DK158346C - Analogifremgangsmaade til fremstilling af 4-amino-5-alkylsulfonyl-o-anisamid-derivater samt 2-methoxy-4-amino-5-alkylsulfonylbenzoesyrer til anvendelse som mellemprodukter ved fremgangsmaaden - Google Patents

Analogifremgangsmaade til fremstilling af 4-amino-5-alkylsulfonyl-o-anisamid-derivater samt 2-methoxy-4-amino-5-alkylsulfonylbenzoesyrer til anvendelse som mellemprodukter ved fremgangsmaaden

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Publication number
DK158346C
DK158346C DK020979A DK20979A DK158346C DK 158346 C DK158346 C DK 158346C DK 020979 A DK020979 A DK 020979A DK 20979 A DK20979 A DK 20979A DK 158346 C DK158346 C DK 158346C
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DK
Denmark
Prior art keywords
fruit
sodane
amino
intermediatric
acroduced
Prior art date
Application number
DK020979A
Other languages
Danish (da)
English (en)
Other versions
DK20979A (da
DK158346B (da
Inventor
Michel Thominet
Jacques Acher
Jean-Claude Monier
Original Assignee
Ile De France
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ile De France filed Critical Ile De France
Publication of DK20979A publication Critical patent/DK20979A/da
Publication of DK158346B publication Critical patent/DK158346B/da
Application granted granted Critical
Publication of DK158346C publication Critical patent/DK158346C/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • C07D207/09—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyrrole Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
DK020979A 1978-01-20 1979-01-18 Analogifremgangsmaade til fremstilling af 4-amino-5-alkylsulfonyl-o-anisamid-derivater samt 2-methoxy-4-amino-5-alkylsulfonylbenzoesyrer til anvendelse som mellemprodukter ved fremgangsmaaden DK158346C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR7801632 1978-01-20
FR7801632A FR2415099A1 (fr) 1978-01-20 1978-01-20 Nouveaux derives de 4-amino-5-alkylsulfonyl ortho-anisamides, leurs procedes de preparation et leur application comme psychotropes

Publications (3)

Publication Number Publication Date
DK20979A DK20979A (da) 1979-07-21
DK158346B DK158346B (da) 1990-05-07
DK158346C true DK158346C (da) 1990-10-08

Family

ID=9203689

Family Applications (1)

Application Number Title Priority Date Filing Date
DK020979A DK158346C (da) 1978-01-20 1979-01-18 Analogifremgangsmaade til fremstilling af 4-amino-5-alkylsulfonyl-o-anisamid-derivater samt 2-methoxy-4-amino-5-alkylsulfonylbenzoesyrer til anvendelse som mellemprodukter ved fremgangsmaaden

Country Status (42)

Country Link
US (2) US4294828A (Sortimente)
JP (1) JPS6049192B2 (Sortimente)
AR (2) AR221354A1 (Sortimente)
AT (1) AT377977B (Sortimente)
AU (1) AU528561B2 (Sortimente)
BE (1) BE872585A (Sortimente)
BG (2) BG31497A3 (Sortimente)
CA (1) CA1101430A (Sortimente)
CH (1) CH637927A5 (Sortimente)
CS (1) CS226181B2 (Sortimente)
CY (1) CY1201A (Sortimente)
DD (1) DD141520A5 (Sortimente)
DE (1) DE2901181C2 (Sortimente)
DK (1) DK158346C (Sortimente)
EG (1) EG14045A (Sortimente)
ES (2) ES476755A1 (Sortimente)
FI (1) FI71126C (Sortimente)
FR (1) FR2415099A1 (Sortimente)
GB (2) GB2012765B (Sortimente)
GR (1) GR64431B (Sortimente)
HK (1) HK12184A (Sortimente)
HU (1) HU179793B (Sortimente)
IE (1) IE47798B1 (Sortimente)
IL (1) IL56411A (Sortimente)
IN (1) IN150226B (Sortimente)
IT (1) IT1164655B (Sortimente)
LU (1) LU80786A1 (Sortimente)
MC (1) MC1232A1 (Sortimente)
MX (2) MX7623E (Sortimente)
NL (1) NL191707C (Sortimente)
NO (1) NO151320C (Sortimente)
NZ (1) NZ189378A (Sortimente)
OA (1) OA06156A (Sortimente)
PH (2) PH15725A (Sortimente)
PL (2) PL118151B1 (Sortimente)
PT (1) PT69068A (Sortimente)
RO (2) RO80311A (Sortimente)
SE (2) SE448874B (Sortimente)
SU (1) SU820659A3 (Sortimente)
YU (2) YU42172B (Sortimente)
ZA (1) ZA79219B (Sortimente)
ZM (1) ZM579A1 (Sortimente)

