DK1644395T3 - Fremgangsmåde til fremstilling af 4azido-nukleosidderivater - Google Patents

Fremgangsmåde til fremstilling af 4azido-nukleosidderivater

Info

Publication number
DK1644395T3
DK1644395T3 DK04739843T DK04739843T DK1644395T3 DK 1644395 T3 DK1644395 T3 DK 1644395T3 DK 04739843 T DK04739843 T DK 04739843T DK 04739843 T DK04739843 T DK 04739843T DK 1644395 T3 DK1644395 T3 DK 1644395T3
Authority
DK
Denmark
Prior art keywords
alkyl
preparation
4azido
halogen
hydrogen
Prior art date
Application number
DK04739843T
Other languages
Danish (da)
English (en)
Inventor
Terrence Joseph Connolly
Kieran Durkin
Keshab Sarma
Jiang Zhu
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of DK1644395T3 publication Critical patent/DK1644395T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals
    • C07H19/067—Pyrimidine radicals with ribosyl as the saccharide radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK04739843T 2003-06-19 2004-06-11 Fremgangsmåde til fremstilling af 4azido-nukleosidderivater DK1644395T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US47979603P 2003-06-19 2003-06-19
PCT/EP2004/006357 WO2005000864A1 (fr) 2003-06-19 2004-06-11 Methodes de preparation de derives de 4'azido nucleoside

Publications (1)

Publication Number Publication Date
DK1644395T3 true DK1644395T3 (da) 2007-04-02

Family

ID=33551901

Family Applications (1)

Application Number Title Priority Date Filing Date
DK04739843T DK1644395T3 (da) 2003-06-19 2004-06-11 Fremgangsmåde til fremstilling af 4azido-nukleosidderivater

Country Status (14)

Country Link
US (1) US20050038240A1 (fr)
EP (1) EP1644395B1 (fr)
JP (1) JP2006527719A (fr)
KR (1) KR20060026426A (fr)
CN (1) CN1809582A (fr)
AT (1) ATE346078T1 (fr)
CA (1) CA2528294A1 (fr)
DE (1) DE602004003389T2 (fr)
DK (1) DK1644395T3 (fr)
ES (1) ES2276311T3 (fr)
IL (1) IL172275A0 (fr)
MX (1) MXPA05013452A (fr)
TW (1) TW200519122A (fr)
WO (1) WO2005000864A1 (fr)

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Also Published As

Publication number Publication date
CA2528294A1 (fr) 2005-01-06
MXPA05013452A (es) 2006-03-09
CN1809582A (zh) 2006-07-26
DE602004003389D1 (de) 2007-01-04
TW200519122A (en) 2005-06-16
KR20060026426A (ko) 2006-03-23
JP2006527719A (ja) 2006-12-07
ATE346078T1 (de) 2006-12-15
EP1644395B1 (fr) 2006-11-22
IL172275A0 (en) 2006-04-10
WO2005000864A1 (fr) 2005-01-06
ES2276311T3 (es) 2007-06-16
US20050038240A1 (en) 2005-02-17
DE602004003389T2 (de) 2007-09-13
EP1644395A1 (fr) 2006-04-12

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