DK169761B1 - N-(4-piperidinyl)substituerede bicyclisk kondenserede 2-imidazolaminderivater, fremgangsmåde til fremstilling deraf og præparater indeholdende disse derivater - Google Patents

N-(4-piperidinyl)substituerede bicyclisk kondenserede 2-imidazolaminderivater, fremgangsmåde til fremstilling deraf og præparater indeholdende disse derivater Download PDF

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Publication number
DK169761B1
DK169761B1 DK333288A DK333288A DK169761B1 DK 169761 B1 DK169761 B1 DK 169761B1 DK 333288 A DK333288 A DK 333288A DK 333288 A DK333288 A DK 333288A DK 169761 B1 DK169761 B1 DK 169761B1
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Prior art keywords
formula
alk
methyl
compound
phenyl
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DK333288A
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Danish (da)
English (en)
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DK333288D0 (da
DK333288A (da
Inventor
Frans Eduard Janssens
Joseph Leo Ghislanus Torremans
Gaston Stanislas Marcell Diels
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Janssen Pharmaceutica Nv
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Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of DK333288D0 publication Critical patent/DK333288D0/da
Publication of DK333288A publication Critical patent/DK333288A/da
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)
  • Lubricants (AREA)
DK333288A 1987-06-19 1988-06-17 N-(4-piperidinyl)substituerede bicyclisk kondenserede 2-imidazolaminderivater, fremgangsmåde til fremstilling deraf og præparater indeholdende disse derivater DK169761B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US6389987A 1987-06-19 1987-06-19
US6389987 1987-06-19

Publications (3)

Publication Number Publication Date
DK333288D0 DK333288D0 (da) 1988-06-17
DK333288A DK333288A (da) 1988-12-20
DK169761B1 true DK169761B1 (da) 1995-02-20

Family

ID=22052235

Family Applications (1)

Application Number Title Priority Date Filing Date
DK333288A DK169761B1 (da) 1987-06-19 1988-06-17 N-(4-piperidinyl)substituerede bicyclisk kondenserede 2-imidazolaminderivater, fremgangsmåde til fremstilling deraf og præparater indeholdende disse derivater

Country Status (22)

Country Link
US (1) US4897401A (fr)
EP (1) EP0295742B1 (fr)
JP (1) JP2609464B2 (fr)
KR (1) KR970001158B1 (fr)
CN (1) CN1029964C (fr)
AT (1) ATE79878T1 (fr)
AU (1) AU600144B2 (fr)
CA (1) CA1324133C (fr)
DE (1) DE3874013T2 (fr)
DK (1) DK169761B1 (fr)
ES (1) ES2045083T3 (fr)
FI (1) FI90233C (fr)
GR (1) GR3006205T3 (fr)
HU (1) HU201755B (fr)
IE (1) IE61728B1 (fr)
IL (1) IL86788A (fr)
NO (1) NO167803C (fr)
NZ (1) NZ224928A (fr)
PH (1) PH25532A (fr)
PT (1) PT87742B (fr)
SU (1) SU1644717A3 (fr)
ZA (1) ZA884346B (fr)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8716313D0 (en) * 1987-07-10 1987-08-19 Janssen Pharmaceutica Nv 2-(heterocyclylalkyl)imidazopyridines
GB8900380D0 (en) * 1989-01-09 1989-03-08 Janssen Pharmaceutica Nv 2-aminopyrimidinone derivatives
PH30434A (en) * 1989-04-07 1997-05-09 Janssen Pharmaceutica Nv Hydroxyalkylfuranyl derivatives
US5272150A (en) * 1989-04-07 1993-12-21 Janssen Pharmaceutica N.V. Hydroxyalkylfuranyl derivatives
KR100190299B1 (ko) * 1990-07-19 1999-06-01 디르크 반테 신규한 옥사졸릴 유도체
NZ238863A (en) * 1990-07-19 1993-03-26 Janssen Pharmaceutica Nv Substituted thiazolyl and pyridinyl derivatives
US5217980A (en) * 1990-07-19 1993-06-08 Janssen Pharmaceutica N.V. Oxazolyl and piperidinyl substituted benimidazolyl compounds
FR2725986B1 (fr) * 1994-10-21 1996-11-29 Adir Nouveaux derives de piperidine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
AU778218B2 (en) 1999-06-28 2004-11-25 Janssen Pharmaceutica N.V. Respiratory syncytial virus replication inhibitors
EE04592B1 (et) * 1999-06-28 2006-02-15 Janssen Pharmaceutica N.V. Respiratoorse süntsütiaalviiruse replikatsiooni inhibiitorid, nende valmistamismeetod, kasutamine ja vaheühendid, farmatseutiline kompositsioon ja selle valmistamismeetod ning produkt
PL198021B1 (pl) * 1999-06-28 2008-05-30 Janssen Pharmaceutica Nv Pochodna benzoimidazolu lub imidazopirydyny, jej zastosowanie i sposób otrzymywania oraz kompozycja farmaceutyczna