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NZ199080A (en) * 1980-12-12 1984-07-31 Beecham Group Ltd 2-alkoxy-4-amino-5-alkylsulphonyl-n-(3beta-(8-hydrocarbyl-8-azabicyclo (3,2,1)octyl))benzamides
FR2550447B1 (fr) * 1983-08-10 1986-01-17 Ile De France Application du n-(ally-2-pyrrolidinylmethyl) 2-methoxy 4-amino 5-methylsulfamoyl benzamide comme antiagregant plaquettaire
FR2574795B1 (fr) * 1984-12-18 1987-11-20 Ile De France Nouveau procede industriel de synthese du n-((1'-allyl 2'-pyrrolidinyl) methyl) 2-methoxy 4,5-azimido benzamide
FR2584401B1 (fr) * 1985-07-04 1987-11-20 Ile De France Nouveau benzamide, son procede de preparation et son application dans le domaine therapeutique
US5227388A (en) * 1989-12-26 1993-07-13 Hoechst-Roussel Pharmaceuticals Incorporated Thienobenzoxepins and naphthothiophenes
US5260319A (en) * 1989-12-26 1993-11-09 Hoechst-Roussel Pharmaceuticals Incorporated Thienobenzoxepins and naphthothiophenes
FR2678266A1 (fr) * 1991-06-28 1992-12-31 Delagrange Laboratoires Nouveaux derives de 2-hydroxy 4-amino 5-ethylsulfonyl benzamide utiles comme anxiolytiques.
FR2699533A1 (fr) * 1992-12-21 1994-06-24 Mouhtaram Mohamed Dérivés de N-((1,4-dialkyl-6-arylpipérazine-2-yl)méthyl)benzamides. (Isomères cis et trans) Propriétés pharmacologiques et applications.
FR2753376B1 (fr) * 1996-09-18 1998-10-16 Synthelabo Compositions pharmaceutiques comprenant de l'amisulpride et leurs applications therapeutiques
FR2762213B1 (fr) * 1997-04-18 1999-05-14 Synthelabo Composition pharmaceutique a retention gastrique
US6169094B1 (en) 1998-07-14 2001-01-02 Sanofi-Synthelabo Compositions of (S) (-)-amisulpride
EP1554572B1 (en) 2001-07-25 2009-10-14 Raptor Pharmaceutical Inc. Compositions and methods for modulating blood-brain barrier transport
BRPI0410271A (pt) * 2003-05-16 2006-05-16 Pfizer Prod Inc combinações terapêuticas de antipsicóticos atìpicos com moduladores de gaba, anticonvulsivantes ou benzodiazepinas
FR2857263B1 (fr) * 2003-07-09 2005-09-09 Sanofi Synthelabo Nouvelle composition pharmaceutique solide comprenant de l'amisulpride
WO2005107808A2 (en) * 2004-05-11 2005-11-17 Pfizer Products Inc. Combination of atypical antipsychotics and 5-ht1b receptor antagonists
PE20061318A1 (es) * 2005-04-22 2006-12-28 Wyeth Corp Nuevas combinaciones terapeuticas para el tratamiento o la prevencion de trastornos psicoticos
CN102379684B (zh) 2005-04-28 2014-11-19 普罗透斯数字保健公司 药物信息系统
CN101594878A (zh) 2006-09-18 2009-12-02 雷普特药品公司 通过给予受体相关蛋白（rap）-缀合物对肝病症的治疗
US7825156B2 (en) * 2007-02-02 2010-11-02 Copharms Method of treating bipolar depression with a benzamide derivative
WO2009156889A1 (en) * 2008-06-25 2009-12-30 Pfizer Inc. Diaryl compounds and uses thereof
US20100105755A1 (en) * 2008-09-12 2010-04-29 Auspex Pharmaceuticals, Inc. Substituted benzamide modulators of dopamine receptor
NZ616673A (en) 2009-02-20 2014-08-29 To Bbb Holding B V Glutathione-based drug delivery system
CN110075069A (zh) 2009-05-06 2019-08-02 实验室护肤股份有限公司 包含活性剂-磷酸钙颗粒复合物的皮肤递送组合物及其应用
CN101898991B (zh) * 2009-05-31 2013-09-25 江苏天士力帝益药业有限公司 一种(s)(-)-氨磺必利d-(-)-酒石酸盐的合成方法
CN101628886B (zh) * 2009-08-25 2012-12-12 北京紫萌同达科技有限公司 一种2-甲氧基-4-氨基-5-乙砜基苯甲酸的合成方法
AU2014202535B2 (en) * 2010-03-11 2016-05-26 Acacia Pharma Limited The use of amisulpride as an anti-emetic
AU2016216578B2 (en) * 2010-03-11 2017-11-23 Acacia Pharma Limited The use of amisulpride as an anti-emetic
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CN103450058B (zh) * 2013-09-18 2015-10-14 广安凯特医药化工有限公司 一种氨磺必利酸的制备方法
CN104725292B (zh) * 2015-03-23 2017-07-25 湖北荆江源制药股份有限公司 一种(s)(‑)‑氨磺必利的制备方法
GB201618425D0 (en) * 2016-11-01 2016-12-14 Acacia Pharma Ltd method
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US11377421B2 (en) 2016-11-28 2022-07-05 Lb Pharmaceuticals Inc. Psychotropic agents and uses thereof
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GB201702250D0 (en) 2017-02-10 2017-03-29 Acacia Pharma Ltd Method
CN112236138B (zh) 2017-12-05 2024-05-31 赛诺维信制药公司 晶体形式及其制备方法
JP7268026B2 (ja) 2017-12-05 2023-05-02 サノビオン ファーマシューティカルズ インク 非ラセミ混合物およびその使用
CN110790693A (zh) * 2018-08-02 2020-02-14 北京万全德众医药生物技术有限公司 一种(s)(-)-氨磺必利的制备方法
EP3980009A4 (en) 2019-06-04 2023-07-05 Sunovion Pharmaceuticals Inc. MODIFIED RELEASE FORMULATIONS AND ASSOCIATED USES
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CN116003304A (zh) * 2023-02-08 2023-04-25 浙江皓华制药有限公司 一种氨磺必利的合成方法

