0228606A3 (en) | 1989-01-11 |
HU196812B (en) | 1989-01-30 |
EP0228606A2 (en) | 1987-07-15 |
DK630686A (da) | 1987-07-01 |
DE3677485D1 (de) | 1991-03-14 |
SG67091G (en) | 1991-09-13 |
EP0228606B1 (en) | 1991-02-06 |
KR870006057A (ko) | 1987-07-09 |
HK97391A (en) | 1991-12-13 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B1 | Patent granted (law 1993) | ||
PBP | Patent lapsed |