DK157860C - Analogifremgangsmaade til fremstilling af benzylimidazolderivater samt farmaceutisk acceptable syreadditionssalte deraf - Google Patents

Analogifremgangsmaade til fremstilling af benzylimidazolderivater samt farmaceutisk acceptable syreadditionssalte deraf

Info

Publication number
DK157860C
DK157860C DK239980A DK239980A DK157860C DK 157860 C DK157860 C DK 157860C DK 239980 A DK239980 A DK 239980A DK 239980 A DK239980 A DK 239980A DK 157860 C DK157860 C DK 157860C
Authority
DK
Denmark
Prior art keywords
benzylimidazold
analogue
derivatives
preparation
acid addition
Prior art date
Application number
DK239980A
Other languages
Danish (da)
English (en)
Other versions
DK157860B (da
DK239980A (da
Inventor
Masaru Ogata
Katsuya Tawara
Yoshihachi Watanabe
Hiroshi Matsumoto
Toshio Takahashi
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP54071953A external-priority patent/JPS6011904B2/ja
Priority claimed from JP11546579A external-priority patent/JPS5639073A/ja
Application filed by Shionogi & Co filed Critical Shionogi & Co
Publication of DK239980A publication Critical patent/DK239980A/da
Publication of DK157860B publication Critical patent/DK157860B/da
Application granted granted Critical
Publication of DK157860C publication Critical patent/DK157860C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/501,3-Diazoles; Hydrogenated 1,3-diazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C53/00Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen
    • C07C53/08Acetic acid
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C55/00Saturated compounds having more than one carboxyl group bound to acyclic carbon atoms
    • C07C55/02Dicarboxylic acids
    • C07C55/06Oxalic acid
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C55/00Saturated compounds having more than one carboxyl group bound to acyclic carbon atoms
    • C07C55/02Dicarboxylic acids
    • C07C55/10Succinic acid
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/235Saturated compounds containing more than one carboxyl group
    • C07C59/245Saturated compounds containing more than one carboxyl group containing hydroxy or O-metal groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/235Saturated compounds containing more than one carboxyl group
    • C07C59/245Saturated compounds containing more than one carboxyl group containing hydroxy or O-metal groups
    • C07C59/255Tartaric acid
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/235Saturated compounds containing more than one carboxyl group
    • C07C59/245Saturated compounds containing more than one carboxyl group containing hydroxy or O-metal groups
    • C07C59/265Citric acid
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C65/00Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C65/01Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing hydroxy or O-metal groups
    • C07C65/03Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing hydroxy or O-metal groups monocyclic and having all hydroxy or O-metal groups bound to the ring
    • C07C65/05Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing hydroxy or O-metal groups monocyclic and having all hydroxy or O-metal groups bound to the ring o-Hydroxy carboxylic acids
    • C07C65/10Salicylic acid
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
DK239980A 1979-06-07 1980-06-03 Analogifremgangsmaade til fremstilling af benzylimidazolderivater samt farmaceutisk acceptable syreadditionssalte deraf DK157860C (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP7195379 1979-06-07
JP54071953A JPS6011904B2 (ja) 1979-06-07 1979-06-07 1−ベンジルイミダゾ−ル誘導体
JP11546579A JPS5639073A (en) 1979-09-07 1979-09-07 1- alpha-styryl imidazole
JP11546579 1979-09-07

Publications (3)

Publication Number Publication Date
DK239980A DK239980A (da) 1980-12-08
DK157860B DK157860B (da) 1990-02-26
DK157860C true DK157860C (da) 1990-07-30

Family

ID=26413076

Family Applications (1)

Application Number Title Priority Date Filing Date
DK239980A DK157860C (da) 1979-06-07 1980-06-03 Analogifremgangsmaade til fremstilling af benzylimidazolderivater samt farmaceutisk acceptable syreadditionssalte deraf

Country Status (15)