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US3342826A (en) * 1964-01-13 1967-09-19 Ile De France Heterocyclic aminoalkyl benzamides
FR2313935A1 (fr) * 1975-06-10 1977-01-07 Ile De France Nouveaux benzamides substitues, leurs derives et leur procede de preparation
US3862139A (en) * 1972-06-23 1975-01-21 Delmar Chem Heterocyclic benzamide compounds
FR2244760B1 (Sortimente) * 1973-09-25 1980-06-27 Ile De France
FR2299862B1 (en) * 1975-02-07 1978-07-21 Soc Et Scient Et Ind Substd. N-(1-benzylpyrrolidinyl-2-alkyl)benzamides - used as antiemetics, anti-ulcer agents and CNS active
FR2294698A1 (fr) * 1974-12-18 1976-07-16 Synthelabo Nouveaux derives des methoxy-2 benzamides substitues, leurs sels, leur preparation et les medicaments qui en renferment
CA1039731A (en) * 1974-12-18 1978-10-03 Synthelabo Process for preparing new 2-methoxy-benzamide derivatives

Also Published As

Publication number Publication date
SE8603773D0 (sv) 1986-09-09
IE47798B1 (en) 1984-06-27
MX5793E (es) 1984-07-19
IL56411A (en) 1982-09-30
YU25483A (en) 1983-10-31
DK20979A (da) 1979-07-21
DE2901181C2 (de) 1984-07-19
PL212899A1 (Sortimente) 1980-01-14
LU80786A1 (fr) 1979-09-07
IL56411A0 (en) 1979-03-12
CY1201A (en) 1983-12-31
YU5079A (en) 1983-06-30
NL7900457A (nl) 1979-07-24
PL118151B1 (en) 1981-09-30
DD141520A5 (de) 1980-05-07
NO790180L (no) 1979-07-23
AU4337379A (en) 1979-07-26
PL116532B1 (en) 1981-06-30
AR220574A1 (es) 1980-11-14
SU820659A3 (ru) 1981-04-07
NZ189378A (en) 1983-03-15
RO76393A (ro) 1981-03-30
PH22287A (en) 1988-07-22
GR64431B (en) 1980-03-21
RO80311A (ro) 1982-12-06
AR221354A1 (es) 1981-01-30
IE790092L (en) 1979-07-20
NO151320C (no) 1985-04-17
FR2415099A1 (fr) 1979-08-17
SE460968B (sv) 1989-12-11
AT377977B (de) 1985-05-28
IT1164655B (it) 1987-04-15
BG31497A3 (bg) 1982-01-15
YU42172B (en) 1988-06-30
IT7947706A0 (it) 1979-01-18
GB2012765A (en) 1979-08-01
MX7623E (es) 1990-03-27
CS226181B2 (en) 1984-03-19
NL191707C (nl) 1996-04-02
US4294828A (en) 1981-10-13
IN150226B (Sortimente) 1982-08-21
FI71126C (fi) 1986-11-24
NL191707B (nl) 1995-12-01
ZM579A1 (en) 1979-12-21
OA06156A (fr) 1981-06-30
SE448874B (sv) 1987-03-23
AU528561B2 (en) 1983-05-05
SE8603773L (sv) 1986-09-09
FI71126B (fi) 1986-08-14
CH637927A5 (fr) 1983-08-31
YU41278B (en) 1986-12-31
BG31496A3 (bg) 1982-01-15
JPS54145658A (en) 1979-11-14
ES477782A1 (es) 1979-09-16
GB2083458A (en) 1982-03-24
GB2012765B (en) 1982-09-08
FI790182A7 (fi) 1979-07-21
BE872585A (fr) 1979-06-07
PH15725A (en) 1983-03-18
EG14045A (en) 1983-09-30
DK158346B (da) 1990-05-07
CA1101430A (en) 1981-05-19
HU179793B (en) 1982-12-28
NO151320B (no) 1984-12-10
JPS6049192B2 (ja) 1985-10-31
FR2415099B1 (Sortimente) 1981-02-20
ZA79219B (en) 1980-01-30
PT69068A (fr) 1979-02-01
HK12184A (en) 1984-02-24
US4401822A (en) 1983-08-30
GB2083458B (en) 1983-03-09
DE2901181A1 (de) 1979-07-26
SE7900380L (sv) 1979-07-21
ATA39879A (de) 1983-12-15
ES476755A1 (es) 1979-06-01
MC1232A1 (fr) 1979-10-26

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