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4219559A (en) * 1979-01-10 1980-08-26 Janssen Pharmaceutica N.V. N-Heterocyclyl-4-piperidinamines
US4556660A (en) * 1982-07-12 1985-12-03 Janssen Pharmaceutica N.V. N-(Bicyclic heterocyclyl)-4-piperidinamines
US4634704A (en) * 1983-10-06 1987-01-06 Janssen Pharmaceutica, N.V. Anti-allergic five membered heterocyclic ring containing N-(bicyclic heterocycyl)-4-piperidinamines
US4695569A (en) * 1983-11-30 1987-09-22 Janssen Pharmaceutica N.V. Bicyclic heterocyclyl containing N-(bicyclic heterocyclyl)-4-piperidinamines
US4588722A (en) * 1984-01-09 1986-05-13 Janssen Pharmaceutica N.V. N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives
ATE79620T1 (de) * 1986-02-03 1992-09-15 Janssen Pharmaceutica Nv N-heterozyklische-4-piperidinamine enthaltende anti-histaminische zusammensetzungen.
CA1317939C (fr) * 1987-07-01 1993-05-18 Janssen Pharmaceutica Naamloze Vennootschap Hexahydro-1h-azepines et pyrrolidines a substitution par des ((heterocyclyle bicyclique) methyle et -hetero

Also Published As

Publication number Publication date
IE61728B1 (en) 1994-11-30
IL86788A (en) 1992-08-18
DE3874013D1 (de) 1992-10-01
CA1324133C (fr) 1993-11-09
JPS6425776A (en) 1989-01-27
DK333288D0 (da) 1988-06-17
PT87742A (pt) 1988-07-01
EP0295742A1 (fr) 1988-12-21
NO167803C (no) 1991-12-11
FI882909A0 (fi) 1988-06-17
DK333288A (da) 1988-12-20
NO167803B (no) 1991-09-02
HU201755B (en) 1990-12-28
AU1810988A (en) 1988-12-22
FI90233C (fi) 1994-01-10
KR890000484A (ko) 1989-03-15
SU1644717A3 (ru) 1991-04-23
FI882909A (fi) 1988-12-20
ZA884346B (en) 1990-02-28
NO882641L (no) 1988-12-20
IE881849L (en) 1988-12-19
PT87742B (pt) 1992-10-30
DE3874013T2 (de) 1993-01-07
NO882641D0 (no) 1988-06-15
CN88103784A (zh) 1988-12-28
KR970001158B1 (ko) 1997-01-29
PH25532A (en) 1991-07-24
AU600144B2 (en) 1990-08-02
ATE79878T1 (de) 1992-09-15
JP2609464B2 (ja) 1997-05-14
EP0295742B1 (fr) 1992-08-26
CN1029964C (zh) 1995-10-11
IL86788A0 (en) 1988-11-30
ES2045083T3 (es) 1994-01-16
NZ224928A (en) 1990-04-26
US4897401A (en) 1990-01-30
FI90233B (fi) 1993-09-30
HUT48628A (en) 1989-06-28
GR3006205T3 (fr) 1993-06-21

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Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
PBP Patent lapsed