Country Link
US (3) US4328348A (nl)
AR (2) AR226847A1 (nl)
CA (1) CA1141388A (nl)
CH (1) CH646693A5 (nl)
DE (1) DE3021467A1 (nl)
DK (1) DK157860C (nl)
FR (1) FR2458545B1 (nl)
GB (2) GB2054560B (nl)
HU (1) HU188607B (nl)
IE (1) IE49604B1 (nl)
IL (1) IL60252A (nl)
IT (1) IT1129813B (nl)
MX (1) MX5880E (nl)
NL (1) NL184003C (nl)
SE (1) SE453991B (nl)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5216007A (en) * 1980-10-01 1993-06-01 Rohm And Haas Company Substituted ethylene imidazole and triazoles
JPS6036427B2 (ja) * 1980-12-05 1985-08-20 塩野義製薬株式会社 1−ベンジルイミダゾ−ル誘導体
DK162882A (da) * 1981-04-13 1982-10-14 Searle & Co Imidazolderivater eller syreadditionssalte deraf,deres fremstilling og anvendelse
JPS57188570A (en) * 1981-05-14 1982-11-19 Shionogi & Co Ltd Benzylazole derivative
GB2126218B (en) * 1982-08-14 1986-01-22 Wellcome Found Imidazoles
US4579862A (en) * 1983-07-05 1986-04-01 G. D. Searle & Co. Certain 1H-imidazol-1-yl-1-lower-alkanoic acid derivatives having anti-thrombotic activity
JPS60155163A (ja) * 1984-01-09 1985-08-15 Mitsui Toatsu Chem Inc イミダゾ−ル誘導体
US5135943A (en) * 1984-02-02 1992-08-04 Ferrer Internacional S.A. 1H-imidazole derivative compounds and pharmaceutical compositions containing the same
US4629795A (en) * 1984-05-25 1986-12-16 Shionogi & Co., Ltd. Process for preparing imidazole derivatives
US4755526A (en) * 1984-06-18 1988-07-05 Eli Lilly And Company Method of inhibiting aromatase
JPS62149666A (ja) * 1985-12-25 1987-07-03 Shionogi & Co Ltd N−ビニルアゾ−ル類
US4937250A (en) * 1988-03-07 1990-06-26 Ciba-Geigy Corporation Alpha-heterocycle substituted tolunitriles
US4978672A (en) * 1986-03-07 1990-12-18 Ciba-Geigy Corporation Alpha-heterocyclc substituted tolunitriles
US4749713A (en) * 1986-03-07 1988-06-07 Ciba-Geigy Corporation Alpha-heterocycle substituted tolunitriles
JPH064598B2 (ja) * 1986-07-01 1994-01-19 塩野義製薬株式会社 アゾ−ル誘導体、およびそれを含有する植物病害防除剤
US5138069A (en) * 1986-07-11 1992-08-11 E. I. Du Pont De Nemours And Company Angiotensin II receptor blocking imidazoles
IL86134A (en) * 1987-05-02 1993-06-10 Basf Ag N-substituted azoles, their manufacture and their use as pesticides and compositions containing them
DE3812483A1 (de) * 1987-06-27 1989-01-05 Bayer Ag (azolyl-vinyl)-phenol-alkenylether
US4880804A (en) * 1988-01-07 1989-11-14 E. I. Du Pont De Nemours And Company Angiotensin II receptor blocking benzimidazoles
US5210079A (en) * 1988-01-07 1993-05-11 E. I. Du Pont De Nemours And Company Treatment of chronic renal failure with imidazole angiotensin-II receptor antagonists
DE3811574A1 (de) * 1988-03-31 1989-10-19 Schering Ag N-substituierte imidazole, verfahren zu ihrer herstellung sowie ihre verwendung in arzneimitteln
US5354867A (en) * 1988-12-06 1994-10-11 E. I. Du Pont De Nemours And Company Angiotensin II receptor blocking imidazoles
CA2006309C (fr) * 1988-12-29 2001-12-18 Jean Hutt Azolylmethylcyclopentane benzylidene fongicide
US5256683A (en) * 1988-12-29 1993-10-26 Rhone-Poulenc Agrochimie Fungicidal compositions containing (benzylidene)-azolylmethylcycloalkane
DE3901723A1 (de) 1989-01-21 1990-07-26 Bayer Ag Azolyl-derivate
KR950009860B1 (ko) * 1989-06-30 1995-08-29 이. 아이. 듀퐁 드 네모아 앤드 캄파니 융합된 환 아릴 치환된 이미다졸과 약제학적으로 허용되는 이의 염, 이들의 제조방법 및 이들을 함유하는 약제학적 조성물
JPH03130266A (ja) * 1989-07-28 1991-06-04 Hodogaya Chem Co Ltd 置換フェニルアルキルイミダゾール誘導体
US5466704A (en) * 1991-02-26 1995-11-14 E. R. Squibb & Sons, Inc. N-substituted imidazole and benzimidazole derivatives useful as angiotenson II antagonists
EP0757988A4 (en) * 1994-04-27 2000-07-26 Nippon Soda Co IMIDAZOLE DERIVATIVE AND PROCESS FOR PRODUCING THE SAME
US6436395B1 (en) 1996-09-18 2002-08-20 Merck & Co., Inc. Rosellinia subiculata ATCC 74386 and fungus ATCC 74387 for producing sordarin compounds for fungi control
ATE332292T1 (de) * 2003-04-16 2006-07-15 Huntsman Adv Mat Switzerland 1-imidazolylmethyl-substituirte-2-naphtol unh ihre verwendung als niedertemperatur- härtungsbeschleuniger
GB0526252D0 (en) * 2005-12-22 2006-02-01 Novartis Ag Organic compounds

