DK169760B1 - 4H-1-Benzopyran-4-on-derivater, fremgangsmåde til deres fremstilling og deres anvendelse i lægemidler - Google Patents

4H-1-Benzopyran-4-on-derivater, fremgangsmåde til deres fremstilling og deres anvendelse i lægemidler Download PDF

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Publication number
DK169760B1
DK169760B1 DK185287A DK185287A DK169760B1 DK 169760 B1 DK169760 B1 DK 169760B1 DK 185287 A DK185287 A DK 185287A DK 185287 A DK185287 A DK 185287A DK 169760 B1 DK169760 B1 DK 169760B1
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DK
Denmark
Prior art keywords
hydroxy
methyl
cis
alkyl
formula
Prior art date
Application number
DK185287A
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Danish (da)
English (en)
Other versions
DK185287A (da
DK185287D0 (da
Inventor
Samba Laxminarayan Kattige
Ramchandra Ganapati Naik
Aftab Dawoodbhai Lakdawalla
Alihussein Nomanbha Dohadwalla
Richard Helmut Rupp
Noel John De Souza
Original Assignee
Hoechst Ag
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Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of DK185287D0 publication Critical patent/DK185287D0/da
Publication of DK185287A publication Critical patent/DK185287A/da
Application granted granted Critical
Publication of DK169760B1 publication Critical patent/DK169760B1/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/42—Oxygen atoms attached in position 3 or 5
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pulmonology (AREA)
  • Transplantation (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK185287A 1986-04-11 1987-04-10 4H-1-Benzopyran-4-on-derivater, fremgangsmåde til deres fremstilling og deres anvendelse i lægemidler DK169760B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3612337 1986-04-11
DE19863612337 DE3612337A1 (de) 1986-04-11 1986-04-11 4h-1-benzopyran-4-on-derivate, ein verfahren zu ihrer herstellung und ihre verwendung als arzneimittel

Publications (3)

Publication Number Publication Date
DK185287D0 DK185287D0 (da) 1987-04-10
DK185287A DK185287A (da) 1987-10-12
DK169760B1 true DK169760B1 (da) 1995-02-20

Family

ID=6298535

Family Applications (1)

Application Number Title Priority Date Filing Date
DK185287A DK169760B1 (da) 1986-04-11 1987-04-10 4H-1-Benzopyran-4-on-derivater, fremgangsmåde til deres fremstilling og deres anvendelse i lægemidler

Country Status (16)

Country Link
US (1) US4900727A (US20040106767A1-20040603-C00005.png)
EP (1) EP0241003B1 (US20040106767A1-20040603-C00005.png)
JP (1) JPH0686446B2 (US20040106767A1-20040603-C00005.png)
KR (1) KR950009861B1 (US20040106767A1-20040603-C00005.png)
AT (2) ATE95519T1 (US20040106767A1-20040603-C00005.png)
AU (1) AU602891B2 (US20040106767A1-20040603-C00005.png)
CA (1) CA1332238C (US20040106767A1-20040603-C00005.png)
DE (2) DE3612337A1 (US20040106767A1-20040603-C00005.png)
DK (1) DK169760B1 (US20040106767A1-20040603-C00005.png)
ES (1) ES2060582T3 (US20040106767A1-20040603-C00005.png)
HK (1) HK1006021A1 (US20040106767A1-20040603-C00005.png)
IE (1) IE62244B1 (US20040106767A1-20040603-C00005.png)
IL (1) IL82149A (US20040106767A1-20040603-C00005.png)
IN (1) IN164232B (US20040106767A1-20040603-C00005.png)
PT (1) PT84654B (US20040106767A1-20040603-C00005.png)
ZA (1) ZA872555B (US20040106767A1-20040603-C00005.png)

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US7335650B2 (en) 2000-01-14 2008-02-26 Sterix Limited Composition
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US6821990B2 (en) * 2000-01-18 2004-11-23 Aventis Pharma Deutschland Gmbh Ethanol solvate of (-)-cis-2-(2-chlorophenyl)-5, 7-dihydroxy-8 [4R-(3S-hydroxy-1-M ethyl) piperidinyl]-4H-1-benzopyran-4-one
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KR100423899B1 (ko) 2000-05-10 2004-03-24 주식회사 엘지생명과학 세포 증식 억제제로 유용한 1,1-디옥소이소티아졸리딘을갖는 인다졸
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Also Published As

Publication number Publication date
PT84654A (de) 1987-05-01
KR950009861B1 (en) 1995-08-29
ATA260587A (de) 1989-07-15
EP0241003B1 (de) 1993-10-06
KR870010045A (ko) 1987-11-30
EP0241003A3 (en) 1988-10-12
AT389875B (de) 1990-02-12
JPH0686446B2 (ja) 1994-11-02
US4900727A (en) 1990-02-13
IN164232B (US20040106767A1-20040603-C00005.png) 1989-02-04
HK1006021A1 (en) 1999-02-05
AU7139787A (en) 1987-10-15
AU602891B2 (en) 1990-11-01
DE3787661D1 (de) 1993-11-11
CA1332238C (en) 1994-10-04
ES2060582T3 (es) 1994-12-01
IL82149A0 (en) 1987-10-30
IL82149A (en) 1994-01-25
ZA872555B (en) 1987-11-25
IE62244B1 (en) 1995-01-11
PT84654B (pt) 1989-12-29
JPS62242680A (ja) 1987-10-23
DE3612337A1 (de) 1987-10-15
DK185287A (da) 1987-10-12
EP0241003A2 (de) 1987-10-14
DK185287D0 (da) 1987-04-10
ATE95519T1 (de) 1993-10-15
IE870941L (en) 1987-10-11

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Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
PUP Patent expired