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1806995C3 (de) * 1968-11-05 1978-09-28 Bayer Ag, 5090 Leverkusen Bisimidazolyl-bisphenylmethane und deren Salze
BR6915465D0 (pt) * 1969-03-07 1973-01-04 Bayer Ag Processo para preparar n-benzimidazois substituidos na posicao alfa por heterociclos penta-membrados com atividade antimicotica
IE40911B1 (en) * 1974-04-11 1979-09-12 Schering Ag Imidazole derivatives and process for their manufacture
GR70061B (nl) * 1977-03-31 1982-07-26 Nippon Soda Co
DE2862340D1 (en) * 1978-02-01 1983-11-24 Wellcome Found Imidazole derivatives and salts thereof, their synthesis, and pharmaceutical formulations thereof
DE2808086A1 (de) * 1978-02-24 1979-08-30 Bayer Ag Substituierte diphenyl-imidazolyl- methane, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel
JPS55313A (en) * 1978-06-13 1980-01-05 Kissei Pharmaceut Co Ltd Imidazole derivative
DK531479A (da) * 1979-01-19 1980-07-20 Pfizer Fremgangsmaade til fremstilling af imidazolderivater og salte deraf

Also Published As

Publication number Publication date
GB2054560B (en) 1983-09-01
IL60252A (en) 1987-02-27
NL184003C (nl) 1989-03-16
HU188607B (en) 1986-04-28
DK157860B (da) 1990-02-26
IT1129813B (it) 1986-06-11
FR2458545A1 (fr) 1981-01-02
SE453991B (sv) 1988-03-21
US4328348A (en) 1982-05-04
GB2054560A (en) 1981-02-18
GB2118549A (en) 1983-11-02
US4483866A (en) 1984-11-20
IL60252A0 (en) 1980-09-16
IT8067889A0 (it) 1980-06-06
AR226847A1 (es) 1982-08-31
US4463011A (en) 1984-07-31
DE3021467C2 (nl) 1989-11-02
CH646693A5 (de) 1984-12-14
DE3021467A1 (de) 1980-12-18
SE8004194L (sv) 1980-12-08
CA1141388A (en) 1983-02-15
GB2118549B (en) 1984-04-11
MX5880E (es) 1984-08-16
NL8003310A (nl) 1980-12-09
AR230184A1 (es) 1984-03-01
IE801159L (en) 1980-12-07
IE49604B1 (en) 1985-10-30
FR2458545B1 (fr) 1986-04-18
NL184003B (nl) 1988-10-17
DK239980A (da) 1980-12-08

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